Zobrazeno 1 - 10
of 31
pro vyhledávání: '"Vera Klimesova"'
Autor:
Vera Klimesova, Petra Herzigová, Karel Palát, Miloš Macháček, Jiřina Stolaříková, Hans Martin Dahse, Ute Möllmann
Publikováno v:
ARKIVOC, Vol 2012, Iss 3, Pp 90-103 (2012)
Externí odkaz:
https://doaj.org/article/4d612f14f0044a81b9181082900c53d7
Autor:
Ilkay Yildiz, Karel Nesměrák, Ismail Yalcin, Marketa Brozikova, Karel Waisser, Alla P. Toropova, Andrey A. Toropov, Vera Klimesova
Publikováno v:
Analytical and Bioanalytical Chemistry. 407:9185-9189
The CORAL software ( http://www.insilico.eu/coral ) was used to build up quantitative structure-property relationships (QSPRs) for the retention characteristics of 93 derivatives of three groups of heterocyclic compounds: 2-phenyl-1,3-benzoxazoles, 4
Autor:
Gunther Buehrdel, Helmar Goerls, Rainer Beckert, Petra Herzigova, Eva Petrlikova, Jan Fleischhauer, Vera Klimesova
Publikováno v:
Synthesis. 2008:3071-3080
A short and efficient synthesis for a series of 1,6-diaryl- 3,4-diarylaminohexa-2,4-diene-1,6-diones was developed. Based on the acylation-prototropism sequence during the reaction of vari- ous aryl methyl ketones with bis-imidoyl chlorides, the prod
Autor:
Josef Matyk, Jarmila Kaustová, Petra Husáková, Hana Divišová, Karel Waisser, Jiri Kunes, Vera Klimesova, Karel Palát
Publikováno v:
Archiv der Pharmazie. 340:264-267
Based on our previous studies, 21 new halogenated 3-(4-alkylphenyl)-1,3-benzoxazine-2,4-(3H)-diones were synthesized by the reaction of salicylanilides and methyl-chloroformate. All compounds were screened in vitro against three different strains of
Publikováno v:
Il Farmaco. 59:615-625
The series of derivatives of substituted N-pyridinylsalicylamides were synthesized. The compounds were evaluated for in vitro antimycobacterial activity against Mycobacterium avium and two strains of Mycobacterium kansasii. In the quantitative struct
Publikováno v:
Journal of Liquid Chromatography & Related Technologies. 25:2849-2856
Lipophilicity is one of the properties which influence the partition of a substance in biological media. The reversed-phase high-performance liquid chromatographic (RP-HPLC) capacity factors k of two series of 2-benzylthioderivatives, newly synthesiz
Publikováno v:
Il Farmaco. 57:259-265
A set of 2-alkylsulfanyl derivatives of 5-methylbenzimidazole was synthesized and evaluated for antimycobacterial activity. The structures of the compounds were confirmed by 1H NMR and IR data, and their purity by elemental analysis. Antimycobacteria
Autor:
Hynek Dostál, Lenka Kubicová, Jiøı́ Kuneš, Jiří Gregor, Karel Waisser, Vera Klimesova, Jarmila Kaustová
Publikováno v:
Il Farmaco. 56:803-807
Series of 3-phenyl-6,8-dichloro-2H-1,3-benzoxazine-2,4(3H)-dithiones, 3-arylquinazoline-2,4(1H,3H)-diones and 3-arylquinazoline-2,4(1H,3H)-dithiones were synthesized, and the antimycobacterial activities of the derivatives evaluated in vitro. The com
Autor:
Jarmila Kaustová, Jiri Kunes, Vera Klimesova, Lenka Kubicová, Karel Waisser, Miloš Macháček, Jiří Gregor
Publikováno v:
European Journal of Medicinal Chemistry. 35:733-741
A series of 6-chloro-3-phenyl-4-thioxo-2H-1,3-benzoxazine-2(3H)-ones 3 and a series of 6-chloro-3-phenyl-2H-1,3-benzoxazine-2,4(3H)-dithiones 4 were synthesized by melting 6-chloro-3-phenyl-2H-1,3-benzoxazine-2,4(3H)-dione and its derivatives substit
Publikováno v:
Il Farmaco. 54:666-672
A set of pyridine derivatives bearing a substituted alkylthio chain or a piperidyl ring in position 2 or 4 were synthesized, and their antimycobacterial and antifugal activities were evaluated. Chemical structures were confirmed by IR and NMR data, a