One-pot synthesis of tetrahydropyrimidinecarboxamides enabling in vitro anticancer activity: a combinative study with clinically relevant brain-penetrant drugs.

Autor: Upadhyay DB; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar Gujarat India hm_patel@spuvvn.edu., Nogales J; Division of Cancer Research, School of Medicine, University of Dundee Dundee DD1 9SY UK s.y.banerjee@dundee.ac.uk., Mokariya JA; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar Gujarat India hm_patel@spuvvn.edu., Vala RM; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar Gujarat India hm_patel@spuvvn.edu., Tandon V; Division of Cancer Research, School of Medicine, University of Dundee Dundee DD1 9SY UK s.y.banerjee@dundee.ac.uk., Banerjee S; Division of Cancer Research, School of Medicine, University of Dundee Dundee DD1 9SY UK s.y.banerjee@dundee.ac.uk., Patel HM; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar Gujarat India hm_patel@spuvvn.edu.

Publikováno v: RSC advances [RSC Adv] 2024 Aug 27; Vol. 14 (37), pp. 27174-27186. Date of Electronic Publication: 2024 Aug 27 (Print Publication: 2024).

Catalyst-Free, Room-Temperature Accessible Regioselective Synthesis of Spiroquinolines and Their Antioxidant Study.

Autor: Patel PJ; Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar388120, Gujarat, India., Patel DM; Department of Chemistry, AEPS Institute of Science, Ankleshwar393002, Gujarat, India.; Veer Narmad South Gujarat University, Surat395007, Gujarat, India., Vala RM; Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar388120, Gujarat, India., Patel SG; Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar388120, Gujarat, India., Upadhyay DB; Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar388120, Gujarat, India., Pannerselvam Y; Branch laboratory, CSIR-North East Institute of Science & Technology (NEIST), Imphal795004, Manipur, India., Patel HM; Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar388120, Gujarat, India.

Publikováno v: ACS omega [ACS Omega] 2022 Dec 19; Vol. 8 (1), pp. 444-456. Date of Electronic Publication: 2022 Dec 19 (Print Publication: 2023).

Microwave-assisted multicomponent synthesis of antiproliferative 2,4-dimethoxy-tetrahydropyrimido[4,5- b ]quinolin-6(7 H )-ones.

Autor: Patel SG; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar 388120 Gujarat India hm_patel@spuvvn.edu., González-Bakker A; BioLab, Instituto Universitario de Bio-Orgánica Antonio González (IUBO-AG), Universidad de La Laguna La Laguna E-38206 Spain., Vala RM; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar 388120 Gujarat India hm_patel@spuvvn.edu., Patel PJ; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar 388120 Gujarat India hm_patel@spuvvn.edu., Puerta A; BioLab, Instituto Universitario de Bio-Orgánica Antonio González (IUBO-AG), Universidad de La Laguna La Laguna E-38206 Spain., Malik A; Sustainable Materials and Catalysts Research Laboratory (SMCRL), Department of Chemistry, Indian Institute of Technology Jodhpur India., Sharma RK; Sustainable Materials and Catalysts Research Laboratory (SMCRL), Department of Chemistry, Indian Institute of Technology Jodhpur India., Padrón JM; BioLab, Instituto Universitario de Bio-Orgánica Antonio González (IUBO-AG), Universidad de La Laguna La Laguna E-38206 Spain., Patel HM; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar 388120 Gujarat India hm_patel@spuvvn.edu.

Publikováno v: RSC advances [RSC Adv] 2022 Oct 25; Vol. 12 (47), pp. 30404-30415. Date of Electronic Publication: 2022 Oct 25 (Print Publication: 2022).

One-pot two-step catalytic synthesis of 6-amino-2-pyridone-3,5-dicarbonitriles enabling anti-cancer bioactivity.

Autor: Nicely LG; Department of Cellular and Systems Medicine, School of Medicine, University of Dundee Dundee DD1 9SY UK s.y.banerjee@dundee.ac.uk., Vala RM; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar 388120 Gujarat India hm_patel@spuvvn.edu., Upadhyay DB; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar 388120 Gujarat India hm_patel@spuvvn.edu., Nogales J; Department of Cellular and Systems Medicine, School of Medicine, University of Dundee Dundee DD1 9SY UK s.y.banerjee@dundee.ac.uk., Chi C; Department of Medical Biochemistry and Microbiology, Uppsala University SE-75123 Uppsala Sweden., Banerjee S; Department of Cellular and Systems Medicine, School of Medicine, University of Dundee Dundee DD1 9SY UK s.y.banerjee@dundee.ac.uk., Patel HM; Department of Chemistry, Sardar Patel University Vallabh Vidyanagar 388120 Gujarat India hm_patel@spuvvn.edu.

Publikováno v: RSC advances [RSC Adv] 2022 Aug 24; Vol. 12 (37), pp. 23889-23897. Date of Electronic Publication: 2022 Aug 24 (Print Publication: 2022).

Syrbactin-class dual constitutive- and immuno-proteasome inhibitor TIR-199 impedes myeloma-mediated bone degeneration in vivo.

Autor: Tandon V; Department of Cellular Medicine, School of Medicine, University of Dundee, Dundee DD1 9SY, U.K., Vala RM; Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar 388120, Gujarat, India., Chen A; Department of Bioengineering, University of California, San Diego, La Jolla, CA 92093, U.S.A., Sah RL; Department of Bioengineering, University of California, San Diego, La Jolla, CA 92093, U.S.A., Patel HM; Department of Chemistry, Sardar Patel University, Vallabh Vidyanagar 388120, Gujarat, India., Pirrung MC; Department of Chemistry, University of California, Riverside, CA 92521, U.S.A.; Department of Pharmaceutical Sciences, University of California, Irvine, CA 92697, U.S.A., Banerjee S; Department of Cellular Medicine, School of Medicine, University of Dundee, Dundee DD1 9SY, U.K.

Publikováno v: Bioscience reports [Biosci Rep] 2022 Feb 25; Vol. 42 (2).