Zobrazeno 1 - 10
of 37
pro vyhledávání: '"Stéphane Krief"'
Autor:
Stéphane Krief, Isabelle Berrebi‐Bertrand, Isabelle Nagmar, Martin Giret, Simon Belliard, David Perrin, Marilyne Uguen, Philippe Robert, Jeanne‐Marie Lecomte, Jean‐Charles Schwartz, Olivier Finance, Xavier Ligneau
Publikováno v:
Pharmacology Research & Perspectives, Vol 9, Iss 5, Pp n/a-n/a (2021)
Abstract Several therapeutic options are currently available to treat excessive daytime sleepiness (EDS) in patients suffering from narcolepsy or obstructive sleep apnea. However, there are no comparisons between the various wake‐promoting agents i
Externí odkaz:
https://doaj.org/article/e830e577b22a4caea7b0671677b09699
Autor:
Lionel Clément, Hélène Poirier, Isabelle Niot, Virginie Bocher, Michèle Guerre-Millo, Stéphane Krief, Bart Staels, Philippe Besnard
Publikováno v:
Journal of Lipid Research, Vol 43, Iss 9, Pp 1400-1409 (2002)
Conjugated linoleic acids (CLA) are a class of positional, geometric, conjugated dienoic isomers of linoleic acid (LA). Dietary CLA supplementation results in a dramatic decrease in body fat mass in mice, but also causes considerable liver steatosis.
Externí odkaz:
https://doaj.org/article/77aafeebd9134e05bcf6ab77dd494f5b
Autor:
Martin Giret, Isabelle Nagmar, Jean-Charles Schwartz, Marilyne Uguen, Philippe Robert, Perrin David, Olivier Finance, Isabelle Berrebi-Bertrand, Stéphane Krief, Jeanne-Marie Lecomte, Simon Belliard, Xavier Ligneau
Publikováno v:
Pharmacology Research & Perspectives, Vol 9, Iss 5, Pp n/a-n/a (2021)
Pharmacology Research & Perspectives
Pharmacology Research & Perspectives
Several therapeutic options are currently available to treat excessive daytime sleepiness (EDS) in patients suffering from narcolepsy or obstructive sleep apnea. However, there are no comparisons between the various wake‐promoting agents in terms o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d9a37fbc305ba557b08a98ba979ed8a5
https://doaj.org/article/e830e577b22a4caea7b0671677b09699
https://doaj.org/article/e830e577b22a4caea7b0671677b09699
Autor:
David, Reiner, Aleksandra, Zivkovic, Olivier, Labeeuw, Stéphane, Krief, Marc, Capet, Holger, Stark
Publikováno v:
European journal of medicinal chemistry. 191
Since the discovery and early characterization of the histamine H
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::df515ce28d1f46eebb87a175fd1cfa14
https://pubmed.ncbi.nlm.nih.gov/32105981
https://pubmed.ncbi.nlm.nih.gov/32105981
Autor:
Bruno Adler, Stéphane Krief
Assez de rester bouche bée, marre d'être déstabilisé et ras le bol de penser deux heures après : « J'aurais dû dire cela »? Répondre du tac au tac est une puissante arme de séduction et de pouvoir. Le secret de ceux qui ont le sens de la re
Autor:
Thorsten Schäfer, Joachim Wegener, Sebastian Lieb, Timo Littmann, Günther Bernhardt, Miho Tanaka, Kristina Friedland, Armin Buschauer, Stéphane Krief, Sigurd Elz, Takeaki Ozawa, Nicole Plank, Johannes Felixberger
Publikováno v:
Pharmacological Research. 114:13-26
A set of histamine H1 receptor (H1R) agonists and antagonists was characterized in functional assays, using dynamic mass redistribution (DMR), electric cell-substrate impedance sensing (ECIS) and various signaling pathway specific readouts (Fura-2 an
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::f7070fd392bd258bb0676b1a86d15024
https://doi.org/10.1016/j.phrs.2016.10.010
https://doi.org/10.1016/j.phrs.2016.10.010
Autor:
Thierry Calmels, Olivier Labeeuw, Xavier Billot, Xavier Ligneau, Jeanne-Marie Lecomte, Isabelle Berrebi-Bertrand, Stéphane Krief, Denis Danvy, Nicolas Levoin, Marc Capet, Jean-Charles Schwartz, Philippe Robert
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 26:5263-5266
Synthesis and biological evaluation of a new class of histamine H4 receptor ligands, distinct from the previously reported chemotypes, are described. A virtual screening of our corporate compound collection identified a hit with an undesired dual H3R
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6a7b7ff1da6a5c21956feeeb57c288e6
https://doi.org/10.1016/j.bmcl.2016.09.049
https://doi.org/10.1016/j.bmcl.2016.09.049
Autor:
Alessandro Pini, Maria Concetta Durante, Holger Stark, Paul L. Chazot, Cecilia Lanzi, Emanuela Masini, Annemarie Schreeb, Laura Lucarini, Arianna Carolina Rosa, Stéphane Krief
Publikováno v:
Pharmacological research, 2016, Vol.111, pp.740-748 [Peer Reviewed Journal]
BASE-Bielefeld Academic Search Engine
BASE-Bielefeld Academic Search Engine
Fibrosis of lung tissue is a disease where a chronic inflammatory process determines a pathological remodelling of lung parenchyma. The animal model obtained by intra-tracheal administration of bleomycin in C57BL/6 mice is one of the most validated m
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bff43fe053a71537f292e8967754e84f
https://doi.org/10.1016/j.phrs.2016.07.037
https://doi.org/10.1016/j.phrs.2016.07.037
Publikováno v:
European Journal of Medicinal Chemistry. 191:112150
Since the discovery and early characterization of the histamine H3 receptor (H3R) in the 1980′s, predominantly imidazole-based agonists were presented to the scientific community such as Nα-methylhistamine (Nα-MeHA) or (R)-α-methylhistamine ((R)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::071c37c53e7dfa5c3776bece06f241b3
https://doi.org/10.1016/j.ejmech.2020.112150
https://doi.org/10.1016/j.ejmech.2020.112150
Autor:
Thierry Calmels, Jean-Charles Schwartz, Nicolas Levoin, Denis Danvy, Xavier Billot, Isabelle Berrebi-Bertrand, Marc Capet, Stéphane Krief, Jeanne-Marie Lecomte, Olivier Labeeuw
Publikováno v:
European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, 2017, 125, pp.565-572. ⟨10.1016/j.ejmech.2016.09.074⟩
European Journal of Medicinal Chemistry, Elsevier, 2017, 125, pp.565-572. ⟨10.1016/j.ejmech.2016.09.074⟩
European Journal of Medicinal Chemistry, 2017, 125, pp.565-572. ⟨10.1016/j.ejmech.2016.09.074⟩
European Journal of Medicinal Chemistry, Elsevier, 2017, 125, pp.565-572. ⟨10.1016/j.ejmech.2016.09.074⟩
International audience; The involvement of histamine H4 receptor (H4R) in immune cells chemotaxis and mediator release makes it an attractive target for the treatment of inflammation disorders. A decade of medicinal chemistry efforts has led to sever
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::90e8c3ee3a7850571d827909378c18b6
https://normandie-univ.hal.science/hal-02046295
https://normandie-univ.hal.science/hal-02046295