Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Simone, Gastaldi"'
Autor:
Elisabetta Marini, Marco Marino, Giulia Gionfriddo, Federica Maione, Marta Pandini, Daniele Oddo, Marta Giorgis, Barbara Rolando, Federica Blua, Simone Gastaldi, Serena Marchiò, Sandra Kovachka, Francesca Spyrakis, Eleonora Gianquinto, Federica Di Nicolantonio, Massimo Bertinaria
Publikováno v:
Molecules, Vol 27, Iss 23, p 8513 (2022)
BRAF is a serine/threonine kinase frequently mutated in human cancers. BRAFV600E mutated protein is targeted through the use of kinase inhibitors which are approved for the treatment of melanoma; however, their long-term efficacy is hampered by resis
Externí odkaz:
https://doaj.org/article/321ff11884e9491784732a391526bf64
Autor:
Simone Gastaldi, Valentina Boscaro, Eleonora Gianquinto, Christina F. Sandall, Marta Giorgis, Elisabetta Marini, Federica Blua, Margherita Gallicchio, Francesca Spyrakis, Justin A. MacDonald, Massimo Bertinaria
Publikováno v:
Molecules, Vol 26, Iss 13, p 3975 (2021)
In the search for new chemical scaffolds able to afford NLRP3 inflammasome inhibitors, we used a pharmacophore-hybridization strategy by combining the structure of the acrylic acid derivative INF39 with the 1-(piperidin-4-yl)1,3-dihydro-2H-benzo[d]im
Externí odkaz:
https://doaj.org/article/3c3494cec8624421abf07d12c3ebe214
Autor:
Carolina Pellegrini, Matteo Fornai, Rocchina Colucci, Laura Benvenuti, Vanessa D’Antongiovanni, Gianfranco Natale, Federica Fulceri, Marta Giorgis, Elisabetta Marini, Simone Gastaldi, Massimo Bertinaria, Corrado Blandizzi, Luca Antonioli
Publikováno v:
Frontiers in Pharmacology, Vol 9 (2018)
Nucleotide-binding oligomerization domain leucine rich repeat and pyrin domain-containing protein 3 (NLRP3) inflammasome is pivotal in maintaining intestinal homeostasis and sustaining enteric immune responses in the setting of inflammatory bowel dis
Externí odkaz:
https://doaj.org/article/87239b7fac1d4ddc9c7d0f80aba67650
Publikováno v:
Inflammasome Biology ISBN: 9780323918022
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ea6c603e20a6fa89d9f72499b48e64ed
https://doi.org/10.1016/b978-0-323-91802-2.00037-2
https://doi.org/10.1016/b978-0-323-91802-2.00037-2
Autor:
Antonio Abbate, Ivona Aksentijevich, Marcelo Pires Amaral, Magaiver Andrade-Silva, Diego Angosto-Bazarra, Luca Antonioli, Kübra Aral, Juan I. Aróstegui, Jillian Barlow, Laura Benvenuti, Nunzia Bernardini, Massimo Bertinaria, Monika Biasizzo, Karina Ramalho Bortoluci, Dave Boucher, Laura Migliari Branco, David Brough, Petr Broz, Clare E. Bryant, Mark Cahill, Matthew Campbell, Soo Jung Cho, Shelbi Christgen, Rebecca C. Coll, Isabelle Couillin, Brianna Cyr, Sarah Dalmon, Juan Pablo de Rivero Vaccari, Francesco Di Virgilio, Andrea Dorfleutner, Sarah L. Doyle, Vanessa D'Antongiovanni, Ariel E. Feldstein, Matteo Fornai, Carlos García-Palenciano, Simone Gastaldi, Matthias Geyer, François Ghiringhelli, Anna Lisa Giuliani, José Manuel González-Navajas, Iva Hafner-Bratkovič, Shaima'a Hamarsheh, Michael T. Heneka, Thomas Henry, Jun-ichi Hikima, Inga V. Hochheiser, Alexander Hogg, Alexander Hooftman, Christopher Hoyle, Yin Huang, Sarah Huot-Marchand, Laura Hurtado-Navarro, Sushmita Jha, Thirumala-Devi Kanneganti, Benedikt Kaufmann, Andrea D. Kim, Nataša Kopitar-Jerala, Jordana Kron, Silvia Lucena Lage, Beatriz Lozano-Ruiz, Elisabetta Marini, Billie Matchett, Adolfo G. Mauro, Eleonora Mezzaroma, Michael R. Milward, Ingrid Kazue Mizuno Watanabe, Natsuki Morimoto, Sandip Mukherjee, Mar Orzáez, Luke A.J. O'Neill, Pablo Pelegrín, Carolina Pellegrini, Anaïs Perrichet, Joanna Picó, Nicola Potere, Alexander Pronko, Kishore Aravind Ravichandran, Nicolas Riteau, Kim S. Robinson, Cédric Rébé, Fadi N. Salloum, Mónica Sancho, Andrew Sandstrom, Niels Olsen Saraiva Câmara, Florian I. Schmidt, Liang Shan, Eoin Silke, Paula M. Soriano-Teruel, Christian Stehlik, Heather Stout-Delgado, Arianne L. Theiss, Jenny P.-Y. Ting, Stefano Toldo, Elviche L. Tsakem, Rebecca E. Tweedell, Amalia Tzoumpa, K. Venuprasad, Rose Wellens, Robert Zeiser, Franklin L. Zhong, Alessia Zotta
Publikováno v:
Inflammasome Biology ISBN: 9780323918022
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1df40277879d3530be000cf63f0ec15f
https://doi.org/10.1016/b978-0-323-91802-2.01002-1
https://doi.org/10.1016/b978-0-323-91802-2.01002-1
Autor:
Stefano Comità, Pasquale Pagliaro, Claudia Penna, Massimo Bertinaria, Francesca Spyrakis, Simone Gastaldi, Valentina Boscaro, Eleonora Gianquinto
Publikováno v:
Journal of Molecular and Cellular Cardiology. 173:123-124
Autor:
Carolina, Pellegrini, Colucci, ROCCHINA LUCIA, Laura, Benvenuti, Vanessa, D'Antongiovanni, Clelia Di Salvo, Simone, Gastaldi, Federica, Blua, Elisabetta, Marini, Barbara, Rolando, Lorettalazzarato, Nunzia, Bernardini, Luca, Antonioli, Massimo, Bertinaria, Matteo, Fornai
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=od______3657::edb05b87c19cf784f8f4dac6317b5e91
http://hdl.handle.net/11577/3456808
http://hdl.handle.net/11577/3456808
Autor:
Justin A. MacDonald, Eleonora Gianquinto, Marta Giorgis, Valentina Boscaro, Francesca Spyrakis, Federica Blua, Christina F. Sandall, Margherita Gallicchio, Elisabetta Marini, Massimo Bertinaria, Simone Gastaldi
Publikováno v:
Molecules
Volume 26
Issue 13
Molecules, Vol 26, Iss 3975, p 3975 (2021)
Volume 26
Issue 13
Molecules, Vol 26, Iss 3975, p 3975 (2021)
In the search for new chemical scaffolds able to afford NLRP3 inflammasome inhibitors, we used a pharmacophore-hybridization strategy by combining the structure of the acrylic acid derivative INF39 with the 1-(piperidin-4-yl)1,3-dihydro-2H-benzo[d]im
Autor:
Carolina Pellegrini, Rocchina Colucci, Laura Benvenuti, Vanessa D'Antongiovanni, Clelia Di Salvo, Simone Gastaldi, Federica Blua, Elisabetta Marini, Barbara Rolando, Loretta Lazzarato, Nunzia Bernardini, Luca Antonioli, Massimo Bertinaria, Matteo Fornai
Publikováno v:
Gastroenterology. 162:S-163
The NOD-like receptor family, pyrin domain-containing 3 (NLRP3) inflammasome is the best recognized and most widely implicated regulator of caspase-1 activation. It is a key regulator of innate immune response and is involved in many pathophysiologic
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c1b3d803df885121213baa22c23999f8
http://hdl.handle.net/2318/1720025
http://hdl.handle.net/2318/1720025