Zobrazeno 1 - 10 of 236 pro vyhledávání: '"Shrinivas D. Joshi"'
1
Akademický článek
Ionic liquid Mediated Pd-catalyzed sonochemistry for facile synthesis of carbazoles: Molecular Modelling and antimicrobial studies
Autor: Imamhusen Jamadar, Athmanand Anchi, Shruti S. Malunavar, Rajesh G. Kalkhambkar, Suraj M. Sutar, Shrinivas D. Joshi
Publikováno v: Tetrahedron Green Chem, Vol 3, Iss , Pp 100038- (2024)
Herein we have described the Pd-catalyzed sonochemistry driven by [BMIM]-IL as re-useable solvent to synthesize various carbazole scaffolds from 2,2′-dibromodiphenyl. Diverse primary amines were utilised as coupling partners in the presence of [PAI
Externí odkaz: https://doaj.org/article/bd73e6a25bc34fd4990f9204a383acc6
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2
Akademický článek
Synthesis, molecular docking study and biological evaluation of new pyrrole scaffolds as potential antitubercular agents for dual targeting of enoyl ACP reductase and dihydrofolate reductase.
Autor: Mater H Mahnashi, Sravanthi Avunoori, Sanjay Gopi, Ibrahim Ahmed Shaikh, Ahmed Saif, Farkad Bantun, Hani Saleh Faidah, Abdulrahman Ali Alhadi, Jaber Hassan Alshehri, Abdullah Ali Alharbi, Prem Kumar S R, Shrinivas D Joshi
Publikováno v: PLoS ONE, Vol 19, Iss 5, p e0303173 (2024)
In this study, new series of N'-(2-(substitutedphenoxy)acetyl)-4-(1H-pyrrol-1-yl)benzohydrazides (3a-j) 4-(2,5-dimethyl-1H-pyrrol-1-yl)-N'-(2-(substitutedphenoxy)acetyl)benzohydrazides (5a-j) were synthesized, characterized and assessed as inhibitors
Externí odkaz: https://doaj.org/article/47dfe48cb4e74c7396f27ecdff2dae44
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3
Akademický článek
In vitro antimicrobial combat, molecular modelling and structure activity relationship studies of novel class of aryl-ethyne tethered coumarin analogues and some 3-aryl coumarin derivatives
Autor: Pavankumar Prabhala, Suraj M. Sutar, Hemantkumar M. Savanur, Shrinivas D. Joshi, Rajesh G. Kalkhambkar
Publikováno v: European Journal of Medicinal Chemistry Reports, Vol 5, Iss , Pp 100048- (2022)
A series of novel class of aryl ethyne-tethered coumarin analogues (series 1) and some 3-aryl coumarin cognates (series 2) were synthesized, and their in vitro antimicrobial activities aided by molecular modelling and the structure activity relations
Externí odkaz: https://doaj.org/article/c6412ae62302463394ecebd8f7208748
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4
Akademický článek
Synthesis, Molecular Docking Study, and Biological Evaluation of New 4-(2,5-Dimethyl-1H-pyrrol-1-yl)-N’-(2-(substituted)acetyl)benzohydrazides as Dual Enoyl ACP Reductase and DHFR Enzyme Inhibitors
Autor: Mater H. Mahnashi, Pooja Koganole, Prem Kumar S. R., Sami S. Ashgar, Ibrahim Ahmed Shaikh, Shrinivas D. Joshi, Ali S. Alqahtani
Publikováno v: Antibiotics, Vol 12, Iss 4, p 763 (2023)
In this study, a new series of 4-(2,5-dimethyl-1H-pyrrol-1-yl)-N’-(2-(substituted)acetyl) benzohydrazides (5a–n) were prepared and new heterocycles underwent thorough characterization and evaluation for antibacterial activity; some of them underw
Externí odkaz: https://doaj.org/article/74418f7c57cb43bd80ab163b1730443c
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5
Akademický článek
Synthesis of novel indole, 1,2,4-triazole derivatives as potential glucosidase inhibitors
Autor: Ramesh S Gani, Karabasanagouda Timanagouda, S. Madhushree, Shrinivas D Joshi, Murigendra B. Hiremath, Salma Begum Hussain Mujawar, Avinash Kundadka Kudva
Publikováno v: Journal of King Saud University: Science, Vol 32, Iss 8, Pp 3388-3399 (2020)
Objective: In the present study a series of eleven bis-heterocyclic compounds with indole derivative carrying 1,2,4-triazole moiety were synthesized and assessed for their in vitro α-amylase and α-glucosidase inhibition activity. Method: The synthe
Externí odkaz: https://doaj.org/article/d15d00bee57248bc97908211872c79e9
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6
Microwave-assisted copper(i) catalyzed A3 cascade coupling of imidazo[1,2-a]pyridines via C–H bond functionalization as selective COX-2 inhibitors and antioxidants, and in silico studies
Autor: Aravind R. Nesaragi, Ravindra R. Kamble, Swati R. Hoolageri, Shruti Dixit, Shrinivas D. Joshi, Shyamkumar Vootla, Vijay M. Kumbar
Publikováno v: New Journal of Chemistry. 47:9401-9413
A proficient copper(i) catalyzed one pot synthetic protocol has been established to synthesize medicinally essential substituted imidazo[1,2-a]pyridines via C–H bond amination followed by acetylene incorporation under microwave irradiation.
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::06d33e630ee76ffafc0c2cd0317ece1a
https://doi.org/10.1039/d3nj00524k
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8
Akademický článek
Synthesis and in vitro anticancer activity of 6-chloro-7-methyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one derivatives: molecular docking and interaction with bovine serum albumin
Autor: Supreet Gaonkar, Manjunath G. Sunagar, Narahari Deshapande, Ningaraddi S. Belavagi, Shrinivas D Joshi, Sheshagiri R Dixit, Imtiyaz Ahmed M. Khazi
Publikováno v: Journal of Taibah University for Science, Vol 12, Iss 4, Pp 382-392 (2018)
A novel series of 6-chloro-7-methyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one derivatives were synthesized. Structure of the newly synthesized compounds was established by their analytical and spectroscopic data. The title compounds were evaluated
Externí odkaz: https://doaj.org/article/bd03bd99d00e4e59b653c8e46abaf65a
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9
Akademický článek
In silico binding affinity studies of N-9 substituted 6-(4-(4-propoxyphenyl)piperazin-1-yl)-9H-purine derivatives-Target for P70-S6K1 & PI3K-δ kinases
Autor: Manjunath G. Sunagar, P. Aravind, Supreet Gaonkar, K.S. Devaraju, Shrinivas D. Joshi, Sheshagiri R. Dixit, B.M. Harish, Imtiyaz Ahmed M. Khazi
Publikováno v: Beni-Suef University Journal of Basic and Applied Sciences, Vol 7, Iss 1, Pp 84-91 (2018)
P70-S6K1 & PI3K-δ kinases are identified to be involved in many physiological processes associated with cancer, therefore many of the inhibitors being designed to target these kinases are in clinical trials. In the current study we have exploited th
Externí odkaz: https://doaj.org/article/007ebcee080b42878ea1f26b09aa4902
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