Zobrazeno 1 - 10
of 16
pro vyhledávání: '"Stanislav Huszár"'
Autor:
Nima Rezaei, Nastaran-Sadat Hosseini, Amene Saghazadeh, Abolfazl Fateh, Adriano Duse, Aijaz Ahmad, Alexander E. Braley, Alican Tahta, Alisha Kamboj, Amer Hayat Khan, Ana Cláudia Coelho, Andrea Fuso, Andrés Varón, Anete Trajman, Anil Kumar Saxena, Ankit Ganeshpurkar, Anthony M. Casapao, Anton Tkachenko, Anushka V. Devnikar, Arfa Moshiri, Arrate Muñoz-Barrutia, Arunava Dasgupta, Arvind Natarajan, Ashish Gupta, Ashlan J. Kunz Coyne, Ashly E. Jordan, Ashok Kumar, Atadzhan Ergeshov, Babak Pourakbari, Basant Joshi, Bibiana Chavarro-Portillo, Carlos Y. Soto, Carly Kanipe, Christiane Mello Schmidt, Christophe Cox, Clara Gómez-Cruz, Claudete Aparecida Araújo Cardoso, Clemax Couto Sant´Anna, Courtney Johnson, Cristhian N. Rodríguez-Silva, Cristian Rosales, Cuauhtémoc Licona-Cassani, Cynthia D. Fast, Damián Pérez-Martínez, Damiano Pizzol, David C. Perlman, Dennis Philips, Diana Viveros, Dina A. Fisher, Dmytro Butov, Eric F. Egelund, Everest de Igartua, Garima Bhatt, Georgies Mgode, Gianluca Quaglio, Giovanni Putoto, G. K. Mini, Govind Thomas-Richardson, Greg Wylie, Guilherme Felipe dos Santos Fernandes, Gustavo Bermúdez, Hélder Quintas, Himanshu Verma, Hyungjin Eoh, Ikhwanuliman Putera, Ilya Sivokozov, Isabel Pires, Jae Jin Lee, Jason E. Lombard, Jean Leandro dos Santos, Jean-Pierre Zellweger, Jenu Thomas-Richardson, Jinbert Lordson, João Lucas Prates, Jorge Cervantes, José M. Porcel, Juan José Vaquero, Justina Prada, Kamal Kamboj, Khalid F. Tabbara, Kirubel Manyazewal Mussie, Krupesh Patel, Laura Porcel, Lena Fiebig, Malu Mohan, Mange Ram Yadav, Marcela López-R, Margarida Correia-Neves, Maria da Conceição Fontes, Maria de Fátima Pombo Bazhuni Sant´Anna, Marina Cañadas-Ortega, Meenakshi Singh, Michael Lause, Milena Maya-Hoyos, Mir Davood Omrani, Mitchell V. Palmer, Mohammad Naiyaz Ahmad, Mohammed Assen Seid, Monica Chauhan, Mridula Saxena, Musa Marimani, Nanduri Srinivas, Negussie Beyene, Nelson E. Arenas, Nicole Cardoso, Olena Oliveira, Om Silakari, Osvaldo Inlamea, Özgür Tanrıverdi, Paola M. Boggiatto, Paola Santos, Paulina Mejía-Ponce, Pedro Soares, Philip Sell, Prashant R. Murumkar, Praveen Devanandan, Qi Zheng, Rachel K. Lim, Rafaela Baroni Aurílio, Rahul B. Ghuge, Rahul R. Barot, null Rahul, Ranadheer Chowdary Puvvada, Raquel Duarte, Ravi Singh, Richa Sinha, Rina La Distia Nora, Robert Burny, Roberto Zenteno-Cuevas, Sagar Mali, Samir S. Shoughy, Samira Tarashi, Sapna Mishra, Satyaveni Malasala, Setareh Mamishi, Seyed Davar Siadat, Shalki Choudhary, Shima Mahmoudi, Sidharth Chopra, Sisir Nandi, Sobia Faisal, Sonu Goel, Stanislav Huszár, Stephen K. Field, Sushil Kumar Singh, Teresa Rito, Tetiana Butova, Thomas Manning, Tjip S. van der Werf, Valeriy Myasoedov, Vanessa Vásquez, Vijey Aanandhi Muthukumar, Vinayak Singh, Walter A. Hall, Wandya Hikmahwati, Yaşar Barış Turgut, Yatri Thaker, Yoshinori Kawabata, Yvette A. de Reus
Publikováno v:
Integrated Science ISBN: 9783031159541
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7f42d8bf60e80a29de1dee0aaef53f38
https://doi.org/10.1007/978-3-031-15955-8_51
https://doi.org/10.1007/978-3-031-15955-8_51
Publikováno v:
Integrated Science ISBN: 9783031159541
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::300a589b0dc926c99609f265ae72a24f
https://doi.org/10.1007/978-3-031-15955-8_13
https://doi.org/10.1007/978-3-031-15955-8_13
Publikováno v:
Drug Discovery Today
Highlights • In 2018 1.2 million people died of tuberculosis. • The ideal drug candidate should be active against replicating and nonreplicating Mycobacterium tuberculosis. • New drug targets such as EfpA, PptT, ClpP, Pks13, DnaN and QcrB have
Structural and Activity Relationships of 6-Sulfonyl-8-Nitrobenzothiazinones as Antitubercular Agents
Autor:
Chunhua Qiao, Yu Lu, Karin Savková, Rui Shi, Quanquan Han, Giovanni Stelitano, Stanislav Huszár, Dongguang Fan, Katarína Mikušová, Laurent R. Chiarelli, Bin Wang
Publikováno v:
Journal of medicinal chemistry. 64(19)
The benzothiazinone (BTZ) scaffold compound PBTZ169 kills Mycobacterium tuberculosis by inhibiting the essential flavoenzyme DprE1, consequently blocking the synthesis of the cell wall component arabinans. While extraordinarily potent against M. tube
Autor:
Zuzana Pakanová, Karin Savková, Michal Kaliňák, Martina Tesařová, Jana Korduláková, Marie Vancová, Stanislav Kozmon, Stanislav Huszár, Jaroslav Blaško, Peter Barath, Katarína Mikušová, Vinayak Singh
Publikováno v:
Proc Natl Acad Sci U S A
Mycobacterium tuberculosis, one of the deadliest pathogens in human history, is distinguished by a unique, multilayered cell wall, which offers the bacterium a high level of protection from the attacks of the host immune system. The primary structure
Autor:
Dongguang Fan, Katarína Mikušová, Yiwen Xu, Josè Camilla Sammartino, Zhaogang Sun, Karin Savková, Laurent R. Chiarelli, Chengcheng Kong, Lingfeng Liu, Marco Fumagalli, Stanislav Huszár, Chunhua Qiao
Publikováno v:
European journal of medicinal chemistry. 208
Decaprenylphosphoryl-β-d-ribose 2'-oxidoreductase (DprE1) is a promising drug target for the development of novel anti-tubercular agents, and inhibitors of DprE1 are being investigated extensively. Among them, the 1,3-benzothiazinone compounds such
Autor:
Clara Franch, Rosangela Frita, Joel S. Freundlich, Alexandre Vandeputte, Maria Rosalia Pasca, Courtney Veilleux, Mohamad Sabbah, Rajiv Kumar Jha, Beatrice Silvia Orena, Eik Hoffmann, Katarína Mikušová, Liliana Rodrigues, Adwait Anand Godbole, Lesley A. Mitchenall, Pradeep Kumar, Valakunja Nagaraja, Nathalie Deboosere, Stanislav Huszár, Priscille Brodin, Clara Aguilar-Pérez, José A. Aínsa, Sean Ekins, Riccardo Russo, Nancy D. Connell, Anthony Maxwell, Júlia Zemanová, Martin Forbak, Thomas J. Lane, Giorgia Mori
Publikováno v:
Tuberculosis. 112:98-109
The search for compounds with biological activity for many diseases is turning increasingly to drug repurposing. In this study, we have focused on the European Union-approved antimalarial pyronaridine which was found to have in vitro activity against
Autor:
Jarmila Vinšová, František Trejtnar, Jiřina Stolaříková, Markéta Švarcová, Jana Korduláková, Katarína Mikušová, Martin Krátký, Jiří Janoušek, Jan Madacki, Stanislav Huszár, Rudolf Vosátka
Publikováno v:
European Journal of Medicinal Chemistry. 151:824-835
The development of novel drugs is essential for the treatment of tuberculosis and other mycobacterial infections in future. A series of N-alkyl-2-isonicotinoylhydrazine-1-carboxamides was synthesized from isoniazid (INH) and then cyclized to N-alkyl-
Autor:
Elena Kazakova, Olga Riabova, Júlia Zemanová, Stanislav Huszár, Arseny S. Kaprelyants, Jan S. Keruchenko, Tatyana L. Azhikina, Elena G. Salina, Vadim Makarov, Artyom Grigorov, Katarína Mikušová
Publikováno v:
Metallomics. 10:992-1002
With the emerging primary resistance of Mycobacterium tuberculosis to current drugs and wide distribution of latent tuberculosis infection, the need for new compounds with a novel mode of action is growing. Copper-mediated innate immunity and its ant
Autor:
Katarína Mikušová, Galina Karabanovich, Věra Klimešová, Alexandr Hrabálek, Karin Savková, Jan Dušek, Jaroslav Roh, Jana Korduláková, Ivona Pavkova, Oto Pavliš, Zuzana Konyariková, Tomas Kucera, Kateřina Vávrová, Jiřina Stolaříková, Jan Korábečný, Petr Pavek, Klára Konečná, Ondřej Jand’ourek, Hana Vlčková, Stanislav Huszár
Publikováno v:
Journal of medicinal chemistry. 62(17)
We report herein the discovery of 3,5-dinitrophenyl 1,2,4-triazoles with excellent and selective antimycobacterial activities against Mycobacterium tuberculosis strains, including clinically isolated multidrug-resistant strains. Thorough structure-ac