Zobrazeno 1 - 10
of 64
pro vyhledávání: '"Vaccaro, Henry"'
Autor:
Vaccaro, Henry Sebastian.
Thesis: M.S., Massachusetts Institute of Technology, Department of Civil Engineering, 1974
Bibliography: leaves 246-249.
M.S.
M.S. Massachusetts Institute of Technology, Department of Civil Engineering
Bibliography: leaves 246-249.
M.S.
M.S. Massachusetts Institute of Technology, Department of Civil Engineering
Externí odkaz:
https://hdl.handle.net/1721.1/155524
Autor:
McKittrick, Brian A., Caldwell, John P., Bara, Thomas, Boykow, George, Chintala, Madhu, Clader, John, Czarniecki, Michael, Courneya, Brandy, Duffy, Ruth, Fleming, Linda, Giessert, Rachel, Greenlee, William J., Heap, Charles, Hong, Liwu, Huang, Ying, Iserloh, Ulrich, Josien, Hubert, Khan, Tanweer, Korfmacher, Walter, Liang, Xian, Mazzola, Robert, Mitra, Soumya, Moore, Kristina, Orth, Peter, Rajagopalan, Murali, Roy, Sudipta, Sakwa, Samuel, Strickland, Corey, Vaccaro, Henry, Voigt, Johannes, Wang, Hongwu, Wong, Jesse, Zhang, Rumin, Zych, Andrew
Publikováno v:
In Bioorganic & Medicinal Chemistry Letters 1 April 2015 25(7):1592-1596
Autor:
Tony Priestley, Vaccaro Henry A, Andrew Stamford, Deborra E Mullins, Michael W. Miller, Tin-Yau Chan, Robert A. Hodgson, Scott Jack D, William J. Greenlee, Liwu Hong, Mario Guzzi, Sarah W. Li, Eric M. Parker, Geoffrey B. Varty, Jay Weinstein, Sue-Ing Lin, Mckittrick Brian A
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 19:6018-6022
Vasopressin 1b (V1b) antagonists have been postulated as possible treatments for depression and anxiety. A novel series of potent and selective V1b antagonists has been identified starting from an in-house screen hit. The incorporation of a sulfonami
Autor:
Piwinski John J, Neng-Yang Shih, Robert E. West, Shirley M. Williams, Robert G. Aslanian, Vaccaro Henry A, Xiaohong Zhu
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 18:5032-5036
A series of non-imidazole histamine H(3) receptor antagonists based on the (3-phenoxypropyl)amine motif, which is a common pharmacophore for H(3) antagonists, has been identified. A preliminary SAR study around the amine moiety has identified 8a as a
Autor:
Zhiqiang Zhao, Lili Zhang, Giuseppe Terracina, Dmitri A. Pissarnitski, Lixin Song, Vaccaro Henry A, John W. Clader
Publikováno v:
Journal of Combinatorial Chemistry. 10:56-62
A novel methodology for parallel liquid-phase synthesis of carbamates suitable for the preparation of sterically hindered molecules is disclosed. The alcohols are converted to 4-nitrophenylcarbonates, followed by the reaction with amines. Side produc
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Autor:
Vaccaro Henry A, Ahmad Fawzi, Hongtao Zhang, Robert W. Watkins, Hsingan Tsai, Renee Cleven, Yan Xia, Michael Czarniecki, John Cook, Samuel Chackalamannil
Publikováno v:
Journal of Medicinal Chemistry. 40:4372-4377
Polycyclic pyrazolo[3,4-d]pyrimidines (represented by 3 and 4) were synthesized as analogues of the recently reported polycyclic guanine phosphodiesterase (PDE) inhibitors. From the structure-activity relationship (SAR) development of a series of com
Akademický článek
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Autor:
Vaccaro Henry A, Robert W. Watkins, Yan Xia, Hsingan Tsai, Renee Cleven, Hongtao Zhang, Ahmad Fawzi, Michael Czarniecki, Samuel Chackalamannil, John Cook
Publikováno v:
ChemInform. 29
Polycyclic pyrazolo[3,4-d]pyrimidines (represented by 3 and 4) were synthesized as analogues of the recently reported polycyclic guanine phosphodiesterase (PDE) inhibitors. From the structure−activ...
Autor:
Piwinski John J, Corey O. Strickland, Jing Sun, Patrick J. Curran, Vinay Girijavallabhan, Zhuyan Guo, Li Wang, Shih Neng-Yang, Liwu Hong, Yongqi Deng, Pauline C. Ting, Daniel Lundell, Guowei Zhou, Gerald W. Shipps, Chan Tin Yau, Wensheng Yu, Zhidan Liu, Joe F. Lee, M. Arshad Siddiqui, Janeta Popovici-Muller, Xiaoda Niu, Brian J. Lavey, Vincent Madison, Tong Wang, Chaoyang Dai, Joseph A. Kozlowski, Mckittrick Brian A, Kristin E. Rosner, David B. Belanger, Vaccaro Henry A, Dansu Li, Peter Orth
Publikováno v:
Bioorganicmedicinal chemistry letters. 20(3)
A novel series of TNF-α convertase (TACE) inhibitors which are non-hydroxamate have been discovered. These compounds are bis-amides of l -tartaric acid (tartrate) and coordinate to the active site zinc in a tridentate manner. They are selective for