Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Suen Lm"'
Autor:
Tekle-Smith Ma, Infantine, Sackett Dl, Reznik Sk, Casselman Td, Tanis Ps, Leighton J, Williamson Ks, Suen Lm
With an average GI50 value against the NCI panel of 60 human cancer cell lines of 0.12 nM, spongistatin 1 is among the most potent anti-proliferative agents ever discovered rendering it an attractive candidate for development as a payload for antibod
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fc8a27966d1c9e02af0289ebd3288bb6
https://doi.org/10.26434/chemrxiv.5773830.v1
https://doi.org/10.26434/chemrxiv.5773830.v1
Autor:
Suen LM; Department of Chemistry, Columbia University, New York, NY, 10027, USA., Tekle-Smith MA; Department of Chemistry, Columbia University, New York, NY, 10027, USA., Williamson KS; Department of Chemistry, Columbia University, New York, NY, 10027, USA., Infantine JR; Department of Chemistry, Columbia University, New York, NY, 10027, USA., Reznik SK; Department of Chemistry, Columbia University, New York, NY, 10027, USA., Tanis PS; Department of Chemistry, Columbia University, New York, NY, 10027, USA., Casselman TD; Department of Chemistry, Columbia University, New York, NY, 10027, USA., Sackett DL; Eunice Kennedy Shriver National Institute of Child Health and Human Development, National Institutes of Health, Bethesda, MD, 20892, USA. sackettd@mail.nih.gov., Leighton JL; Department of Chemistry, Columbia University, New York, NY, 10027, USA. jll43@columbia.edu.
Publikováno v:
Nature communications [Nat Commun] 2018 Nov 09; Vol. 9 (1), pp. 4710. Date of Electronic Publication: 2018 Nov 09.
Autor:
Sanders JM; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Beshore DC; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Culberson JC; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Fells JI; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Imbriglio JE; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Gunaydin H; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Haidle AM; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Labroli M; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Mattioni BE; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Sciammetta N; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Shipe WD; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Sheridan RP; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Suen LM; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Verras A; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Walji A; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Joshi EM; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States., Bueters T; Modeling & Informatics, ‡Discovery Chemistry, and §Pharmacokinetics, Pharmacodynamics, and Drug Metabolism, Merck & Co., Inc. , Kenilworth, New Jersey 07065, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2017 Aug 24; Vol. 60 (16), pp. 6771-6780. Date of Electronic Publication: 2017 May 05.
Autor:
Suen LM; Department of Chemistry, Columbia University, 3000 Broadway, New York, New York, 10027, USA. ; Tel: (+1) 212-854-4262., Steigerwald ML; Department of Chemistry, Columbia University, 3000 Broadway, New York, New York, 10027, USA. ; Tel: (+1) 212-854-4262., Leighton JL; Department of Chemistry, Columbia University, 3000 Broadway, New York, New York, 10027, USA. ; Tel: (+1) 212-854-4262.
Publikováno v:
Chemical science [Chem Sci] 2013 Jun 01; Vol. 4 (6), pp. 2413-2417.