Zobrazeno 1 - 10
of 151
pro vyhledávání: '"Thierry, Cresteil"'
Autor:
Angela Zampella, Carmen Festa, Maria Valeria D’Auria, Cecile Debitus, Thierry Cresteil, Simona De Marino
Publikováno v:
Marine Drugs, Vol 9, Iss 6, Pp 1133-1141 (2011)
In our ongoing search for new pharmacologically active leads from Solomon organisms, we have examined the sponge Theonella swinhoei. Herein we report the isolation and structure elucidation of swinholide A (1) and one new macrolide, swinholide J (2).
Externí odkaz:
https://doaj.org/article/198523d1659f4bb4a82ba41df12f9ab0
Autor:
Marie-Lise Bourguet-Kondracki, Cécile Debitus, Sylvain Petek, Thierry Cresteil, Brent R. Copp, Elodie Quévrain, Betty Kientz, Mélanie Roué, Arlette Longeon
Publikováno v:
Marine Drugs, Vol 9, Iss 5, Pp 879-888 (2011)
Indole derivatives including bromoindoles have been isolated from the South Pacific marine sponges Rhopaloeides odorabile and Hyrtios sp. Their structures were established through analysis of mass spectra and 1D and 2D NMR spectroscopic data. Their p
Externí odkaz:
https://doaj.org/article/217c52df19a340a29a440eb779321b67
Publikováno v:
PLoS ONE, Vol 8, Iss 4, p e60895 (2013)
The molecular chaperone CCT/TRiC plays a central role in maintaining cellular proteostasis as it mediates the folding of the major cytoskeletal proteins tubulins and actins. CCT/TRiC is also involved in the oncoprotein cyclin E, the Von Hippel-Lindau
Externí odkaz:
https://doaj.org/article/aefc9d9f3ea44b1bb6474dfc69125643
Autor:
Girish Beedessee, Daniel E. P. Marie, Rob W. M. Van Soest, Prerna Roy, Jay Rovisham Singh Doorga, Avin Ramanjooloo, Thierry Cresteil
Publikováno v:
Hematology and Medical Oncology. 5
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b1de66c5c586b7a76aeb4880208f6f1e
https://doi.org/10.15761/hmo.1000208
https://doi.org/10.15761/hmo.1000208
Autor:
Thierry Cresteil, Embarek Bentouhami, Stéphan Vagner, Laurent Désaubry, Caroline Robert, Giuseppe Campiani, Caroline Welsch, Nora Chouha, Hassan Hammoud, Simone Brogi
Publikováno v:
The Open Medicinal Chemistry Journal. 12:74-83
In our quest to identify inhibitors of the eukaryotic translation initiation factor 4F (eIF4F), we serendipitously discovered a novel cytotoxic agent. Even though this compound did not inhibit translation, we explored the structural requirements for
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::23283f7584d05a65b150e84d3d64c89f
https://doi.org/10.2174/1874104501812010074
https://doi.org/10.2174/1874104501812010074
Autor:
Jean-Pierre Majoral, Régis Laurent, Sonia Ladeira, Mosto Bousmina, Eligia M. Szewczyk, Maria Bryszewska, Elzbieta Pedziwiatr-Werbicka, Anne-Marie Caminade, Serge Mignani, Thierry Cresteil, Nabil El Brahmi, Saïd El Kazzouli
Publikováno v:
Molecular Pharmaceutics
Molecular Pharmaceutics, American Chemical Society, 2017, 14 (11), pp.4087-4097. ⟨10.1021/acs.molpharmaceut.7b00771⟩
Molecular Pharmaceutics, American Chemical Society, 2017, 14 (11), pp.4087-4097. ⟨10.1021/acs.molpharmaceut.7b00771⟩
International audience; Original metallophosphorus dendrimers (generation 3, 48 terminal groups) have been prepared via the complexation of phosphorus dendrimers bearing imino-pyridino end groups with Au(III) or with both Au(III) and Cu(II). The comp
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5803362ac3b7bd72cbdf8514f46e840c
https://doi.org/10.1021/acs.molpharmaceut.7b00771
https://doi.org/10.1021/acs.molpharmaceut.7b00771
Autor:
Dong Wang, Embarek Bentouhami, Canan G. Nebigil, Amel Djehal, Hassan Hammoud, Laurent Désaubry, Mohammad Krayem, Ahmad Najem, Thierry Cresteil, Peng Yu, Ghanem Elias Ghanem
Publikováno v:
European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, Elsevier, 2018, 155, pp.880-888. ⟨10.1016/j.ejmech.2018.06.052⟩
European Journal of Medicinal Chemistry, Elsevier, 2018, 155, pp.880-888. ⟨10.1016/j.ejmech.2018.06.052⟩
Prohibitins 1 and 2 (PHB1/2) are scaffold proteins that are involved in both melanogenesis and oncogenic pathways. We hypothesized that a PHB1 ligand, melanogenin, may display anti-cancer effects in addition to its known melanogenic activity in melan
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ec8b66e4b1da253ddf42a9877f19b012
https://hal.archives-ouvertes.fr/hal-03014913
https://hal.archives-ouvertes.fr/hal-03014913
Publikováno v:
Phosphorous Dendrimers in Biology and Nanomedicine: Syntheses, Characterization, and Properties
Caminade, A.-M. and Turrin, C.-O. and Majoral, J.-P. Phosphorous Dendrimers in Biology and Nanomedicine: Syntheses, Characterization, and Properties, 9, Pan Stanford Publishing, pp.245-264, 2018, 978-9-814-77433-8
Phosphorus Dendrimers in Biology and Nanomedicine ISBN: 9781315110851
Caminade, A.-M. and Turrin, C.-O. and Majoral, J.-P. Phosphorous Dendrimers in Biology and Nanomedicine: Syntheses, Characterization, and Properties, 9, Pan Stanford Publishing, pp.245-264, 2018, 978-9-814-77433-8
Phosphorus Dendrimers in Biology and Nanomedicine ISBN: 9781315110851
International audience
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::22fe0288d918bc1f99ac179ba27b0263
https://hal.archives-ouvertes.fr/hal-02042500
https://hal.archives-ouvertes.fr/hal-02042500
Publikováno v:
Oncology
Oncology, Karger, 2018, 94 (5), pp.324-328. ⟨10.1159/000486680⟩
Oncology, Karger, 2018, 94 (5), pp.324-328. ⟨10.1159/000486680⟩
International audience; The metallo-phosphorus dendrimer 1G3-Cu (generation 3 dendrimer bearing 48 conjugated copper(II) on its surface) has antiproliferative activity related to its capacity to activate Bax translocation. In the present study, we ev
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::92d38b905747ddd497b55e3dc7bd6563
https://hal.archives-ouvertes.fr/hal-01957977
https://hal.archives-ouvertes.fr/hal-01957977
Autor:
Serge M. Mignani, Nabil El Brahmi, Saïd El Kazzouli, Regis Laurent, Sonia Ladeira, Anne-Marie Caminade, Elzbieta Pedziwiatr-Werbicka, Eligia M. Szewcyk, Maria Bryszewska, Mosto M. Bousmina, Thierry Cresteil, Jean Pierre Majoral
Original metallophosphorus dendrimers (generation 3, 48 terminal groups) have been prepared via the complexation of phosphorus dendrimers bearing imino-pyridino end groups with Au(III) or with both Au(III) and Cu(II). The complexation of the dendrime
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=od______2659::ef4be0b03ef3c9fe948f67196d5c9311
https://zenodo.org/record/2707730
https://zenodo.org/record/2707730