Zobrazeno 1 - 10 of 24 pro vyhledávání: '"Tulshiram L. Dadmal"'
1
Synthesis and Antimicrobial Activity of 1,2,3-Triazole Linked Benzo[d]oxazole-2-thiol/ oxazolo[4,5-b]pyridine-2-thiol Derivatives
Autor: Tulshiram L. Dadmal, Lata Deshmukh, Archana M. Ramteke, Pankaj B. Gour
Publikováno v: Asian Journal of Organic & Medicinal Chemistry. 6:7-12
A new series of 1,2,3-triazole linked mercaptobenzoxazole/oxazolo- [4,5-b] pyridine-2-thiol derivatives (6a-j) were synthesized starting from 2-aminophenol/2-aminopyridin-3-ol in three steps via cyclization, alkylation followed by reaction with vario
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::66c380e4b9ce1bd2c24af628f2588844
https://doi.org/10.14233/ajomc.2021.ajomc-p293
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4
Contemporary progress in the synthesis and reactions of 2-aminobenzothiazole: a review
Autor: Ravindra M. Kumbhare, Mustapha Mandewale, Sangita D. Katre, Tulshiram L. Dadmal
Publikováno v: New Journal of Chemistry. 42:776-797
In the past few decades, heterocyclic compounds and their derivatives have gained popularity due to their prominent medicinal importance. The versatile and synthetically accessible 2-aminobenzothiazole scaffolds are quite fascinating for multiple app
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::433210952f21b651d191a0017fc89d8f
https://doi.org/10.1039/c7nj03776g
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5
Synthesis and biological evaluation of triazole and isoxazole-tagged benzothiazole/benzoxazole derivatives as potent cytotoxic agents
Autor: Ravindra M. Kumbhare, Tulshiram L. Dadmal, K. Appalanaidu, Manika Pal Bhadra, Tanmoy Mondal, M. Janaki Ramaiah
Publikováno v: New Journal of Chemistry. 42:15546-15551
Cancer is a major health problem and the most upsetting disease in humans, leading to death in both developed and developing countries. Proper treatment of the disease is still a challenge. Chemotherapy is considered one of the regimens to cure this
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::b49ce96211c748e0d5ce431636122997
https://doi.org/10.1039/c8nj01249k
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6
Synthesis and biological evaluation of novel 2-imino-4-thiazolidinone derivatives as potent anti-cancer agents
Autor: K. Appalanaidu, Rajesh Kotcherlakota, Vishnu Sravan Bollu, Chitta Ranjan Patra, Tulshiram L. Dadmal, Ravindra M. Kumbhare
Publikováno v: Bioorganic & Medicinal Chemistry Letters. 26:5361-5368
A new series of 2-imino-4-thiazolidinone derivatives (7a–7t) has been synthesised and screened for their cytotoxicity against three cancer cell lines (B16F10, A549, PANC-1) and normal cell line (CHO). Among the compounds tested, compounds 7k, 7m, 7
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7fc77e1c8f23dde9bf84db923fb017d6
https://doi.org/10.1016/j.bmcl.2016.08.013
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7
Synthesis and anticancer evaluation of novel triazole linked N-(pyrimidin-2-yl)benzo[d]thiazol-2-amine derivatives as inhibitors of cell survival proteins and inducers of apoptosis in MCF-7 breast cancer cells
Autor: S.N.C.V.L. Pushpa Valli, Manika Pal Bhadra, M. Janaki Ramaiah, Tulshiram L. Dadmal, Ravindra M. Kumbhare, Sudheer Kumar Tiwari, Y. Khageswar Rao, K. Appalanaidu, K.S.V. Kishore
Publikováno v: Bioorganic & Medicinal Chemistry Letters. 25:654-658
A series of novel triazole linked N-(pyrimidin-2yl)benzo[d]thiazol-2-amine 5a-k were synthesized and evaluated for anticancer activity against breast (MCF-7), lung (A549) and skin (A375) cancer cell lines and their cytotoxic effects were compared aga
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::76bcf3b47655c2128ce5a24b62dd890d
https://doi.org/10.1016/j.bmcl.2014.11.083
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8
An improved one-pot multicomponent strategy for the preparation of thiazoline, thiazolidinone and thiazolidinol scaffolds
Autor: Ravindra M. Kumbhare, K. Appalanaidu, Tulshiram L. Dadmal, N. Jagadeesh Babu
Publikováno v: RSC Advances. 5:88063-88069
A facile multicomponent synthesis of desirable medicinal scaffolds based on thiazoline, thiazolidinone and thiazolidinol derivatives has been disclosed. The synthesis employs the reaction of a primary amine and carbon disulphide in a microwave, to ge
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::a1256c7e0994148e3d3db05b010bafe1
https://doi.org/10.1039/c5ra17278k
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9
Synthesis of novel fluoro 1,2,3-triazole tagged amino bis(benzothiazole) derivatives, their antimicrobial and anticancer activity
Autor: Y. Khageswara Rao, J. Venkateswara Rao, Umesh B. Kosurkar, Rajesh Pamanji, Ravindra M. Kumbhare, L. R. Velatooru, Tulshiram L. Dadmal, K. Appalanaidu
Publikováno v: Medicinal Chemistry Research. 23:4404-4413
A new series of fluoro 1,2,3-triazole tagged amino bis (benzothiazole) derivatives 8, 9 were prepared starting from 2-amino benzothiazole in four steps via amination, cyclization, alkylation followed by reaction with various azides under sharpless co
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::ed29b73c54936c9d2f1d46209d6cd2c5
https://doi.org/10.1007/s00044-014-1006-0
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10
An Environmentally Benign Water Promoted Catalyst Free Highly Efficient, One-pot Synthesis of 2-Imino-4-thiazolidinone
Autor: Tulshiram L. Dadmal, Ravindra M. Kumbhare, Balasubramanian Sridhar, Umesh B. Kosurkar
Publikováno v: Journal of Heterocyclic Chemistry. 51:1522-1527
A practical and efficient protocol has been developed for the synthesis of 2-imino-4-thiazolidinone through a unique one pot three-component reaction of variety of amines, isothiocyanate and ethylbromoacetate in water. The method is free of catalyst
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::4864c3a79067422a266e5056a1fc9913
https://doi.org/10.1002/jhet.1812
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