Výsledky vyhledávání - "Sunil V. Mali"

Design and synthesis of taxane derivatives of valproic acid as potent and selective cytotoxic agents

Autor: Himaja Malipeddi, Moonjit Das, Sunil V. Mali

Publikováno v: Medicinal Chemistry Research. 25:2512-2520

Resistance to anticancer agents has important implications for cancer chemotherapy. Small changes in chemical structures of cytotoxic agents can alter their biological interactions that can be beneficial in overcoming the drug resistance problem. Val

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::fb1dc8b6b80fa9413055fe2c68e01adc
https://doi.org/10.1007/s00044-016-1635-6

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Synthesis of New (Pyrazol-3-yl)-1,3,4-oxadiazole Derivatives by Unexpected Aromatization During Oxidative Cyclization of 4,5-Dihydro-1H-pyrazole-3-carbohydrazones and Their Biological Activities

Autor: Sunil V. Mali, D. Munirajasekhar, M. Himaja, K. Jagadeesh Prathap

Publikováno v: Journal of Heterocyclic Chemistry. 51:726-732

A series of novel 2-(4-(4-chlorophenyl)-1H-pyrazol-3-yl)-5-(Aryl)-1,3,4-oxadiazoles were synthesized by unexpected aromatization during oxidative cyclization of 4-(4-chlorophenyl)-4,5-dihydro-1H-pyrazole-3-carbohydrazones using chloramine-T as an oxi

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::91d285683bd6a4807e2221ad1507df33
https://doi.org/10.1002/jhet.1765

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A Facile and Efficient Synthesis of 2-(5-(4-Substitutedphenyl)-4, 5-dihydro-3-phenylpyrazol-1-yl)-6-Substitutedbenzothiazoles and Their Biological Studies

Autor: Sunil V. Mali, D. Munirajasekhar, M. Himaja

Publikováno v: Journal of Heterocyclic Chemistry. 51:459-465

A series of new 1-substituted 3, 5-diarylpyrazolines () were synthesized in good yield by both conventional and microwave-assisted synthesis from α, β- unsaturated ketones () in n-butanol and benzothiazole hydrazines (). All the new compounds were

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::42242fb783d44cf8724cc40d8305791b
https://doi.org/10.1002/jhet.1618

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Synthesis, docking and anticancer activity studies of D-proline-incorporated wainunuamide

Autor: A Ranjitha, M. Himaja, Sunil V Mali

Publikováno v: Journal of Chemical Sciences. 124:1049-1055

D-proline-incorporated wainunuamide — a cyclic octapeptide was synthesized and characterized by FTIR, 1H and 13C NMR and Mass spectral analysis. Molecular docking studies were carried out for the designed cyclic octapeptide and the results showed g

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::79421df57bdd78fb503879c15d30fbf3
https://doi.org/10.1007/s12039-012-0301-x

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Facile Synthesis of 3,6-Disubstituted-1,2,4-triazolo-[3,4-b]-1,3,4-thiadiazoles via Oxidative Cyclization ofn-Heteroaryl-Substituted Hydrazones and Their Biological Activity

Autor: K. Jagadeesh Prathap, M. Himaja, Sunil V. Mali

Publikováno v: Journal of Heterocyclic Chemistry. 49:823-828

Fused 3,6-disubstituted triazolothiadiazoles were synthesized in good yield from a rapid and convenient oxidative cyclization of N-heteroaryl-substituted hydrazones promoted by chloramine-T trihydrate at ambient temperature. The structure of the synt

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::d78cf740be4af6462b31bf77bd9eb983
https://doi.org/10.1002/jhet.870

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ChemInform Abstract: A Facile and Efficient Synthesis of 2-(5-(4-Substitutedphenyl)-4,5-dihydro-3-phenylpyrazol-1-yl) -6-substitutedbenzothiazoles and Their Biological Studies

Autor: Sunil V. Mali, M. Himaja, D. Munirajasekhar

Publikováno v: ChemInform. 45

16 Title compounds of type (III) are prepared under microwave irradiation and screened for their antibacterial and anthelmintic activities.

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::ba540462ba1632b1a2649e5720ced491
https://doi.org/10.1002/chin.201435151

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ChemInform Abstract: Facile Synthesis of 3,6-Disubstituted-1,2,4-triazolo-[3,4-b]-1,3,4-thiadiazoles via Oxidative Cyclization of n-Heteroaryl-Substituted Hydrazones and Their Biological Activity

Autor: M. Himaja, K. Jagadeesh Prathap, Sunil V. Mali

Publikováno v: ChemInform. 44

All the title triazolothiadiazoles (IV) (9 examples) and their hydrazone precursors (III) show good antitubercular activity.

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::78b91c7416ac3db19d2106e4e6d23311
https://doi.org/10.1002/chin.201306088

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