Zobrazeno 1 - 10
of 16
pro vyhledávání: '"Sukumar Bepary"'
Publikováno v:
Indonesian Journal of Chemistry, Vol 24, Iss 5, Pp 1541-1555 (2024)
Several 2-phenoxyacetic acid derivatives and their isosteres were synthesized in moderate to high yield (57–96%) for searching newer and safer alternatives to these existing anti-inflammatory agents. The compounds were characterized by 1H-NMR, 13C-
Externí odkaz:
https://doaj.org/article/3ba6231a2e1d4ab1960d9af72ecb2c9f
Publikováno v:
Journal of Molecular Docking, Vol 1, Iss 2 (2021)
Acetamides (S30A1 and S30) were synthesized from benzo[d]thiazol-2-amine and 6-nitrobenzo[d]thiazol-2-amine by direct use of acetic acid instead of acetylating agents. The usual acetylating agents, acetic anhydride and acetyl chloride are very unstab
Externí odkaz:
https://doaj.org/article/843d95d63948448ba392e4620209bd81
Autor:
Shahenul Islam, Tran Quang De, Shamima Akhter, Rahen Mahmuda, Sukumar Bepary, Pranoy Saha, Khadija Akhter Poly, Negar Sultana Shoshi
Publikováno v:
Can Tho University Journal of Science. 12
Resorcinol with its two hydroxyl groups was derivatized in laboratory to observe the anti-inflammatory potential in vitro. Subsequently in silico docking analysis was done for observing the binding modes in cyclooxygenase enzyme to have idea about th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::241685b61d0a8f11e57f056b3d624cc3
https://doi.org/10.22144/ctu.jen.2020.027
https://doi.org/10.22144/ctu.jen.2020.027
Synthesis and evaluation of PI3Kγ enzyme inhibitory activity of Novel (1H-pyrazol-4-yl)methanamines.
Publikováno v:
Thai Journal of Pharmaceutical Sciences. Apr-Jun2016, Vol. 40 Issue 2, p82-86. 5p.
Publikováno v:
Bulletin of the Korean Chemical Society. 37:2054-2057
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d2f51f92a6df4541a941c8834483cf60
https://doi.org/10.1002/bkcs.10994
https://doi.org/10.1002/bkcs.10994
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 26:51-54
Synthesis, SAR study and BACE1 inhibitory activity of (3S,4S)-4-aminopyrrolidine-3-ol derivatives (2) were described. The compound 7c exhibited more inhibition activity than 11a (IC50: 0.05μM vs 0.12μM, respectively), but the latter was more effect
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::66bc4e439432dcdbd2db40bb567c0d7c
https://doi.org/10.1016/j.bmcl.2015.11.033
https://doi.org/10.1016/j.bmcl.2015.11.033
Objective: This study was intended to evaluate the phytochemical, analgesic and anti-inflammatory activity of 70% ethanolic extracts of Ardisia colorata in swiss albino mice and long evans rats. Methods: The ethanolic extract of A. colorata stem and
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1817bae6809583ddadc1dd183be59fa0
Publikováno v:
Synthetic Communications. 44:1876-1880
2-Aminoimidazolidin-4-ones have been synthesized by using di-2-pyridyl thiocarbonate (DPT), taking the thioureas tethered to amides as the starting materials. Both the primary amides and secondary amides have been subjected to this cyclization method
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d348e75358175ea1692b7c1109a6997f
https://doi.org/10.1080/00397911.2013.827724
https://doi.org/10.1080/00397911.2013.827724
Publikováno v:
Bulletin of the Korean Chemical Society. 34:2829-2832
E-mail: yink@pcu.ac.krReceived May 30, 2013, Accepted June 25, 2013Key Words : Phenylpyrazole, PI3 kinase gamma, In vitro assay, SAR, Inhibitory activityPhosphatidylinositol-3-kinase gamma (PI3Kγ), with itscatalytic subunit P110γ and regulatory sub
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e20924d57f055e8bb8aa6aab7343a5e7
https://doi.org/10.5012/bkcs.2013.34.9.2829
https://doi.org/10.5012/bkcs.2013.34.9.2829
Publikováno v:
Bulletin of the Korean Chemical Society. 31:3788-3790
solution using tetramethylsilane as internal standard. Analytical thin-layer chromatography was performed on precoated silica gel plates (0.25-mm 60 F-254 E. Merck). The products were pu rified by flash column chro-matography on silica gel 60 (Merck,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::6bce5022b6923eed392ff1dc62d70cb9
https://doi.org/10.5012/bkcs.2010.31.12.3788
https://doi.org/10.5012/bkcs.2010.31.12.3788