Zobrazeno 1 - 7
of 7
pro vyhledávání: '"T B, Stensbøl"'
Autor:
S, Natesan, S, Ashworth, J, Nielsen, S-P, Tang, C, Salinas, S, Kealey, J B, Lauridsen, T B, Stensbøl, R N, Gunn, E A, Rabiner, S, Kapur
Publikováno v:
Translational Psychiatry
A number of phosphodiesterase 10A (PDE10) inhibitors are about to undergo clinical evaluation for their efficacy in treating schizophrenia. As phosphodiesterases are in the same signalling pathway as dopamine D2 receptors, it is possible that prior a
Autor:
T N, Johansen, T B, Stensbøl, B, Nielsen, S B, Vogensen, K, Frydenvang, F A, Sløk, H, Bräüner-Osborne, U, Madsen, P, Krogsgaard-Larsen
Publikováno v:
Chirality. 13(9)
We have previously described (RS)-2-amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA) as a potent agonist at the (RS)-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptor subtype of (S)-glutamic acid (Glu) receptors.
Publikováno v:
Archiv der Pharmazie. 334(2)
We have previously reported the synthesis and pharmacological characterization of analogues of 2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA, 1a), in which the methyl group was replaced by a phenyl group (APPA, 1b) or heteroaryl gro
Autor:
S B, Vogensen, H S, Jensen, T B, Stensbøl, K, Frydenvang, B, Bang-Andersen, T N, Johansen, J, Egebjerg, P, Krogsgaard-Larsen
Publikováno v:
Chirality. 12(10)
We have previously shown that (RS)-2-amino-3-[3-hydroxy-5-(2-methyl-2H-tetrazol-5-yl)isoxazol -4-yl] propionic acid (2-Me-Tet-AMPA) is a selective agonist at (RS)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic acid (AMPA) receptors, markedly mo
Autor:
E H, Møller, J, Egebjerg, L, Brehm, T B, Stensbøl, T N, Johansen, U, Madsen, P, Krogsgaard-Larsen
Publikováno v:
Chirality. 11(10)
The phosphono amino acid, (RS)-2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl+ ++]propio nic acid (ATPO), is a structural hybrid between the NMDA antagonist (RS)-2-amino-7-phosphonoheptanoic acid (AP7) and the AMPA and GluR5 agonist, (RS)-
Autor:
T B, Stensbøl, F A, Sløk, J, Trometer, S, Hurt, B, Ebert, C, Kjøller, J, Egebjerg, U, Madsen, N H, Diemer, P, Krogsgaard-Larsen
Publikováno v:
European journal of pharmacology. 373(2-3)
(RS)-2-Amino-3-(3-carboxy-5-methyl-4-isoxazolyl)propionic acid (ACPA), which is a potent and selective agonist at (RS)-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid (AMPA) receptors, has previously been shown to desensitize AMPA receptors
Autor:
G. De Sarro, Ulf Madsen, M. De Amici, Paola Conti, T. B. Stensbøl, Hans Bräuner-Osborne, C. De Micheli
Publikováno v:
Journal of medicinal chemistry. 41(20)