Zobrazeno 1 - 9 of 9 pro vyhledávání: '"Vijay J, Medhane"'
1
Akademický článek
Investigation of Mechanistic Pathway for Trimethyl borate mediated Amidation of (R)-Mandelic Acid for the Synthesis of Mirabegron, an Antimuscarinic Agent
Autor: Vijayavitthal Thippannachar Mathad, Dattatray G. Deshmukh, Mukund N. Bangal, Mukunda R. Patekar, Vijay J. Medhane
Publikováno v: Acta Chimica Slovenica, Vol 65, Iss 1, Pp 239-245 (2018)
The present work describes investigation of mechanistic pathway for trimethyl borate mediated amidation of (R)-mandelic acid (3) with 4-nitophenylethylamine (2) to provide (R)-2-hydroxy-N-[2-(4-nitrophenyl)ethyl]-2-phenylacetamide (4) during mirabegr
Externí odkaz: https://doaj.org/article/6c90b873f4c445cbab1c2a2a72db7038
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3
Akademický článek
First Direct Isolation of Stable α-Form Crystals of Mirabegron, a Selective β3–Adrenoceptor Agonist
Autor: Vijayavitthal T. Mathad, Dattatray G. Deshmukh, Mukund N. Bangal, Anil C. Mali, Vijay J. Medhane
Publikováno v: Acta Chimica Slovenica, Vol 64, Iss 2, Pp 461-466 (2017)
An efficient and scalable method for the direct isolation of stable α-form crystals of mirabegron (1) is developed. The developed method negates transformation of metastable β-form crystals into α-form crystals thereby overcome the limitations of
Externí odkaz: https://doaj.org/article/e3e3214f5ae5454e930d62e7039ed542
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4
Synthesis of Novel Oxazolidinone Derivatives Bearing Benzo[b]thiophene Moiety and their Antimicrobial Evaluation
Autor: Mukunda R. Patekar, Ghanshyam R. Jadhav, Dattatray G. Deshmukh, Vijay J. Medhane
Publikováno v: Asian Journal of Chemistry. 34:1197-1205
Literature survey revealed that the oxazolidinone derivatives exhibit pharmacological significance. Thus, by targeting to design new antimicrobial agent, a novel series of oxazolidinone derivatives (11a-t) having benzo[b]thiophene moiety were synthes
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::c56057bb380192acc7b2d60e0b8f1704
https://doi.org/10.14233/ajchem.2022.23633
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5
Efficient Synthesis of Novel Thiazole Substituted Pyrrolidine Derivatives and their Antimicrobial Evaluation
Autor: Ghanshyam R. Jadhav, Avinash D. Bholay, Mahendra B. Bodake, Vijay J. Medhane
Publikováno v: Asian Journal of Chemistry. 32:2007-2012
A series of new molecules containing pyrrolidine and thiazole moiety (4a-l) were designed and synthesized. The structures of the synthesized compounds were characterized by IR, 1H NMR and mass spectral data. All the synthesized compounds were screene
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::976e4036083bdb871d06429965955b9a
https://doi.org/10.14233/ajchem.2020.22772
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6
2,5-Disubstituted 1,3,4-oxadiazole derivatives of chromeno[4,3-b]pyridine: synthesis and study of antimicrobial potency
Autor: Avinash D. Bholay, Ghanshyam R. Jadhav, Dattatray G. Deshmukh, Vijay J. Medhane, Vishwas B. Gaikwad
Publikováno v: Heterocyclic Communications. 22:123-130
A convenient synthesis of 1,3,4-oxadiazole containing derivatives of chromeno[4,3-b]pyridine (6a–e, 8a–e and 9a–e) starting from 4-hydroxycoumarin is presented. The synthesized compounds were screened for in vitro antimicrobial activity against
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::2a73ffead201a802c15e0c0df222b58e
https://doi.org/10.1515/hc-2015-0215
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7
Investigation of Mechanistic Pathway for Trimethyl Borate Mediated Amidation of (R)-Mandelic Acid for the Synthesis of Mirabegron, an Antimuscarinic Agent
Autor: Dattatray G, Deshmukh, Mukund N, Bangal, Mukunda R, Patekar, Vijay J, Medhane, Vijayavitthal Thippannachar, Mathad
Publikováno v: Acta chimica Slovenica. 65(1)
The present work describes investigation of mechanistic pathway for trimethyl borate mediated amidation of (R)-mandelic acid (3) with 4-nitophenylethylamine (2) to provide (R)-2-hydroxy-N-[2-(4-nitrophenyl)ethyl]-2-phenylacetamide (4) during mirabegr
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::e4236e660f92a6f9b4a915b880a5b6ef
https://pubmed.ncbi.nlm.nih.gov/29562093
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9
Facile approach for the synthesis of rivaroxaban using alternate synthon: reaction, crystallization and isolation in single pot to achieve desired yield, quality and crystal form
Autor: Anil C. Mali, Vijay J. Medhane, Priyank I Patel, Hitesh D Lad, Dattatray G. Deshmukh, Divyesh R. Joshi, Vijayavitthal T. Mathad
Publikováno v: Sustainable Chemical Processes. 3(1)
An efficient and high yielding process for the production of impurity free rivaroxaban (1), an anti-coagulant agent using alternate synthon is reported. The key components of the process involve; synthesis of 4-(4-aminophenyl)-3-morpholinone (5) usin
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7622325127ec20928cb75c2a348b5835
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