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DFT-based ranking of zinc-binding groups in histone deacetylase inhibitors

Autor: Vanommeslaeghe, K., Loverix, S., Geerlings, P., Tourwé, D.

Publikováno v: In Bioorganic & Medicinal Chemistry 2005 13(21):6070-6082

Rapid construction of substituted 3-amino-1,5-benzothiazepin-4(5H)-one dipeptide scaffolds through an Ugi-4CR - Ullmann cross-coupling sequence. IF 3.49

Autor: Van der Poorten, O, Van Den Hauwe, R, Hollanders, K, Tourwé, D, Jida, M, Ballet, S

A 3-step methodology for the synthesis of 1,5-benzothiazepin-4(5H)-one dipeptidomimetics has been elaborated via an Ugi-4CR followed by a S-trityl deprotection and an intramolecular Cu(i)-catalyzed Ullmann condensation with moderate to good yields. I

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=od______3848::94fc0cfae61c056849349a42bea3dd4a
https://doi.org/10.1039/c7ob03094k

Synthesis, biological evaluation and automated docking of constrained analogs of the opioid peptide H-Dmt-D-AlapPhe-Gly-NH2 using the 4- or 5-metyl substsituted 4-amino-1,2,3,4-tetrahydro-2-benzazepin-3-one scaffold

Autor: Wachter, R., Chris de Graaf, Keresztes, C., Vandormael, B., Ballet, S., Toth, G., Rognan, D., Tourwé, D.

Publikováno v: de Wachter, R, de Graaf, C, Keresztes, C, Vandormael, B, Ballet, S, Toth, G, Rognan, D & Tourwé, D 2011, ' Synthesis, biological evaluation and automated docking of constrained analogs of the opioid peptide H-Dmt-D-AlapPhe-Gly-NH2 using the 4-or 5-metyl substsituted 4-amino-1,2,3,4-tetrahydro-2-benzazepin-3-one scaffold. ', Journal of Medicinal Chemistry, vol. 54, pp. 3384-3393 .
Journal of Medicinal Chemistry, 54, 3384-3393. American Chemical Society
Vrije Universiteit Amsterdam

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::c1ab2cec994469a07c3e8339dcf19cf7
https://hdl.handle.net/1871.1/95c629e8-0c0d-4e58-8c86-6c0c187ac193

Carbohydrated [99mTc(CO)3](NalphaHis)Ac-bombesin(7-14) analogs

Autor: Maes, V, Brans, L, Schweinsberg, C, Garcia-Garayoa, E, Bläuenstein, P, Schubiger, P A, Tourwé, D

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=od_______885::4425c112737086c58c4d6177656ec842
https://www.zora.uzh.ch/id/eprint/26532/