Zobrazeno 1 - 10
of 27
pro vyhledávání: '"Takeshi Terasawa"'
Autor:
Hiroshi Inami, Tsuyoshi Mizutani, Junko Watanabe, Hisashi Hayashida, Tomonori Ito, Takeshi Terasawa, Toru Kontani, Hiroaki Yamagishi, Hiroyuki Usuda, Naohiro Aoyama, Emiko Imamura, Takeshi Ishikawa
Publikováno v:
Bioorganic & Medicinal Chemistry. 87:117302
Publikováno v:
Journal of Pediatric Surgery. 53:223-226
Aim Although many approaches to esophageal replacement have been investigated, these efforts have thus far only met limited success. In-body-tissue-engineered connective tissue tubes have been reported to be effective as vascular replacement grafts.
Autor:
Takeshi Terasawa, Hisashi Takasugi, Hirokazu Tanaka, Satoru Matsumoto, Ayako Nakamura, Hirofumi Yamamoto, Yoshimi Matsumoto, Kohji Kawabata, Shuichi Tawara
Publikováno v:
Bioorganic & Medicinal Chemistry. 9:465-475
A series of 7β-[( Z )-2-(2-aminothiazol-4-yl)-2-hydroxyiminoacetamido]-3-(heteroarylmethylthio)cephalosporins was designed, synthesized and evaluated for antibacterial activity and oral absorption in rats. Antibacterial activity was markedly influen
Autor:
Takeshi Terasawa, Kohji Kawabata, Hirofumi Yamamoto, Satoru Matsumoto, Shuichi Tawara, Kazuo Sakane, Ayako Nakamura, Yoshimi Matsumoto
Publikováno v:
Bioorganic & Medicinal Chemistry. 8:1159-1170
A series of 7beta-[(Z)-2-(2-aminothiazol-4-yl)-2-hydroxyiminoacetamid o]cephalosporins having a pyridine ring connected through various spacer moieties at the C-3 position was designed and synthesized and evaluated for antibacterial activity and oral
Autor:
Takeshi, Terasawa
Publikováno v:
雲雀野 = The Lark Hill. 21:1-17
Autor:
Hiroyuki Hagihara, Akira Tanaka, Hirokazu Tanaka, Masae Sawada, Masaharu Hashimoto, Yuri Sakuma, Hisashi Takasugi, Noriko Ishibe, Takeshi Terasawa
Publikováno v:
Journal of Medicinal Chemistry. 41:4408-4420
A series of N-alkyl-N-[(fluorophenoxy)benzyl]-N'-arylureas were prepared and evaluated for their ability to inhibit intestinal acyl-CoA:cholesterol O-acyltransferase and to inhibit accumulation of cholesteryl esters in macrophages in vitro. In vivo h
Autor:
Masae Sawada, Hisashi Takasugi, Takeshi Terasawa, Noriko Ishibe, Yuri Sakuma, Hirokazu Tanaka, Hiroyuki Hagihara, Akira Tanaka
Publikováno v:
Journal of Medicinal Chemistry. 41:2390-2410
A series of N-alkyl-N-(heteroaryl-substituted benzyl)-N'-arylurea and related derivatives represented by 2 and 3 have been prepared and evaluated for their ability to inhibit acyl-CoA:cholesterol O-acyltransferase in vitro and to lower plasma cholest
Autor:
Noriko Ishibe, Yuri Sakuma, Hisashi Takasugi, Hiroyuki Hagihara, Masae Sawada, Akira Tanaka, Hirokazu Tanaka, Takeshi Terasawa, Takayoshi Kinoshita
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 8:81-86
The synthesis, single crystal X-ray structural analysis, and biological activity of FR186054 (2c), a new, potent, orally efficacious inhibitor of acyl-CoA:cholesterol O-acyltransferase (ACAT), containing a pyrazole ring are described. This compound d
Autor:
Takeshi, Terasawa, Tsutomu, Aoyama
Publikováno v:
雲雀野 = The Lark Hill. 15:27-42
Autor:
Noriko Ishibe, Hiroyuki Hagihara, Masae Sawada, Akira Tanaka, Hirokazu Tanaka, Takeshi Terasawa, Yuri Sakuma, Takayoshi Kinoshita, Hisashi Takasugi
Publikováno v:
ChemInform. 29
The synthesis, single crystal X-ray structural analysis, and biological activity of FR186054 (2c), a new, potent, orally efficacious inhibitor of acyl-CoA:cholesterol O-acyltransferase (ACAT), containing a pyrazole ring are described. This compound d