Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Song X. Huang"'
Autor:
William J. Greenlee, Tsing-Bau Chen, Kristie A. Faust, Stephen E. de Laszlo, Carol S. Quagliato, Victor J. Lotti, Raymond S.L. Chang, Song X. Huang, Eric E. Allen
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 3:1293-1298
We present the design, syntheses, and in vitro biological data of a series of substituted quinazolinone containing, AT1 selective, Angiotensin II (AII) receptor antagonists. Substituents at the 6-position of the quinazolin-4(3H)-ones 3 have pronounce
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b9fa95ce519c3e320b671e481eae2bca
https://doi.org/10.1016/s0960-894x(00)80334-0
https://doi.org/10.1016/s0960-894x(00)80334-0
Autor:
Tsuei Ju Wu, An Hua Mao, Bindhu V. Karanam, Mark T. Goulet, Xiaolan Shen, Rena Ning Ren, Kang Cheng, George R. Mount, Joel B. Yudkovitz, Jisong Cui, Thomas F. Walsh, Kathryn A. Lyons, Matthew J. Wyvratt, Jonathan R. Young, Stella H. Vincent, Josephine R. Carlin, Song X. Huang, Yi Tien Yang
Publikováno v:
Bioorganicmedicinal chemistry letters. 12(5)
A series of 2-arylindoles containing novel heteroaromatic substituents on the tryptamine tether, based on compound 1, was prepared and evaluated for their ability to act as gonadotropin releasing hormone (GnRH) antagonists. Successful modifications o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::be551d8bebe4fcd25627e7c540845563
https://pubmed.ncbi.nlm.nih.gov/11859012
https://pubmed.ncbi.nlm.nih.gov/11859012
Autor:
Roy G. Smith, Song X. Huang, Matthew J. Wyvratt, Jane Lo, Thomas F. Walsh, Yi Tien Yang, Kang Cheng, Ning Ren, Irene Chen, Mark T. Goulet, Jonathan R. Young, Joel B. Yudkovitz, Robert J. DeVita
Publikováno v:
Bioorganicmedicinal chemistry letters. 10(15)
A series of 3-arylquinolones was prepared and evaluated for their ability to act as gonadotropin releasing hormone (GnRH) antagonists. A variety of substitution patterns of the 3-aryl substituent are described. The 3,4,5-trimethylphenyl substituent (
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::273702354e5e688fb6fda23fbb065457
https://pubmed.ncbi.nlm.nih.gov/10937733
https://pubmed.ncbi.nlm.nih.gov/10937733
Potent antagonists of gonadotropin releasing hormone receptors derived from quinolone-6-carboxamides
Autor:
Joel B. Yudkovitz, Kang Cheng, Roy G. Smith, Jane-Ling Lo, Robert J. DeVita, Mark T. Goulet, Richard B. Toupence, Thomas F. Walsh, Ning Ren, Feroze Ujjainwalla, Michael H. Fisher, Matthew J. Wyvratt, Jonathan R. Young, Song X. Huang, Yi Tien Yang
Publikováno v:
Bioorganicmedicinal chemistry letters. 10(5)
SAR studies which focused upon the C-6 position of a recently described series of quinolone gonadotropin releasing hormone antagonists are reported. Synthetic access to diverse quinolone-6-carboxamides was achieved via the palladium-catalyzed amino-c
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::26b961ad3dc3f709697d007cf5ae01a6
https://pubmed.ncbi.nlm.nih.gov/10743944
https://pubmed.ncbi.nlm.nih.gov/10743944