Zobrazeno 1 - 10
of 27
pro vyhledávání: '"Venkata Madhavi, Yaddanapudi"'
Autor:
Shaik Mahammad Ghouse, Kavyaraj Bahatam, Andrea Angeli, Gaurav Pawar, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Arifuddin Mohammed, Claudiu T. Supuran, Srinivas Nanduri
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)
The Carbonic anhydrase isoforms IX and XII play a significant role in regulating the intracellular and extracellular pH in hypoxic tumours abetting the metastasis of solid tumours. Selective and potent inhibitors targeting carbonic anhydrase IX and X
Externí odkaz:
https://doaj.org/article/a0d393337b584c69bfede9d13cb105d8
Autor:
Mohammed Arifuddin, Claudiu T. Supuran, Srinivas Nanduri, Krishna Kartheek Chinchilli, Priti Singh, Baijayantimala Swain, Nerella Sridhar Goud, Dilep Kumar Sigalapalli, Abhishek Choli, Andrea Angeli, Venkata Madhavi Yaddanapudi
Publikováno v:
Anti-Cancer Agents in Medicinal Chemistry. 23:1225-1233
Background: Carbonic anhydrases (CAs, EC 4.2.1.1) catalyze the reversible hydration of carbon dioxide to bicarbonate and a proton. Inhibition of isoforms IX and XII has induced potent anticancer effects. Objective: A series of indole-3-sulfonamide-he
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::73a09c6e8824cb7080a648f840592128
https://doi.org/10.2174/1871520623666230227092821
https://doi.org/10.2174/1871520623666230227092821
Autor:
Baijayantimala Swain, Abrar Khan, Priti Singh, Vaibhav S. Marde, Andrea Angeli, Krishna Kartheek Chinchilli, Venkata Madhavi Yaddanapudi, Simone Carradori, Claudiu T. Supuran, Mohammed Arifuddin
Publikováno v:
Molecules, Vol 27, Iss 22, p 8028 (2022)
A novel series of twenty-five rhodamine-linked benzenesulfonamide derivatives (7a–u and 9a–d) were synthesized and screened for their inhibitory action against four physiologically relevant human (h) carbonic anhydrase (CA) isoforms, namely hCA I
Externí odkaz:
https://doaj.org/article/a422a55ee080449dab1df6c758b9bb1d
Autor:
Gaurav Pawar, Shaik Mahammad Ghouse, Swanand Vinayak Joshi, Md Naiyaz Ahmad, Arunava Dasgupta, Venkata Madhavi Yaddanapudi, Siddharth Chopra, Srinivas Nanduri
Publikováno v:
New Journal of Chemistry. 47:5961-5969
One-pot tandem synthesis of diverse pyrido[2′,1′:2,3]imidazo[4,5-c]quinolines as new antimycobacterial agents through a Cu(i)-catalyzed microwave-assisted protocol.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::231cb4fa319caac661f8304b4315008a
https://doi.org/10.1039/d2nj06165a
https://doi.org/10.1039/d2nj06165a
Autor:
Ramulu Parupalli, Ravikumar Akunuri, Grace Kaul, Abdul Akhir, Deepanshi Saxena, Shaik Mahammad Ghouse, Venkata Madhavi Yaddanapudi, Sidharth Chopra, Srinivas Nanduri
Publikováno v:
Future Medicinal Chemistry. 14:1621-1634
Background: In the authors' previous study, 4-(2-((3-methyl-4-oxo-2-thioxo/dioxothiazolidin-5-ylidene) methyl) hydrazineyl) benzonitriles were found to demonstrate potent antibacterial activity against Acinetobacter baumannii. Interestingly, the afor
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4db725b7ac9b6518f60b46dd7fe00305
https://doi.org/10.4155/fmc-2022-0156
https://doi.org/10.4155/fmc-2022-0156
Autor:
Mohammed Arifuddin, Claudiu T. Supuran, Venkata Madhavi Yaddanapudi, Baijayantimala Swain, Priti Singh, Andrea Angeli, Santosh Kumar Sahoo
Publikováno v:
Anti-Cancer Agents in Medicinal Chemistry. 22:2358-2366
Background: A high yielding green protocol has been developed and delineated for the synthesis of 3,3- di(indolyl)indolin-2-ones, potentially bioactive compounds, involving one pot aqueous medium condensation of isatin with indole in the presence of
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::457bd76743ee26ed3f1db099f9c908ee
https://doi.org/10.2174/1871520622666220202112014
https://doi.org/10.2174/1871520622666220202112014
Autor:
Santosh Kumar Sahoo, Mohammad Naiyaz Ahmad, Grace Kaul, Srinivas Nanduri, Arunava Dasgupta, Sidharth Chopra, Venkata Madhavi Yaddanapudi
Publikováno v:
RSC Med Chem
With growing concerns regarding target residue mutation hovering over established anti-TB pharmacophores, it is imperative to have reserve chemotypes at our disposal to curb unrestrained spread of tuberculosis. In this context, we herein present the
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::97ba592e0c5a5bdfae27c33dc6f20b3a
https://doi.org/10.1039/d1md00387a
https://doi.org/10.1039/d1md00387a
Autor:
Venkata Madhavi Yaddanapudi, Ojaswitha Ommi, Mohammed Naiyaz Ahmad, Siva Nageswara Rao Gajula, Parita Wanjari, Shashikanta Sahu, Puja Kumari Agnivesh, Santosh Kumar Sahoo, Nitin Pal Kalia, Rajesh Sonti, Srinivas Nanduri, Arunava Dasgupta, Sidharth Chopra
Publikováno v:
RSC Medicinal Chemistry.
The urgent development of newer alternatives has been deemed a panacea for tackling emerging antimicrobial resistance effectively. Herein, we report the design, synthesis, and biological evaluation of 1,3-diaryl substituted pyrazole-based...
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::aaa7868770e34fd93f57388e380a15e9
https://doi.org/10.1039/d3md00079f
https://doi.org/10.1039/d3md00079f
Autor:
Santosh Kumar Sahoo, Ojaswitha Ommi, Sarvan Maddipatla, Priti Singh, Mohammad Naiyaz Ahmad, Grace Kaul, Srinivas Nanduri, Arunava Dasgupta, Sidharth Chopra, Venkata Madhavi Yaddanapudi
Publikováno v:
Molecular Diversity.
In our continued efforts to find potential chemotherapeutics active against drug-resistant (DR) Mycobacterium tuberculosis (Mtb), causative agent of Tuberculosis (TB) and to curb the current burdensome treatment regimen, herein we describe the synthe
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c1f33d504964a38c74c3ff3d0e5a4eda
https://doi.org/10.1007/s11030-022-10543-0
https://doi.org/10.1007/s11030-022-10543-0
Autor:
Nikhil Baliram Gaikwad, Santosh Kumar Sahoo, Ojaswitha Ommi, Mohammad Naiyaz Ahmad, Afroz Pathan, Grace Kaul, Srinivas Nanduri, Arunava Dasgupta, Sidharth Chopra, Venkata Madhavi Yaddanapudi
Publikováno v:
ChemistrySelect. 7
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f58cfe4ebf33f65d49f3a87222760f22
https://doi.org/10.1002/slct.202203333
https://doi.org/10.1002/slct.202203333