Zobrazeno 1 - 10
of 21
pro vyhledávání: '"Thomas N. Riley"'
Autor:
Nadezda Vukicevic-Nikolic, Danica Agbaba, Aleksandar Todorovic, Thomas N. Riley, Katarina Karljikovic-Rajic
Publikováno v:
Pharmacy Education
The role of the pharmacist and of pharmacy education within a modern patient-based approach is important as is having an adequate curricula for a professional pharmaceutical degree. Although there are various approaches in the field of education, thi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ca6e123f5d220571e92d9a12aac7b7c0
https://doi.org/10.1080/1560221021000061823
https://doi.org/10.1080/1560221021000061823
Publikováno v:
Journal of Heterocyclic Chemistry. 29:779-786
Methods are explored to enhance the efficiency and versatility of the synthesis of the 1-substituted 4-(propananilido)perhydroazepine analgesics. The modified synthesis begins with ring expansion of 1-carbethoxy-4-piperidinone 3 with ethyl diazoaceta
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f8cd118b2b73a9bdfcd82495541b3bd9
https://doi.org/10.1002/jhet.5570290417
https://doi.org/10.1002/jhet.5570290417
Publikováno v:
SAE Technical Paper Series.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fdf34162b1c56fff1783390e3ff82af8
https://doi.org/10.4271/902277
https://doi.org/10.4271/902277
Publikováno v:
Journal of Chromatographic Science. 18:153-158
A method for the prediction of the retention index of drugs on C18 reversed-phase columns was developed and then applied to a series of drugs that were structurally related to morphine and to a series related to fentanyl. The HPLC retention index (/)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::33e2936914921d532ca367a48eecd576
https://doi.org/10.1093/chromsci/18.4.153
https://doi.org/10.1093/chromsci/18.4.153
Autor:
Thomas N. Riley, Jerome R. Bagley
Publikováno v:
Journal of Heterocyclic Chemistry. 14:599-602
The isomeric 3-anilino and 3-propananilidotropanes have been synthesized and obtained in isomerically pure form. The configurations and solute conformations of these isomers were studied via glc and nrar analysis. The 3β-isomers have been shown to e
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::597c70ed8892ea6a1db91b453b41629c
https://doi.org/10.1002/jhet.5570140412
https://doi.org/10.1002/jhet.5570140412
Publikováno v:
Journal of Medicinal Chemistry. 30:1105-1110
The exo- and endo-2-amino-5,8-dimethoxy-1,2,3,4-tetrahydro-1,4-epoxynaphthalenes++ + (3b and 4b, respectively) were prepared and evaluated as conformationally defined analogues of the alpha 1-agonist methoxamine. Only compound 3b exhibited significan
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8b185260b779ba62c7fd423aaa30abdf
https://doi.org/10.1021/jm00389a023
https://doi.org/10.1021/jm00389a023
Autor:
Thomas N. Riley, Frank W. Crawford
Publikováno v:
Journal of Pharmaceutical Sciences. 65:544-547
Several series of N, N ‐diaralkyl‐ and N ‐aryloxyalkyl‐ N ‐aralkyl‐β‐haloethylamines were synthesized containing centers of chirality in the aralkyl substituent and in the β‐haloethyl moiety to study the stereoselectivity of α‐ad
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4ff59aeb2efbd8cdfe3a3e0803c467c3
https://doi.org/10.1002/jps.2600650416
https://doi.org/10.1002/jps.2600650416
Autor:
Thomas N. Riley, Jerome R. Bagley
Publikováno v:
Journal of Heterocyclic Chemistry. 19:485-488
In an attempt to investigate stereochemical requirements of antagonists of the histamine H2-receptor, tropane analogues of cimetidine and metiamide have been synthesized possessing axial and equatorial N-methylthiourea and N-methyl-N-cyanoguanidine m
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8f0fbdce2e11bef89f70e9e2eb9e7be9
https://doi.org/10.1002/jhet.5570190307
https://doi.org/10.1002/jhet.5570190307
Autor:
Thomas N. Riley, Jerome R. Bagley
Publikováno v:
Journal of Medicinal Chemistry. 22:1167-1171
Relatively little information is available concerning the influence of conformational factors on the potent analgesic actions of the 4-anilidopiperidines. A series of N-substituted 3 alpha- and 3 beta-(propananilido)nortropanes have been designed, sy
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9de384dc4a276a35a61a9e3ee440712d
https://doi.org/10.1021/jm00196a004
https://doi.org/10.1021/jm00196a004
Publikováno v:
Journal of Pharmaceutical Sciences. 62:983-986
In view of the potency-enhancing effect of methyl substitution of the piperidine ring of the 4-phenylpiperidine analgesics and (he alkylene chain of the acyclic basic anilide analgesics, the 1-methyl, 1-benzyl, and 1-phenylethyl derivatives of 2-meth
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a67b235ab364e62a131a36294915d9de
https://doi.org/10.1002/jps.2600620627
https://doi.org/10.1002/jps.2600620627