Zobrazeno 1 - 10
of 1 095
pro vyhledávání: '"TOURWÉ, D."'
Autor:
De Neve J; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, 1050 Brussels, Belgium., Breault É; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Previti S; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, 1050 Brussels, Belgium., Vangeloven E; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, 1050 Brussels, Belgium., Loranger B; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Chartier M; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Brouillette R; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Lanoie A; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Holleran BJ; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Longpré JM; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Gendron L; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Tourwé D; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, 1050 Brussels, Belgium., Sarret P; Institut de Pharmacologie de Sherbrooke, Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Université de Sherbrooke, 3001, 12e Avenue Nord, J1H 5N4 Sherbrooke, Quebec, Canada., Ballet S; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, 1050 Brussels, Belgium.
Publikováno v:
ACS pharmacology & translational science [ACS Pharmacol Transl Sci] 2024 Aug 19; Vol. 7 (9), pp. 2784-2798. Date of Electronic Publication: 2024 Aug 19 (Print Publication: 2024).
Autor:
Previti S; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Brussels, Belgium.; Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, Messina, Italy., Desgagné M; Department of Pharmacology-Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, Sherbrooke, Quebec, Canada., Tourwé D; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Brussels, Belgium., Cavelier F; Institut des Biomolécules Max Mousseron, IBMM, UMR 5247, CNRS, Université de Montpellier, ENSCM, Montpellier, France., Sarret P; Department of Pharmacology-Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, Sherbrooke, Quebec, Canada., Ballet S; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Brussels, Belgium.
Publikováno v:
Journal of peptide science : an official publication of the European Peptide Society [J Pept Sci] 2023 Jun; Vol. 29 (6), pp. e3471. Date of Electronic Publication: 2023 Jan 11.
Autor:
Gimenez LE; Life Sciences Institute, University of Michigan, Ann Arbor, Michigan 48109, United States., Martin C; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, Brussels B-1050, Belgium., Yu J; iHuman Institute, ShanghaiTech University, Ren Building, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China., Hollanders C; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, Brussels B-1050, Belgium., Hernandez CC; Life Sciences Institute, University of Michigan, Ann Arbor, Michigan 48109, United States., Wu Y; iHuman Institute, ShanghaiTech University, Ren Building, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China., Yao D; iHuman Institute, ShanghaiTech University, Ren Building, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China., Han GW; Departments of Biological Sciences and Chemistry, Bridge Institute, USC Michelson Center for Convergent Bioscience, University of Southern California, Los Angeles, California 90089, United States., Dahir NS; Life Sciences Institute, University of Michigan, Ann Arbor, Michigan 48109, United States.; Department of Molecular and Integrative Physiology, School of Medicine, University of Michigan, Ann Arbor, Michigan 48109, United States., Wu L; iHuman Institute, ShanghaiTech University, Ren Building, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China., Van der Poorten O; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, Brussels B-1050, Belgium., Lamouroux A; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, Brussels B-1050, Belgium., Mannes M; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, Brussels B-1050, Belgium., Zhao S; iHuman Institute, ShanghaiTech University, Ren Building, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China., Tourwé D; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, Brussels B-1050, Belgium., Stevens RC; iHuman Institute, ShanghaiTech University, Ren Building, 393 Middle Huaxia Road, Pudong, Shanghai 201210, China., Cone RD; Life Sciences Institute, University of Michigan, Ann Arbor, Michigan 48109, United States.; Department of Molecular and Integrative Physiology, School of Medicine, University of Michigan, Ann Arbor, Michigan 48109, United States.; Department of Molecular, Cellular, and Developmental Biology, College of Literature, Science, and the Arts, University of Michigan, Ann Arbor, Michigan 48109, United States., Ballet S; Research Group of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, Brussels B-1050, Belgium.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2024 Feb 22; Vol. 67 (4), pp. 2690-2711. Date of Electronic Publication: 2024 Feb 12.
Publikováno v:
In Bioorganic & Medicinal Chemistry 2005 13(21):6070-6082
Publikováno v:
In Bioorganic & Medicinal Chemistry 2005 13(12):3987-3992
A 3-step methodology for the synthesis of 1,5-benzothiazepin-4(5H)-one dipeptidomimetics has been elaborated via an Ugi-4CR followed by a S-trityl deprotection and an intramolecular Cu(i)-catalyzed Ullmann condensation with moderate to good yields. I
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=od______3848::94fc0cfae61c056849349a42bea3dd4a
https://doi.org/10.1039/c7ob03094k
https://doi.org/10.1039/c7ob03094k
Autor:
Wachter, R., Chris de Graaf, Keresztes, C., Vandormael, B., Ballet, S., Toth, G., Rognan, D., Tourwé, D.
Publikováno v:
de Wachter, R, de Graaf, C, Keresztes, C, Vandormael, B, Ballet, S, Toth, G, Rognan, D & Tourwé, D 2011, ' Synthesis, biological evaluation and automated docking of constrained analogs of the opioid peptide H-Dmt-D-AlapPhe-Gly-NH2 using the 4-or 5-metyl substsituted 4-amino-1,2,3,4-tetrahydro-2-benzazepin-3-one scaffold. ', Journal of Medicinal Chemistry, vol. 54, pp. 3384-3393 .
Journal of Medicinal Chemistry, 54, 3384-3393. American Chemical Society
Vrije Universiteit Amsterdam
Journal of Medicinal Chemistry, 54, 3384-3393. American Chemical Society
Vrije Universiteit Amsterdam
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::c1ab2cec994469a07c3e8339dcf19cf7
https://hdl.handle.net/1871.1/95c629e8-0c0d-4e58-8c86-6c0c187ac193
https://hdl.handle.net/1871.1/95c629e8-0c0d-4e58-8c86-6c0c187ac193
Autor:
Tourwé D; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, 1050 Brussels, Belgium. Electronic address: datourwe@vub.be., Tsiailanis AD; Laboratory of Organic Chemistry and Biochemistry, Department of Chemistry, University of Ioannina, Ioannina 45110, Greece., Parisis N; Laboratory of Organic Chemistry and Biochemistry, Department of Chemistry, University of Ioannina, Ioannina 45110, Greece., Hirmiz B; Department of Biochemistry and Molecular Biology, Monash University, Clayton, VIC 3800, Australia., Del Borgo M; Biomedicine Discovery Institute and Department of Pharmacology, Monash University, Clayton, VIC 3800, Australia., Aguilar MI; Department of Biochemistry and Molecular Biology, Monash University, Clayton, VIC 3800, Australia., Van der Poorten O; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, 1050 Brussels, Belgium., Ballet S; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel, Pleinlaan 2, 1050 Brussels, Belgium. Electronic address: Steven.Ballet@vub.be., Widdop RE; Biomedicine Discovery Institute and Department of Pharmacology, Monash University, Clayton, VIC 3800, Australia., Tzakos AG; Laboratory of Organic Chemistry and Biochemistry, Department of Chemistry, University of Ioannina, Ioannina 45110, Greece; University Research Center of Ioannina (URCI), Institute of Materials Science and Computing, Ioannina, Greece. Electronic address: atzakos@uoi.gr.
Publikováno v:
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2021 Jul 01; Vol. 43, pp. 128086. Date of Electronic Publication: 2021 May 07.
Akademický článek
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Autor:
De Neve J; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel Brussels Belgium steven.ballet@vub.be., Barlow TMA; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel Brussels Belgium steven.ballet@vub.be., Tourwé D; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel Brussels Belgium steven.ballet@vub.be., Bihel F; Laboratoire d'Innovation Thérapeutique, Faculté de Pharmacie, UMR 7200, CNRS Université de Strasbourg Illkirch France., Simonin F; Biotechnologie et Signalisation Cellulaire, UMR 7242, CNRS, Université de Strasbourg Illkirch France., Ballet S; Research Group of Organic Chemistry, Departments of Chemistry and Bioengineering Sciences, Vrije Universiteit Brussel Brussels Belgium steven.ballet@vub.be.
Publikováno v:
RSC medicinal chemistry [RSC Med Chem] 2021 Apr 21; Vol. 12 (6), pp. 828-870. Date of Electronic Publication: 2021 Apr 21 (Print Publication: 2021).