Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Tamako Nomura"'
Autor:
Yoshikazu Tasaki, Tokio Yamaguchi, Mitsuyuki Matsumoto, Shoko Tada, Junya Ohmori, Kazuyuki Hidaka, Tamako Nomura, Shinji Usuda
Publikováno v:
British Journal of Pharmacology. 117:1625-1632
1. We investigated some neurochemical properties of a novel benzamide, YM-43611, [(S)-N-(1-benzyl-3-pyrrolidinyl)-5-chloro-4-cyclopropylcarbonylamino+ ++-2- methoxybenzamide] in comparison with putative D2-like receptor antagonists using both rat and
Autor:
Tokio Yamaguchi, Tamako Nomura, Shin-ichi Tsukamoto, Ryo Naito, Toshiyasu Mase, Tomoyuki Yasunaga, Toru Kontani
Publikováno v:
ChemInform. 28
A series of N-[2-[(substituted chroman-8-yl)oxy]ethyl]-4-(4-methoxyphenyl)butylamines was prepared and examined for their 5-HT1A receptor antagonist activity. The parent compound 3a and seven analo...
Autor:
Toshiyasu Mase, Ryo Naito, Tokio Yamaguchi, Shin-ichi Tsukamoto, Takenori Kimura, Tamako Nomura, Tomoyuki Yasunaga, Toru Kontani, T. Wanibuchi, Hiroshi Yamashita
Publikováno v:
ChemInform. 29
Autor:
Toru Kontani, Tamako Nomura, Takenori Kimura, Tokio Yamaguchi, Fumikazu Wanibuchi, Tomoyuki Yasunaga, Toshiyasu Mase, Shin-ichi Tsukamoto, Ryo Naito, Hiroshi Yamashita
Publikováno v:
Journal of medicinal chemistry. 41(15)
A series of novel 6-fluorochroman derivatives was prepared and evaluated as antagonists for the 5-HT1A receptor. N-2-[[(6-Fluorochroman-8-yl)oxy]ethyl]-4-(4-methoxyphenyl)butylami ne (3; J. Med. Chem. 1997, 40, 1252-1257) was chosen as a lead, and st
Autor:
Tokio Yamaguchi, Tamako Nomura, Tomoyuki Yasunaga, Ryo Naito, Toru Kontani, Shin-ichi Tsukamoto, Toshiyasu Mase
Publikováno v:
Journal of medicinal chemistry. 40(8)
A series of N-[2-[(substituted chroman-8-yl)oxy]ethyl]-4-(4-methoxyphenyl)butylamines was prepared and examined for their 5-HT1A receptor antagonist activity. The parent compound 3a and seven analogs bearing five kinds of substituents on the chroman
Autor:
Yasuharu Kimura, Yutaka Kondou, Yasushi Ikeda, Kazuhiro Momose, Hiraku Akiho, Tokio Yamaguchi, Mitsuyuki Matsumoto, Junji Togami, Masamichi Okada, Tamako Nomura
Publikováno v:
The Journal of biological chemistry. 271(44)
Neuropeptide Y (NPY), peptide YY (PYY), and pancreatic polypeptide (PP) belong to a family of structurally related peptides which have numerous functions in both neural and endocrine signaling. By homology screening, we cloned a novel gene sharing th