Výsledky vyhledávání - "Siddharth Phalle"

Optimization of Thiazolidone Scaffolds Using Pocket Modeling for Development of Potential Secretory System Inhibitors of Mycobacterium tuberculosis

Autor: Rakesh P. Dhavale, Prafulla B. Choudhari, Durgacharan A. Bhagwat, Sambhaji R. Masal, Santosh S. Kumbhar, Shivratna V. Khare, Aakash K. Patil, Sujata Choudhari, Atul M. Kadam, Siddharth Phalle

Publikováno v: Turkish Journal of Pharmaceutical Sciences, Vol 16, Iss 2, Pp 196-205 (2019)
Turkish Journal of Pharmaceutical Sciences

Objectives Mycobacterium tuberculosis is the causative organism of tuberculosis, which is the most lethal disease after cancer in the current decade. The development of multidrug and broadly drug-resistant strains is making the problem of tuberculosi

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f92bde8a6aa6c58753f6536732137968
https://doi.org/10.4274/tjps.galenos.2018.12599

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Synthesis and antimycobacterial evaluation of new 5-(1-benzyl-1H-1,2,3-triazol-4-yl)-4-methyl-2-arylthiazole derivatives

Autor: Amit S. Choudhari, Prafulla B. Choudhari, Dhiman Sarkar, Vikas Shinde, Siddharth Phalle, Shakti Chakraborty, Pramod P. Mahulikar, Pravin C. Mhaske

Publikováno v: Medicinal Chemistry Research. 28:805-819

A new series of 5-(1-benzyl-1H-1,2,3-triazol-4-yl)-4-methyl-2-arylthiazole derivatives, 6a−w have been synthesized by click reaction of substituted benzylazide, 5a−d with 5-ethynyl-4-methyl-2-substituted phenylthiazole, 4a−f. The starting compo

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::d6b608413b3d2c34f61464ed9b3cc16c
https://doi.org/10.1007/s00044-019-02310-y

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K Nearest Neighbor and 3D QSAR Analysis of Thiazolidinone Derivatives as Antitubercular Agents

Autor: Siddharth Phalle, Shivaratna Khare, Sujata Choudhari, Santosh S. Kumbhar, Prafulla B. Choudhari, Atul Kadam, Prajakta Subramani

Publikováno v: Journal of Pharmaceutical Research. 15:67

Purpose : The present research communication describes development of kNN and 3D QSAR models for identification of structural features which are responsible for antimycobacterial activity of Thiazolidinone. Methodology/Approach : In the present work,

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::cebe3adf840879525ac73b04745da5a9
https://doi.org/10.18579/jpcrkc/2016/15/3/103037

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