Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Tetsuro Ohgami"'
Autor:
Kenji Sudo, Masao Matsuoka, Hiroshi Inoue, Shunji Kageyama, Toshifumi Hatta, Hiroshi Suzuki, Yasuaki Shimizu, Osamu Yamamoto, Mitsuaki Ohta, Masaya Orita, Naoyuki Masuda, Tetsuro Ohgami, Masahiro Fujii, Eiichi Kodama
Publikováno v:
Scopus-Elsevier
Background: YM-215389 and YM-228855 are thiazolidenebenzenesulfonamide (TBS) derivatives and novel non-nucleoside reverse transcriptase inhibitors (NNRTIs) that inhibit not only wild-type, but also the K103N- and Y181C-substituted reverse transcripta
Autor:
Ayako Moritomo, Mitsuaki Ohta, Shunji Kageyama, Toru Kontani, Osamu Yamamoto, Naoyuki Masuda, Tetsuro Ohgami, Masahiro Fujii
Publikováno v:
Synthetic Communications. 35:2305-2316
Various N‐3‐alkylated thiazolidenesulfonamide derivatives were efficiently prepared by the direct endo‐selective alkylation of thiazolylsulfonamides. The effects of different bases and solvents were investigated, and the NaH–THF combination w
Autor:
Masatoshi Fujiwara, Tetsuro Ohgami, Shiro Shigeta, Jiro Fujiyasu, Yasuaki Shimizu, Osamu Yamamoto, Ayako Moritomo, Toshifumi Hatta, Naoyuki Masuda, Masanori Baba, Toru Kontani, Masahiro Fujii, Hiroyuki Kurihara, Kenji Sudo, Mitsuaki Ohta, Eiichi Kodama, Masao Matsuoka, Shunji Kageyama, Hironobu Koga, Masaya Orita, Hiroshi Inoue, Masafumi Shintani, Tomoyuki Yokota, Hiroshi Suzuki
Publikováno v:
Bioorganicmedicinal chemistry. 13(4)
In a previous study, we described the structure–activity relationships (SARs) for a series of thiazolidenebenzenesulfonamide derivatives. These compounds were found to be highly potent inhibitors of the wild type (WT) and Y181C mutant reverse trans
Autor:
Masaya Orita, Tomoyuki Yokota, Hiroshi Suzuki, Toru Kontani, Hironobu Koga, Masao Matsuoka, Ayako Moritomo, Kenji Sudo, Tetsuro Ohgami, Hideaki Nakahara, Masahiro Fujii, Shunji Kageyama, Osamu Yamamoto, Masanori Baba, Yasuaki Shimizu, Naoyuki Masuda, Hiroyuki Kurihara, Hiroshi Inoue, Jiro Fujiyasu, Toshifumi Hatta, Eiichi Kodama, Masatoshi Fujiwara, Mitsuaki Ohta, Shiro Shigeta
Publikováno v:
Bioorganicmedicinal chemistry. 12(23)
A random high-throughput screening (HTS) program to discover novel nonnucleoside reverse transcriptase inhibitors (NNRTIs) has been carried out with MT-4 cells against a nevirapine-resistant virus, HIV-1 IIIB-R . The primary hit, a thiazolidenebenzen
Publikováno v:
ChemInform. 32
Publikováno v:
Carbohydrate research. 329(2)
Three kanamycin A analogs containing 6-amino-6-deoxyglycofuranoses have been prepared as candidates for potential activity against resistant bacteria producing 6′- N -acetyltransferase. They are 4- O -(6-amino-3,5,6-trideoxy-α- d -, -β- d -, and