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Autor:
Logvinenko IG; Enamine Ltd, Winston Churchill Str. 78, Kyiv 02094, Ukraine.; Address V.P. Kukhar Institute of Bioorganic Chemistry & Petrochemistry, National Academy of Sciences of Ukraine, Academician Kukhar Str. 1, Kyiv 02094, Ukraine., Sadkova IV; Enamine Ltd, Winston Churchill Str. 78, Kyiv 02094, Ukraine., Tolmachova NA; Enamine Ltd, Winston Churchill Str. 78, Kyiv 02094, Ukraine., Shishkina SV; SSI 'Institute for Single Crystals' of the National Academy of Sciences of Ukraine, Nauky Ave. 60, Kharkiv 61072, Ukraine.; Institute of Organic Chemistry of the National Academy of Sciences of Ukraine, Academician Kukhar Str. Str. 5, Kyiv 02660, Ukraine., Daniliuc CG; Organisch-Chemisches Institut, Universität Münster, Corrensstraße 40, Münster 48149, Germany., Haufe G; Organisch-Chemisches Institut, Universität Münster, Corrensstraße 40, Münster 48149, Germany.; Cells-in-Motion Cluster of Excellence, Universität Münster, Waldeyerstraße 15, 48149 Münster, Germany., Kondratov IS; Enamine Ltd, Winston Churchill Str. 78, Kyiv 02094, Ukraine.; Address V.P. Kukhar Institute of Bioorganic Chemistry & Petrochemistry, National Academy of Sciences of Ukraine, Academician Kukhar Str. 1, Kyiv 02094, Ukraine.; Enamine Germany GmbH, Industriepark Hoechst, G837, 65926 Frankfurt am Main, Germany. ivan.s.kondratov@gmail.com.
Publikováno v:
Organic & biomolecular chemistry [Org Biomol Chem] 2024 Oct 09; Vol. 22 (39), pp. 7982-7988. Date of Electronic Publication: 2024 Oct 09.
Autor:
Singh I; Department of Pharmaceutical Chemistry, University of California San Francisco, San Francisco, California 94143, United States., Li F; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada., Fink EA; Department of Pharmaceutical Chemistry, University of California San Francisco, San Francisco, California 94143, United States.; Graduate Program in Biophysics, University of California San Francisco, San Francisco, California 94143, United States., Chau I; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada., Li A; Department of Pharmacology and Toxicology, University of Toronto, Toronto, Ontario M5S 1A8, Canada.; Drug Discovery Program, Ontario Institute for Cancer Research, Toronto, Ontario M5G 0A3, Canada., Rodriguez-Hernández A; Department of Cellular and Molecular Pharmacology, University of California San Francisco, San Francisco, California 94158, United States., Glenn I; Department of Pharmaceutical Chemistry, University of California San Francisco, San Francisco, California 94143, United States., Zapatero-Belinchón FJ; Gladstone Institutes, San Francisco, California 94158, United States., Rodriguez ML; Department of Microbiology, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States.; Global Health and Emerging Pathogens Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States., Devkota K; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada., Deng Z; Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences, Oncological Sciences and Neuroscience, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States., White K; Department of Microbiology, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States.; Global Health and Emerging Pathogens Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States., Wan X; Department of Pharmaceutical Chemistry, University of California San Francisco, San Francisco, California 94143, United States., Tolmachova NA; Enamine Ltd, Kyïv 02094, Ukraine.; Institute of Bioorganic Chemistry and Petrochemistry, National Ukrainian Academy of Science, Kyïv 02660, Ukraine., Moroz YS; National Taras Shevchenko University of Kyïv, Kyïv 01601, Ukraine.; Chemspace, Riga LV-1082, Latvia., Kaniskan HÜ; Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences, Oncological Sciences and Neuroscience, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States., Ott M; Gladstone Institutes, San Francisco, California 94158, United States.; QBI COVID-19 Research Group (QCRG), San Francisco, California 94158, United States.; Department of Medicine, University of California, San Francisco, San Francisco, California 94158, United States.; Chan Zuckerberg Biohub, San Francisco, California 94158, United States., García-Sastre A; Department of Microbiology, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States.; Global Health and Emerging Pathogens Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States.; QBI COVID-19 Research Group (QCRG), San Francisco, California 94158, United States.; Department of Medicine, Division of Infectious Diseases, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States.; The Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States., Jin J; Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences, Oncological Sciences and Neuroscience, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States.; QBI COVID-19 Research Group (QCRG), San Francisco, California 94158, United States., Fujimori DG; Department of Pharmaceutical Chemistry, University of California San Francisco, San Francisco, California 94143, United States.; Department of Cellular and Molecular Pharmacology, University of California San Francisco, San Francisco, California 94158, United States.; QBI COVID-19 Research Group (QCRG), San Francisco, California 94158, United States., Irwin JJ; Department of Pharmaceutical Chemistry, University of California San Francisco, San Francisco, California 94143, United States.; QBI COVID-19 Research Group (QCRG), San Francisco, California 94158, United States., Vedadi M; Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada.; Department of Pharmacology and Toxicology, University of Toronto, Toronto, Ontario M5S 1A8, Canada.; QBI COVID-19 Research Group (QCRG), San Francisco, California 94158, United States.; Drug Discovery Program, Ontario Institute for Cancer Research, Toronto, Ontario M5G 0A3, Canada., Shoichet BK; Department of Pharmaceutical Chemistry, University of California San Francisco, San Francisco, California 94143, United States.; QBI COVID-19 Research Group (QCRG), San Francisco, California 94158, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2023 Jun 22; Vol. 66 (12), pp. 7785-7803. Date of Electronic Publication: 2023 Jun 09.
Autor:
Chernykh AV; Enamine Ltd., Chervonotkatska Street 78, Kyïv 02094, Ukraine. kondratov@enamine.net.; Taras Shevchenko National University of Kyïv, Volodymyrska Street 60, Kyïv 01601, Ukraine. gregor@univ.kiev.ua., Aloshyn D; Bienta/Enamine Ltd., Chervonotkatska Street 78, Kyïv 02094, Ukraine., Kuchkovska YO; Enamine Ltd., Chervonotkatska Street 78, Kyïv 02094, Ukraine. kondratov@enamine.net., Daniliuc CG; Organisch-Chemisches Institut, Westfälische Wilhelms-Universität Münster, Corrensstrasse 40, 48149 Münster, Germany., Tolmachova NA; Enamine Ltd., Chervonotkatska Street 78, Kyïv 02094, Ukraine. kondratov@enamine.net., Kondratov IS; Enamine Ltd., Chervonotkatska Street 78, Kyïv 02094, Ukraine. kondratov@enamine.net.; V.P. Kukhar Institute of Bioorganic Chemistry & Petrochemistry, National Academy of Sciences of, Ukraine, Murmanska Street 1, Kyïv 02660, Ukraine., Zozulya S; Bienta/Enamine Ltd., Chervonotkatska Street 78, Kyïv 02094, Ukraine., Grygorenko OO; Enamine Ltd., Chervonotkatska Street 78, Kyïv 02094, Ukraine. kondratov@enamine.net.; Taras Shevchenko National University of Kyïv, Volodymyrska Street 60, Kyïv 01601, Ukraine. gregor@univ.kiev.ua., Haufe G; Organisch-Chemisches Institut, Westfälische Wilhelms-Universität Münster, Corrensstrasse 40, 48149 Münster, Germany.; Cells-in-Motion Cluster of Excellence, Universität Münster, Waldeyerstraße 15, 48149 Münster, Germany.
Publikováno v:
Organic & biomolecular chemistry [Org Biomol Chem] 2022 Dec 07; Vol. 20 (47), pp. 9337-9350. Date of Electronic Publication: 2022 Dec 07.
Autor:
Fink EA; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, USA.; Graduate Program in Biophysics, University of California, San Francisco, San Francisco, CA, USA., Xu J; Kobilka Institute of Innovative Drug Discovery, School of Life and Health Sciences, Chinese University of Hong Kong, Shenzhen, Guangdong 518172, China.; Department of Molecular and Cellular Physiology, Stanford University School of Medicine, Stanford, CA, USA., Hübner H; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91058 Erlangen, Germany., Braz JM; Department of Anatomy, University of California, San Francisco, San Francisco, CA, USA., Seemann P; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91058 Erlangen, Germany., Avet C; Department of Biochemistry and Molecular Medicine, Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, QC, Canada., Craik V; Department of Anatomy, University of California, San Francisco, San Francisco, CA, USA., Weikert D; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91058 Erlangen, Germany., Schmidt MF; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91058 Erlangen, Germany., Webb CM; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, USA.; Graduate Program in Pharmaceutical Sciences and Pharmacogenomics, University of California, San Francisco, San Francisco, CA, USA., Tolmachova NA; Enamine Ltd., 02094 Kyiv, Ukraine.; Institute of Bioorganic Chemistry and Petrochemistry, National Ukrainian Academy of Science, 02660 Kyiv, Ukraine., Moroz YS; National Taras Shevchenko University of Kyiv, 01601 Kyiv, Ukraine.; Chemspace, Riga LV-1082, Latvia., Huang XP; National Institute of Mental Health Psychoactive Drug Screening Program (NIMH PDSP), School of Medicine, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, NC, USA., Kalyanaraman C; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, USA., Gahbauer S; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, USA., Chen G; Kobilka Institute of Innovative Drug Discovery, School of Life and Health Sciences, Chinese University of Hong Kong, Shenzhen, Guangdong 518172, China., Liu Z; Kobilka Institute of Innovative Drug Discovery, School of Life and Health Sciences, Chinese University of Hong Kong, Shenzhen, Guangdong 518172, China., Jacobson MP; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, USA., Irwin JJ; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, USA., Bouvier M; Department of Biochemistry and Molecular Medicine, Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, QC, Canada., Du Y; Kobilka Institute of Innovative Drug Discovery, School of Life and Health Sciences, Chinese University of Hong Kong, Shenzhen, Guangdong 518172, China., Shoichet BK; Department of Pharmaceutical Chemistry, University of California, San Francisco, San Francisco, CA, USA., Basbaum AI; Department of Anatomy, University of California, San Francisco, San Francisco, CA, USA., Gmeiner P; Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, 91058 Erlangen, Germany.
Publikováno v:
Science (New York, N.Y.) [Science] 2022 Sep 30; Vol. 377 (6614), pp. eabn7065. Date of Electronic Publication: 2022 Sep 30.
Autor:
Tolmachova NA; Enamine Ltd, Chervonotkatska Str. 78, Kyiv, 02094, Ukraine. n.tolmachova@mail.enamine.net., Kondratov IS, Dolovanyuk VG, Pridma SO, Chernykh AV, Daniliuc CG, Haufe G
Publikováno v:
Chemical communications (Cambridge, England) [Chem Commun (Camb)] 2018 Aug 23; Vol. 54 (69), pp. 9683-9686.
Autor:
Kondratov IS; Enamine Ltd, Chervonotkatska St 78, Kyiv, 02094, Ukraine. vanya_ko@mail.ru and Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine, Murmanska Str. 1, Kyiv, 02660, Ukraine., Logvinenko IG; Enamine Ltd, Chervonotkatska St 78, Kyiv, 02094, Ukraine. vanya_ko@mail.ru and Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine, Murmanska Str. 1, Kyiv, 02660, Ukraine., Tolmachova NA; Enamine Ltd, Chervonotkatska St 78, Kyiv, 02094, Ukraine. vanya_ko@mail.ru and Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine, Murmanska Str. 1, Kyiv, 02660, Ukraine., Morev RN; Enamine Ltd, Chervonotkatska St 78, Kyiv, 02094, Ukraine. vanya_ko@mail.ru., Kliachyna MA; Enamine Ltd, Chervonotkatska St 78, Kyiv, 02094, Ukraine. vanya_ko@mail.ru., Clausen F; Organisch-Chemisches Institut, Universität Münster, Corrensstraße 40, Münster 48149, Germany. haufe@uni-muenster.de., Daniliuc CG; Organisch-Chemisches Institut, Universität Münster, Corrensstraße 40, Münster 48149, Germany. haufe@uni-muenster.de., Haufe G; Organisch-Chemisches Institut, Universität Münster, Corrensstraße 40, Münster 48149, Germany. haufe@uni-muenster.de and Cells-in-Motion Cluster of Excellence, Universität Münster, Waldeyerstraße 15, 48149 Münster, Germany.
Publikováno v:
Organic & biomolecular chemistry [Org Biomol Chem] 2017 Jan 18; Vol. 15 (3), pp. 672-679.
Autor:
Kondratov IS; Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine , Murmanska Str. 1, Kyiv, 02660, Ukraine., Bugera MY; Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine , Murmanska Str. 1, Kyiv, 02660, Ukraine., Tolmachova NA; Institute of Bioorganic Chemistry and Petrochemistry, National Academy of Sciences of Ukraine , Murmanska Str. 1, Kyiv, 02660, Ukraine.; Enamine Ltd , Chervonotkatska Str. 78, Kyiv, 02094, Ukraine., Posternak GG; Enamine Ltd , Chervonotkatska Str. 78, Kyiv, 02094, Ukraine., Daniliuc CG; Organisch-Chemisches Institut, Universität Münster , Corrensstraße 40, 48149 Münster, Germany., Haufe G; Organisch-Chemisches Institut, Universität Münster , Corrensstraße 40, 48149 Münster, Germany.; Cells-in-Motion Cluster of Excellence, Universität Münster , Waldeyerstraße 15, 48149 Münster, Germany.
Publikováno v:
The Journal of organic chemistry [J Org Chem] 2015 Dec 18; Vol. 80 (24), pp. 12258-64. Date of Electronic Publication: 2015 Nov 25.
Autor:
Kondratov IS; Institute of Bioorganic Chemistry and Petrochemistry, National Ukrainian Academy of Sciences, Murmanska 1, Kiev-94, 02660, Ukraine., Dolovanyuk VG, Tolmachova NA, Gerus II, Bergander K, Fröhlich R, Haufe G
Publikováno v:
Organic & biomolecular chemistry [Org Biomol Chem] 2012 Nov 28; Vol. 10 (44), pp. 8778-85.