Zobrazeno 1 - 10
of 12
pro vyhledávání: '"Varadaraj G Bhat"'
Autor:
Krishnaraj Somyaji Shirur, Bharath Singh Padya, Abhijeet Pandey, Manasa Manjunath Hegde, Aparna I. Narayan, Bola Sadashiva Satish Rao, Varadaraj G. Bhat, Srinivas Mutalik
Publikováno v:
Nanomaterials, Vol 12, Iss 19, p 3372 (2022)
Microorganisms are the major cause for the failure of root canal treatment, due to the penetration ability within the root anatomy. However, irrigation regimens have at times failed due to the biofilm mode of bacterial growth. Liposomes are vesicular
Externí odkaz:
https://doaj.org/article/624a6dc7426e45f8a4d3b50905b12a82
Publikováno v:
RESEARCH JOURNAL OF PHARMACY AND TECHNOLOGY. 13:5806-5810
An antifungal agent is a drug that eliminates fungal pathogens selectively from host with negligible toxicity to the host. Antifungal agents are classified into classes like antibiotics, antimetabolite, azole, and allyl amine. In this present work, t
Autor:
Gautham G. Shenoy, Helena I. Boshoff, Indira Bairy, Kriti Arora, Ruchi Verma, Mradul Tiwari, Varadaraj G Bhat
Publikováno v:
Journal of Molecular Structure. 1197:117-133
A new series of novel diphenyl ether based 2-oxo-dihydropyridine derivatives were synthesized and screened for their in vitro antimycobacterial and antibacterial activities. Most of the synthesized compounds showed significant activity against Mycoba
Autor:
Girij Pal Singh, Varadaraj G Bhat, Anurag Trivedi, Himanshu M. Godbole, Gautham G. Shenoy, Bhushan B. Borase, Pritesh R. Upadhyay
Publikováno v:
Journal of Chemical Sciences. 133
Herein, we have described a novel and concise synthesis of the potent angiotensin-converting enzyme (ACE) inhibitor, benazepril hydrochloride (7) in trifluoroethanol via an Ugi three-component reaction in shorter reaction times. The key step is the t
Publikováno v:
Mini reviews in medicinal chemistry. 19(17)
Diphenyl ethers (DPE) and its analogs have exhibited excellent potential for therapeutic and industrial applications. Since the 19th century, intensive research is perpetuating on the synthetic routes and biological properties of DPEs. Few well-known
Autor:
Gautham G. Shenoy, Girij Pal Singh, Pritesh R. Upadhyay, Varadaraj G Bhat, Anurag Trivedi, Himanshu M. Godbole, Bhushan B. Borase
A novel, efficient and concise synthesis of chirally pure quinapril hydrochloride is described. The key step is the formation of α-amino amide backbone in one step using Ugi three component reaction. This method allows short access to α-amino amide
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2833cb79370cc63e5eba6df4346ec926
Publikováno v:
Chemical biologydrug design. 93(1)
In our efforts to develop druggable diphenyl ethers as potential antitubercular agents, a series of novel diphenyl ether derivatives (5a-f, 6a-f) were designed and synthesized. The representative compounds showed promising in vitro activity against d
Autor:
Rajeev K Singla, Pawan G. Nayak, K.S.R. Pai, Piya Paul, Girish R. Bankar, Varadaraj G Bhat, Punit Bansal
Publikováno v:
Journal of Ethnopharmacology. 134:50-54
Ethnopharmacological relevance The fruits of Cocos nucifera Linn. (Arecaceae) have long been used in traditional medicine for the treatment of cardio-metabolic disorders. Aim of the study To evaluate the ethanolic extract of Cocos nucifera Linn. endo
Publikováno v:
Current drug metabolism. 15(4)
The aligned manuscript reports synthesis, screening and QSAR analysis of twenty six 1, 2, 4-triazole analogues from their respective aromatic carboxylic acids. The structures of synthesized analogues were characterized using physical and spectral ana
Autor:
Rajeev K Singla, Varadaraj G Bhat
Publikováno v:
Medical hypotheses. 74(3)