Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Sjoerd van Schaik"'
Autor:
Axel Stoit, Sjoerd van Schaik, Josephus H. M. Lange, Annemieke Rensink, Adri van den Hoogenband, Chris G. Kruse, Hein K. A. C. Coolen, Arnold P. den Hartog
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 28:459-465
The synthesis and SAR of a novel class of spirobenzofuranpiperidinyl-derived alkanoic acids 6-34 as sphingosine S1P5 receptor agonists are described. The target compounds generally elicit high S1P5 receptor agonistic potencies and in general are sele
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::bd3ebf6ed30fa1e94992ef7801db2807
https://doi.org/10.1016/j.bmcl.2017.12.018
https://doi.org/10.1016/j.bmcl.2017.12.018
Autor:
Axel R, Stoit, Jos H M, Lange, Hein K A C, Coolen, Annemieke, Rensink, Adri, van den Hoogenband, Arnold P, den Hartog, Sjoerd, van Schaik, Chris G, Kruse
Publikováno v:
Bioorganicmedicinal chemistry letters. 28(3)
The synthesis and SAR of a novel class of spirobenzofuranpiperidinyl-derived alkanoic acids 6-34 as sphingosine S1P
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::76f53879546cda122e1a9dd857a94fb0
https://pubmed.ncbi.nlm.nih.gov/29254642
https://pubmed.ncbi.nlm.nih.gov/29254642
Autor:
Sanne Kuiper, J. Dijkink, Jan H. van Maarseveen, Henk Hiemstra, Sjoerd van Schaik, B. T. Buu Hue
Publikováno v:
European Journal of Organic Chemistry, 1, 127-137. Wiley-VCH Verlag
Studies are reported towards the synthesis of solanoeclepin A (1), the hatching agent of potato cyst nematodes. Two approaches are investigated to access the tricyclic core including the intricate bicyclo[2.1.1]hexanone moiety. The first approach is
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::55562de57649f25d4299ec6f048db4b7
https://doi.org/10.1002/ejoc.200500609
https://doi.org/10.1002/ejoc.200500609
Autor:
Arnold P. den Hartog, Tiny J.P. Adolfs, Sjoerd van Schaik, Jan H. Reinders, Hiskias G. Keizer, Nynke Barkhuijsen, Cees N. J. Stroomer, Hein K. A. C. Coolen, Chris G. Kruse, Axel Stoit, Martina A.W. van der Neut, Harry Mons
Publikováno v:
Bioorganicmedicinal chemistry letters. 18(1)
We have investigated a series of 7-azaindoles as potential partial agonists of the α4β2 nicotinic acetylcholine receptor (nAChR). Three series of 7-azaindole derivatives have been synthesized and evaluated for rat brain neuronal nicotinic receptor
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::91661210ad122c794780ca9e60253d69
https://pubmed.ncbi.nlm.nih.gov/18006307
https://pubmed.ncbi.nlm.nih.gov/18006307
Autor:
B. T. Buu Hue, Jan Dijkink, Sanne Kuiper, Sjoerd van Schaik, Jan H. van Maarseveen, Henk Hiemstra
Publikováno v:
European Journal of Organic Chemistry; Jan2006, Vol. 2006 Issue 1, p127-137, 0p