Zobrazeno 1 - 10
of 15
pro vyhledávání: '"Valentina Lucchesi"'
Autor:
Valentina Lucchesi, Lorenzo Grimaldi, Valentina Mastrantonio, Daniele Porretta, Letizia Di Bella, Tania Ruspandini, Martino Luigi Di Salvo, John Vontas, Romeo Bellini, Agata Negri, Sara Epis, Silvia Caccia, Claudio Bandi, Sandra Urbanelli
Publikováno v:
Insects, Vol 13, Iss 12, p 1109 (2022)
Insecticide resistance is a major threat challenging the control of harmful insect species. The study of resistant phenotypes is, therefore, pivotal to understand molecular mechanisms underpinning insecticide resistance and plan effective control and
Externí odkaz:
https://doaj.org/article/f24278bc98ac493fb88ed612bf85ed48
Autor:
Valentina Mastrantonio, Daniele Porretta, Valentina Lucchesi, Nurper Güz, Naciye Sena Çağatay, Romeo Bellini, John Vontas, Sandra Urbanelli
Publikováno v:
Insects, Vol 12, Iss 8, p 676 (2021)
Insecticide resistance is an informative model for studying the appearance of adaptive traits. Simultaneously, understanding how many times resistance mutations originate is essential to design effective resistance management. In the mosquito Culex p
Externí odkaz:
https://doaj.org/article/38c2fe09a63b46d1acd757420b536c10
Autor:
Daniele Porretta, Valentina Mastrantonio, Valentina Lucchesi, Romeo Bellini, John Vontas, Sandra Urbanelli
Publikováno v:
Pest Management Science. 78:1567-1572
Insecticide resistance is the major threat to vector control and for the prevention of vector-borne diseases. Because almost all insecticides used against insect vectors are or have been used in agriculture, a connection between agricultural insectic
Autor:
Piero A. Salvadori, Valentina Lucchesi, Giuseppe Saccomanni, Giancarlo Pascali, Clementina Manera, Simone Zanoni, Elena Sanguinetti, Daniele Panetta, Silvia Burchielli, Mariarosaria De Simone, Patricia Iozzo
Publikováno v:
Australian Journal of Chemistry. 74:443-452
We successfully radiolabelled a novel prospective cannabinoid type 2 receptor ligand with 18F and tested its biodistribution in animal models by positron emission tomography (PET)/computed tomography (CT) imaging. The radiolabelling process was condu
Autor:
Romeo Bellini, Valentina Mastrantonio, Valentina Lucchesi, Sandra Urbanelli, Nurper Guz, Daniele Porretta, Naciye Sena Çağatay, John Vontas
Publikováno v:
Insects, Vol 12, Iss 676, p 676 (2021)
Insects
Volume 12
Issue 8
Insects
Volume 12
Issue 8
Simple Summary The application of insecticides to control insect pests can result in the evolution of resistance. Within a population, the individuals carrying the resistant mutation survive after insecticide application while the others die, leading
Autor:
Clementina Manera, Piero Salvadori, Giancarlo Pascali, Patricia Iozzo, Valentina Lucchesi, Giuseppe Saccomanni, Daniele Panetta, Simone Zanoni, Mariarosaria De Simone, Silvia Burchielli
Publikováno v:
Nuclear Medicine and Biology. :S35
Autor:
Brandie M. Ehrmann, Mary E. Abood, Giuseppe Saccomanni, Haleli Sharir, Marco Macchia, Filippo Minutolo, Simone Bertini, Valentina Lucchesi, Vincenzo Di Marzo, Lyle Lawrence, Patricia H. Reggio, Marco Allarà, Derek M. Shore, Alessia Ligresti, Dow P. Hurst, Clementina Manera
Publikováno v:
Journal of Medicinal Chemistry
Journal of medicinal chemistry (Online) 57 (2014): 8777–91. doi:10.1021/jm500807e
info:cnr-pdr/source/autori:Lucchesi, Valentina; Hurst, Dow P; Shore, Derek M; Bertini, Simone; Ehrmann, Brandie M; Allara, Marco; Lawrence, Lyle; Ligresti, Alessia; Minutolo, Filippo; Saccomanni, Giuseppe; Sharir, Haleli; Macchia, Marco; Di Marzo, Vincenzo; Abood, Mary E; Reggio, Patricia H; Manera, Clementina/titolo:CB2-Selective Cannabinoid Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Modeling Investigation of 1,8-Naphthyridin-2(1H)-one-3-carboxamides./doi:10.1021%2Fjm500807e/rivista:Journal of medicinal chemistry (Online)/anno:2014/pagina_da:8777/pagina_a:91/intervallo_pagine:8777–91/volume:57
Journal of medicinal chemistry (Online) 57 (2014): 8777–91. doi:10.1021/jm500807e
info:cnr-pdr/source/autori:Lucchesi, Valentina; Hurst, Dow P; Shore, Derek M; Bertini, Simone; Ehrmann, Brandie M; Allara, Marco; Lawrence, Lyle; Ligresti, Alessia; Minutolo, Filippo; Saccomanni, Giuseppe; Sharir, Haleli; Macchia, Marco; Di Marzo, Vincenzo; Abood, Mary E; Reggio, Patricia H; Manera, Clementina/titolo:CB2-Selective Cannabinoid Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Modeling Investigation of 1,8-Naphthyridin-2(1H)-one-3-carboxamides./doi:10.1021%2Fjm500807e/rivista:Journal of medicinal chemistry (Online)/anno:2014/pagina_da:8777/pagina_a:91/intervallo_pagine:8777–91/volume:57
We have recently identified 1,8-naphthyridin-2(1H)-one-3-carboxamide as a new scaffold very suitable for the development of new CB2 receptor potent and selective ligands. In this paper we describe a number of additional derivatives in which the same
Autor:
Valentina Lucchesi, Giuseppe Saccomanni, Maurizio Bifulco, Elena Ciaglia, Teija Parkkari, Simone Bertini, Marco Macchia, Chiara Laezza, Patrizia Gazzerro, Paola Nieri, Sara Carpi, Simona Pisanti, Stefano Fogli, Anna Maria Malfitano, Juha R. Savinainen, Vincenzo Di Marzo, Alessia Ligresti, Clementina Manera
Publikováno v:
European journal of medicinal chemistry 97 (2015): 10–18. doi:10.1016/j.ejmech.2015.04.034
info:cnr-pdr/source/autori:Manera C.; Malfitano A.M.; Parkkari T.; Lucchesi V.; Carpi S.; Fogli S.; Bertini S.; Laezza C.; Ligresti A.; Saccomanni G.; Savinainen J.R.; Ciaglia E.; Pisanti S.; Gazzerro P.; Di Marzo V.; Nieri P.; Macchia M.; Bifulco M./titolo:New quinolone-and 1,8-naphthyridine-3-carboxamides as selective CB2 receptor agonists with anticancer and immuno-modulatory activity/doi:10.1016%2Fj.ejmech.2015.04.034/rivista:European journal of medicinal chemistry/anno:2015/pagina_da:10/pagina_a:18/intervallo_pagine:10–18/volume:97
info:cnr-pdr/source/autori:Manera C.; Malfitano A.M.; Parkkari T.; Lucchesi V.; Carpi S.; Fogli S.; Bertini S.; Laezza C.; Ligresti A.; Saccomanni G.; Savinainen J.R.; Ciaglia E.; Pisanti S.; Gazzerro P.; Di Marzo V.; Nieri P.; Macchia M.; Bifulco M./titolo:New quinolone-and 1,8-naphthyridine-3-carboxamides as selective CB2 receptor agonists with anticancer and immuno-modulatory activity/doi:10.1016%2Fj.ejmech.2015.04.034/rivista:European journal of medicinal chemistry/anno:2015/pagina_da:10/pagina_a:18/intervallo_pagine:10–18/volume:97
Several recent studies suggest that selective CB2 receptor agonists may represent a valid pharmacological approach in the treatment of various diseases due to the absence of relevant psychoactive side effect. In this study, we synthesized and tested
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9c450b3bdf68bbc1780fc891b76638e7
http://hdl.handle.net/11568/750832
http://hdl.handle.net/11568/750832
Autor:
Teija Parkkari, Sara Del Carlo, Marco Macchia, Marco Allarà, Alessia Ligresti, Simone Bertini, Clementina Manera, Giuseppe Saccomanni, Juha R. Savinainen, Francesca Castelli, Anna Maria Malfitano, Valentina Lucchesi, Maurizio Bifulco, Chiara Laezza, Vincenzo Di Marzo
Publikováno v:
European journal of medicinal chemistry (Online) (2014).
info:cnr-pdr/source/autori:Lucchesi V, Parkkari T, Savinainen JR, Malfitano AM, Allarà M, Bertini S, Castelli F, Del Carlo S, Laezza C, Ligresti A, Saccomanni G, Bifulco M, Di Marzo V, Macchia M, Manera C./titolo:1,2-Dihydro-2-oxopyridine-3-carboxamides: the C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor./doi:/rivista:European journal of medicinal chemistry (Online)/anno:2014/pagina_da:/pagina_a:/intervallo_pagine:/volume
info:cnr-pdr/source/autori:Lucchesi V, Parkkari T, Savinainen JR, Malfitano AM, Allarà M, Bertini S, Castelli F, Del Carlo S, Laezza C, Ligresti A, Saccomanni G, Bifulco M, Di Marzo V, Macchia M, Manera C./titolo:1,2-Dihydro-2-oxopyridine-3-carboxamides: The C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor./doi:/rivista:European journal of medicinal chemistry (Online)/anno:2014/pagina_da:/pagina_a:/intervallo_pagine:/volume
info:cnr-pdr/source/autori:Lucchesi V, Parkkari T, Savinainen JR, Malfitano AM, Allarà M, Bertini S, Castelli F, Del Carlo S, Laezza C, Ligresti A, Saccomanni G, Bifulco M, Di Marzo V, Macchia M, Manera C./titolo:1,2-Dihydro-2-oxopyridine-3-carboxamides: the C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor./doi:/rivista:European journal of medicinal chemistry (Online)/anno:2014/pagina_da:/pagina_a:/intervallo_pagine:/volume
info:cnr-pdr/source/autori:Lucchesi V, Parkkari T, Savinainen JR, Malfitano AM, Allarà M, Bertini S, Castelli F, Del Carlo S, Laezza C, Ligresti A, Saccomanni G, Bifulco M, Di Marzo V, Macchia M, Manera C./titolo:1,2-Dihydro-2-oxopyridine-3-carboxamides: The C-5 substituent is responsible for functionality switch at CB2 cannabinoid receptor./doi:/rivista:European journal of medicinal chemistry (Online)/anno:2014/pagina_da:/pagina_a:/intervallo_pagine:/volume
The relevance of CB2R-mediated therapeutic effects is well-known for the treatment of inflammatory and neuropathic pain and neurodegenerative disorders. In our search for new cannabinoid receptor modulators, we report the optimization of a series of
Autor:
Anna Maria Malfitano, Giuseppe Saccomanni, Adriano Martinelli, Valentina Lucchesi, Tiziano Tuccinardi, Francesca Castelli, Simone Bertini, Antonio Giordano, Alessia Ligresti, Clementina Manera, Maurizio Bifulco, Flavio Rizzolio, Chiara Laezza, Vincenzo Di Marzo, Marco Macchia
Publikováno v:
European journal of medicinal chemistry (Online) (2012).
info:cnr-pdr/source/autori:Manera C, Saccomanni G, Malfitano AM, Bertini S, Castelli F, Laezza C, Ligresti A, Lucchesi V, Tuccinardi T, Rizzolio F, Bifulco M, Di Marzo V, Giordano A, Macchia M, Martinelli A./titolo:Rational design, synthesis and anti-proliferative properties of new CB2 selective cannabinoid receptor ligands: an investigation of the 1,8-naphthyridin-2(1H)-one scaffold./doi:/rivista:European journal of medicinal chemistry (Online)/anno:2012/pagina_da:/pagina_a:/intervallo_pagine:/volume
European journal of medicinal chemistry (2012).
info:cnr-pdr/source/autori:Manera C, Saccomanni G, Malfitano AM, Bertini S, Castelli F, Laezza C, Ligresti A, Lucchesi V, Tuccinardi T, Rizzolio F, Bifulco M, Di Marzo V, Giordano A, Macchia M, Martinelli A./titolo:Rational design, synthesis and anti-proliferative properties of new CB2 selective cannabinoid receptor ligands: an investigation of the 1,8-naphthyridin-2(1H)-one scaffold./doi:/rivista:European journal of medicinal chemistry/anno:2012/pagina_da:/pagina_a:/intervallo_pagine:/volume
info:cnr-pdr/source/autori:Manera C, Saccomanni G, Malfitano AM, Bertini S, Castelli F, Laezza C, Ligresti A, Lucchesi V, Tuccinardi T, Rizzolio F, Bifulco M, Di Marzo V, Giordano A, Macchia M, Martinelli A./titolo:Rational design, synthesis and anti-proliferative properties of new CB2 selective cannabinoid receptor ligands: an investigation of the 1,8-naphthyridin-2(1H)-one scaffold./doi:/rivista:European journal of medicinal chemistry (Online)/anno:2012/pagina_da:/pagina_a:/intervallo_pagine:/volume
European journal of medicinal chemistry (2012).
info:cnr-pdr/source/autori:Manera C, Saccomanni G, Malfitano AM, Bertini S, Castelli F, Laezza C, Ligresti A, Lucchesi V, Tuccinardi T, Rizzolio F, Bifulco M, Di Marzo V, Giordano A, Macchia M, Martinelli A./titolo:Rational design, synthesis and anti-proliferative properties of new CB2 selective cannabinoid receptor ligands: an investigation of the 1,8-naphthyridin-2(1H)-one scaffold./doi:/rivista:European journal of medicinal chemistry/anno:2012/pagina_da:/pagina_a:/intervallo_pagine:/volume
CB2 receptor ligands are becoming increasingly attractive drugs due to the potential role of this receptor in several physiopathological processes. Using our previously described series of 1,8-naphthyridin-2(1H)-on-3-carboxamides as a lead class, sev
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::792b5ba1fa57da3022f3c3fd743f9b0e
http://hdl.handle.net/11588/830241
http://hdl.handle.net/11588/830241