Zobrazeno 1 - 10
of 149
pro vyhledávání: '"Tomoyasu Hirose"'
Autor:
Rattiya Janthanom, Yuta Kikuchi, Hiroki Kanto, Tomoyasu Hirose, Arisu Tahara, Takahiro Ishii, Arinthip Thamchaipenet, Yuki Inahashi
Publikováno v:
Beilstein Journal of Organic Chemistry, Vol 20, Iss 1, Pp 497-503 (2024)
Actinomycetes are well-known as the main producers of bioactive compounds such as antibiotics, anticancers, and immunosuppressants. Screening of natural products from actinomycetes has been an essential part of several drug discovery programs. Findin
Externí odkaz:
https://doaj.org/article/32f31054cfde46fb9c7a4c9360946781
Autor:
Kridtapat Sirisereephap, Hikaru Tamura, Jong-Hyung Lim, Meircurius Dwi Condro Surboyo, Toshihito Isono, Takumi Hiyoshi, Andrea L. Rosenkranz, Yurie Sato-Yamada, Hisanori Domon, Akari Ikeda, Tomoyasu Hirose, Toshiaki Sunazuka, Nagako Yoshiba, Hiroyuki Okada, Yutaka Terao, Takeyasu Maeda, Koichi Tabeta, Triantafyllos Chavakis, George Hajishengallis, Tomoki Maekawa
Publikováno v:
iScience, Vol 27, Iss 2, Pp 108798- (2024)
Summary: Aging is associated with increased susceptibility to chronic inflammatory bone loss disorders, such as periodontitis, in large part due to the impaired regenerative potential of aging tissues. DEL-1 exerts osteogenic activity and promotes bo
Externí odkaz:
https://doaj.org/article/b4d1b2b7ec0e4334957f28a8a3880467
Autor:
Kenichi Aizawa, Akari Ikeda, Shota Tomida, Koki Hino, Yuuki Sugita, Tomoyasu Hirose, Toshiaki Sunazuka, Hiroshi Kido, Shigeyuki Yokoyama, Ryozo Nagai
Publikováno v:
Cells, Vol 13, Iss 1, p 87 (2023)
Heart failure with reduced ejection fraction (HFrEF) is characterized not only by reduced left ventricular ejection fraction (EF) but is also combined with symptoms such as dyspnea, fatigue, and edema. Several pharmacological interventions have been
Externí odkaz:
https://doaj.org/article/975d7b0db66346b6a1d334ceaa63364a
Autor:
Ryo Horikoshi, Kimihiko Goto, Masaaki Mitomi, Kazuhiko Oyama, Tomoyasu Hirose, Toshiaki Sunazuka, Satoshi Ōmura
Publikováno v:
Scientific Reports, Vol 12, Iss 1, Pp 1-10 (2022)
Abstract Afidopyropen, a novel insecticide, is a derivative of pyripyropene A, which is produced by the filamentous fungus Penicillium coprobium. Afidopyropen has strong insecticidal activity against aphids and is currently used as a control agent of
Externí odkaz:
https://doaj.org/article/9566497a62084d36acdc9bfd85d36b89
Autor:
Sho Inoue, Yuki Inahashi, Makoto Itakura, Gen Inoue, Kyoko Muneshige, Tomoyasu Hirose, Masato Iwatsuki, Masashi Takaso, Masayuki Miyagi, Kentaro Uchida
Publikováno v:
International Journal of Molecular Sciences, Vol 24, Iss 18, p 13871 (2023)
Synovial inflammation plays a crucial role in the destruction of joints and the experience of pain in osteoarthritis (OA). Emerging evidence suggests that certain antibiotic agents and their derivatives possess anti-inflammatory properties. Medermyci
Externí odkaz:
https://doaj.org/article/422f90b78e25444997c88d5efc50c753
Autor:
Kyoko Muneshige, Yuki Inahashi, Makoto Itakura, Masato Iwatsuki, Tomoyasu Hirose, Gen Inoue, Masashi Takaso, Toshiaki Sunazuka, Yoshihisa Ohashi, Etsuro Ohta, Kentaro Uchida
Publikováno v:
Pharmaceuticals, Vol 16, Iss 1, p 5 (2022)
Synovial inflammation plays a central role in joint destruction and pain in osteoarthritis (OA). The NF-κB pathway plays an important role in the inflammatory process and is activated in OA. A previous study reported that a jietacin derivative (JD),
Externí odkaz:
https://doaj.org/article/2b2d62f0d980468bb2cc51e3a24858bc
Autor:
Anna Nakanishi, Hiroki Okumura, Tadahiro Hashita, Aya Yamashita, Yuka Nishimura, Chihiro Watanabe, Sakina Kamimura, Sanae Hayashi, Shuko Murakami, Kyoko Ito, Takahiro Iwao, Akari Ikeda, Tomoyasu Hirose, Toshiaki Sunazuka, Yasuhito Tanaka, Tamihide Matsunaga
Publikováno v:
Viruses, Vol 14, Iss 11, p 2468 (2022)
Hepatitis B virus (HBV) specifically infects human hepatocytes and increases the risks of cirrhosis and liver cancer. Currently, nucleic acid analogs are the main therapeutics for chronic hepatitis caused by HBV infection. Although nucleic acid analo
Externí odkaz:
https://doaj.org/article/c8cb069c76e847feb81b286bbed86399
Autor:
Chisa Kobayashi, Yoshihiro Watanabe, Mizuki Oshima, Tomoyasu Hirose, Masako Yamasaki, Masashi Iwamoto, Masato Iwatsuki, Yukihiro Asami, Kouji Kuramochi, Kousho Wakae, Hideki Aizaki, Masamichi Muramatsu, Camille Sureau, Toshiaki Sunazuka, Koichi Watashi
Publikováno v:
Viruses, Vol 14, Iss 4, p 764 (2022)
Current anti-hepatitis B virus (HBV) drugs are suppressive but not curative for HBV infection, so there is considerable demand for the development of new anti-HBV agents. In this study, we found that fungus-derived exophillic acid inhibits HBV infect
Externí odkaz:
https://doaj.org/article/9670e2105fe742b1a5396a01e8c5fe35
Autor:
Goh Sennari, Ryo Saito, Tomoyasu Hirose, Masato Iwatsuki, Aki Ishiyama, Rei Hokari, Kazuhiko Otoguro, Satoshi Ōmura, Toshiaki Sunazuka
Publikováno v:
Scientific Reports, Vol 7, Iss 1, Pp 1-9 (2017)
Abstract Divergent synthesis of antimalarial troponoids, including naturally occurring compounds, some of which were identified and isolated by our group, has been achieved utilizing the total synthetic route of puberulic acid. Structure-activity rel
Externí odkaz:
https://doaj.org/article/6625936338a845379b8e4d5e81716ef2
Autor:
Tomoyasu Hirose, Kaori Ozaki, Yukiko Saito, Reiko Takai-Todaka, Hidehito Matsui, Masako Honsho, Masato Iwatsuki, Yukihiro Asami, Kazuhiko Katayama, Toshiaki Sunazuka, Hideaki Hanaki, Toshiaki Teruya
Publikováno v:
Chemical and Pharmaceutical Bulletin. 71:374-379