[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor

Autor: Nebel, Natascha, Strauch, Brigitte, Maschauer, Simone, Lasch, Roman, Rampp, Hannelore, Fehler, Stefanie K., Bock, Leonard R., Hübner, Harald, Gmeiner, Peter, Heinrich, Markus R., Prante, Olaf

Publikováno v: ACS Omega, Vol 2, Iss 12, Pp 8649-8659 (2017)
ACS Omega

18F-Labeled building blocks from the type of [18F]fluorophenylazocarboxylic-tert-butyl esters offer a rapid, mild, and reliable method for the 18F-fluoroarylation of biomolecules. Two series of azocarboxamides were synthesized as potential radioligan

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::41407f02997895a04696aa7aaf3c1bd5
https://opus4.kobv.de/opus4-fau/frontdoor/index/index/docId/10839

Development of 18F-Fluoroglycosylated PSMA-Ligands with Improved Renal Clearance Behavior

Autor: Potemkin, Roman, Strauch, Brigitte, Kuwert, Torsten, Prante, Olaf, Maschauer, Simone

Publikováno v: Molecular Pharmaceutics; March 2020, Vol. 17 Issue: 3 p933-943, 11p

[ ¹⁸ F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor.

Autor: Nebel N; Department of Nuclear Medicine, Molecular Imaging and Radiochemistry, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schwabachanlage 6, Erlangen D-91054, Germany., Strauch B; Department of Nuclear Medicine, Molecular Imaging and Radiochemistry, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schwabachanlage 6, Erlangen D-91054, Germany., Maschauer S; Department of Nuclear Medicine, Molecular Imaging and Radiochemistry, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schwabachanlage 6, Erlangen D-91054, Germany., Lasch R; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schuhstrasse 19, Erlangen D-91052, Germany., Rampp H; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schuhstrasse 19, Erlangen D-91052, Germany., Fehler SK; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schuhstrasse 19, Erlangen D-91052, Germany., Bock LR; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schuhstrasse 19, Erlangen D-91052, Germany., Hübner H; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schuhstrasse 19, Erlangen D-91052, Germany., Gmeiner P; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schuhstrasse 19, Erlangen D-91052, Germany., Heinrich MR; Department of Chemistry and Pharmacy, Medicinal Chemistry, Emil Fischer Center, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schuhstrasse 19, Erlangen D-91052, Germany., Prante O; Department of Nuclear Medicine, Molecular Imaging and Radiochemistry, Friedrich Alexander University Erlangen-Nürnberg (FAU), Schwabachanlage 6, Erlangen D-91054, Germany.

Publikováno v: ACS omega [ACS Omega] 2017 Dec 31; Vol. 2 (12), pp. 8649-8659. Date of Electronic Publication: 2017 Dec 06.