Zobrazeno 1 - 10
of 19
pro vyhledávání: '"Thais Regina Ferreira de Melo"'
Autor:
Beatriz Silva Urias, Aline Renata Pavan, Gabriela Ribeiro Albuquerque, Igor Muccilo Prokopczyk, Tânia Mara Ferreira Alves, Thais Regina Ferreira de Melo, Geraldo Rodrigues Sartori, João Hermínio Martins da Silva, Chung Man Chin, Jean Leandro Dos Santos
Publikováno v:
Pharmaceuticals, Vol 15, Iss 10, p 1260 (2022)
Histone deacetylases (HDAC) are epigenetic enzymes responsible for repressing gene expression through the deacetylation of histone lysine residues. Therefore, inhibition of HDACs has become an interesting approach for the treatment of several disease
Externí odkaz:
https://doaj.org/article/e217a6e15fa74663bcfd8c700da2588a
Autor:
Thais Regina Ferreira de Melo, Rafael Consolin Chelucci, Maria Elisa Lopes Pires, Luiz Antonio Dutra, Karina Pereira Barbieri, Priscila Longhin Bosquesi, Gustavo Henrique Goulart Trossini, Man Chin Chung, Jean Leandro dos Santos
Publikováno v:
International Journal of Molecular Sciences, Vol 15, Iss 4, Pp 5821-5837 (2014)
A series of anti-inflammatory derivatives containing an N-acyl hydrazone subunit (4a–e) were synthesized and characterized. Docking studies were performed that suggest that compounds 4a–e bind to cyclooxygenase (COX)-1 and COX-2 isoforms, but wit
Externí odkaz:
https://doaj.org/article/d58cefcfc6fe415badc1ca4d8f450886
Autor:
Rafael Consolin Chelucci, Luiz Antônio Dutra, Maria Elisa Lopes Pires, Thais Regina Ferreira de Melo, Priscila Longhin Bosquesi, Man Chin Chung, Jean Leandro dos Santos
Publikováno v:
Molecules, Vol 19, Iss 2, Pp 2089-2099 (2014)
Nonsteroidal anti-inflammatory drugs (NSAIDs) 1–5 containing an N-acyl hydrazone subunit were prepared and their antiplatelet and antithrombotic activities assessed in vitro and in vivo. Compounds 1–5 inhibited the platelet aggregation induced by
Externí odkaz:
https://doaj.org/article/e94f9980cf8b4224ad5a42ffb4507e84
Autor:
Daniela Hartmann Jornada, Guilherme Felipe dos Santos Fernandes, Diego Eidy Chiba, Thais Regina Ferreira de Melo, Jean Leandro dos Santos, Man Chin Chung
Publikováno v:
Molecules, Vol 21, Iss 1, p 42 (2015)
Prodrug design is a widely known molecular modification strategy that aims to optimize the physicochemical and pharmacological properties of drugs to improve their solubility and pharmacokinetic features and decrease their toxicity. A lack of solubil
Externí odkaz:
https://doaj.org/article/e28377444f3344d697c7bcaac8bd73a4
Autor:
Thais Regina Ferreira de Melo, Guilherme Felipe dos Santos Fernandes, Brian M. Dulmovits, Cristiane Maria de Souza, Lionel Blanc, Yousef Al Abed, Jean Leandro dos Santos, Minghzu He, Carolina Lanaro, Fernando Ferreira Costa, Man Chin Chung
Publikováno v:
Scopus
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Bioorg Chem
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Bioorg Chem
Made available in DSpace on 2021-06-25T10:32:36Z (GMT). No. of bitstreams: 0 Previous issue date: 2021-09-01 Fetal hemoglobin (HbF) induction constitutes a valuable and validated approach to treat the symptoms of sickle cell disease (SCD). Here, we s
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::489327c495a5f43c4ab434e4120014a8
Publikováno v:
Revista Nordestina de História do Brasil. 1:141-161
This article proposes a study on the debate on the issue of secondary education in the years 1920 and 1930. In the perspective of locating and problematizing the place of the school discipline history in this debate, which occurs in the context of th
Autor:
Fernando Ferreira Costa, Shobha Yerigenahally, Carolina Lanaro, Abdullah Kutlar, Marlene F. Wade, Steffen E. Meiler, Carla F. Franco-Penteado, Fábio H. Silva, Chung Man Chin, Jean Leandro dos Santos, Kleber Yotsumoto Fertrin, Thais Regina Ferreira de Melo
Publikováno v:
Scopus
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Made available in DSpace on 2018-12-11T16:50:49Z (GMT). No. of bitstreams: 0 Previous issue date: 2017-01-01 Fetal hemoglobin (HbF) induction by hydroxyurea (HU) therapy is associated with decreased morbidity and mortality in sickle cell anemia (SCA)
Publikováno v:
Revista Brasileira de Educação, Volume: 24, Article number: e240030, Published: 05 AUG 2019
Revista Brasileira de Educação v.24 2019
Revista Brasileira de Educação
Associação Nacional de Pós-Graduação e Pesquisa em Educação (ANPEd)
instacron:EAA
Revista Brasileira de Educação v.24 2019
Revista Brasileira de Educação
Associação Nacional de Pós-Graduação e Pesquisa em Educação (ANPEd)
instacron:EAA
RESUMO Este artigo apresenta análises e alguns dos resultados de pesquisa sobre as contribuições do Instituto Histórico e Geográfico Brasileiro (IHGB) para a educação. Os temas discutidos estão relacionados aos caminhos para a construção de
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a335627c6668856c01e481aaa37a2645
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S1413-24782019000100228&lng=en&tlng=en
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S1413-24782019000100228&lng=en&tlng=en
Autor:
Konstantin Chegaev, Fernando Ferreira Costa, Chutima Kumkhaek, Ticiana Sidorenko de Oliveira Capote, Jean Leandro dos Santos, Roberta Fruttero, Thais Regina Ferreira de Melo, Man Chin Chung, Rafael Consolin Chelucci, Carolina Lanaro, Karina Pereira Barbieri, Iracilda Zeppone Carlos, Griffin P. Rodgers, Guilherme Felipe dos Santos Fernandes, Fernanda Coelho, Sisi Marcondes, Maria Elisa Lopes Pires, Stefano Guglielmo
Publikováno v:
Scopus
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Repositório Institucional da UNESP
Universidade Estadual Paulista (UNESP)
instacron:UNESP
Made available in DSpace on 2018-12-11T17:37:51Z (GMT). No. of bitstreams: 0 Previous issue date: 2018-06-25 N-oxide derivatives 5(a-b), 8(a-b), and 11(a-c) were designed, synthesized and evaluated in vitro and in vivo as potential drugs that are abl
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa67192e62d6598f778912b5ba9c54e5
Autor:
Thais Regina Ferreira de Melo, Karina Pereira Barbieri, Suzana Madeira Diório, Rafael Consolin Chelucci, Jean Leandro dos Santos, Man Chin Chung, Dejair Caetano do Nascimento, I. Z. Carlos, Patrícia Sammarco Rosa, Paulo Renato Yamasaki, Andréa de Faria Fernandes Belone, Marisa Campos Polesi Placeres
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 24:3084-3087
We synthesized a series of novel dapsone-thalidomide hybrids (3a-i) by molecular hybridization and evaluated their potential for the treatment of type 2 leprosy reactions. All of the compounds had analgesic properties. Compounds 3c and 3h were the mo