Zobrazeno 1 - 10 of 183 pro vyhledávání: '"T, de Paulis"'
1
Synthesis and 5-HT-3 receptor binding activity of 5-[125I]iodo-2,3-dimethoxy-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamide and its 5-halogen-2-alkoxyl homologues
Autor: B. L. Trivedi, T. De Paulis, William A. Hewlett, Dennis E. Schmidt, Michael H. Ebert, N. S. Mason
Publikováno v: European Journal of Medicinal Chemistry. 32:385-396
Summary ( S )-5-Iodo-2,3-dimethoxy- N -(1-azabicyclo[2.2.2]oct-3-yl)benzamide (MIZAC) was prepared from 5-iodo-2,3-dimethoxybenzoyl chloride and ( S )-3-aminoquinuclidine. [ 125 I]Iodode-stannylation of its corresponding 5-tri- n -butyltin derivative
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::7631ac34a863824971cf57a5aeddcf03
https://doi.org/10.1016/s0223-5234(97)81676-5
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7
ChemInform Abstract: Synthesis and 5-HT-3 Receptor Binding Activity of 5-(125I)Iodo-2,3- dimethoxy-N-(1-azabicyclo(2.2.2)oct-3-yl)benzamide and Its 5-Halogen-2- alkoxyl Homologues
Autor: T. De Paulis, B. L. Trivedi, Dennis E. Schmidt, N. S. Mason, William A. Hewlett, Michael H. Ebert
Publikováno v: ChemInform. 28
Summary ( S )-5-Iodo-2,3-dimethoxy- N -(1-azabicyclo[2.2.2]oct-3-yl)benzamide (MIZAC) was prepared from 5-iodo-2,3-dimethoxybenzoyl chloride and ( S )-3-aminoquinuclidine. [ 125 I]Iodode-stannylation of its corresponding 5-tri- n -butyltin derivative
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::960636caae55561fcf34f1834411d19a
https://doi.org/10.1002/chin.199743273
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9
Preparation of [123I]- and [125I]epidepride: A dopamine D-2 receptor antagonist radioligand
Autor: T. De Paulis, Robert M. Kessler, Dennis E. Schmidt, Jeffery A. Clanton, R. M. Baldwin, Mohammed Ansari, Ronald G. Manning
Publikováno v: Journal of Labelled Compounds and Radiopharmaceuticals. 29:745-751
(S)-(−)-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-[123I]iodo-2,3-dimethoxybenzamide (TDP 517) (proposed generic name, [123I]epidepride) is the iodine-123 substituted analogue of isoremoxipride (FLB 457), both of which are very potent dopamine D-2 antago
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::b2d7079bd08fc715833feb1cd41a9a34
https://doi.org/10.1002/jlcr.2580290703
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10
Potential antipsychotic agents. 6. Synthesis and antidopaminergic properties of substituted N-(1-benzyl-4-piperidinyl)salicylamides and related compounds. QSAR based design of more active members
Autor: Sven-Ove Ögren, H. Hall, T. De Paulis, Y. Kumar, Rämsby S, Thomas Högberg
Publikováno v: European Journal of Medicinal Chemistry. 25:507-517
A number of substituted 2-methoxybenzamides, with and without 6-hydroxy groups, with 4-piperidinyl side-chains have been synthesized and evaluated for their antidopaminergic properties. The salicylamides were found to require a lipophilic N-substitue
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::192397911585dca1dc407c893728f4ac
https://doi.org/10.1016/0223-5234(90)90145-s
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