Zobrazeno 1 - 10 of 146 pro vyhledávání: '"Shrinivas D Joshi"'
1
Akademický článek
Synthesis, molecular docking study and biological evaluation of new pyrrole scaffolds as potential antitubercular agents for dual targeting of enoyl ACP reductase and dihydrofolate reductase.
Autor: Mater H Mahnashi, Sravanthi Avunoori, Sanjay Gopi, Ibrahim Ahmed Shaikh, Ahmed Saif, Farkad Bantun, Hani Saleh Faidah, Abdulrahman Ali Alhadi, Jaber Hassan Alshehri, Abdullah Ali Alharbi, Prem Kumar S R, Shrinivas D Joshi
Publikováno v: PLoS ONE, Vol 19, Iss 5, p e0303173 (2024)
In this study, new series of N'-(2-(substitutedphenoxy)acetyl)-4-(1H-pyrrol-1-yl)benzohydrazides (3a-j) 4-(2,5-dimethyl-1H-pyrrol-1-yl)-N'-(2-(substitutedphenoxy)acetyl)benzohydrazides (5a-j) were synthesized, characterized and assessed as inhibitors
Externí odkaz: https://doaj.org/article/47dfe48cb4e74c7396f27ecdff2dae44
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2
Akademický článek
Synthesis of novel indole, 1,2,4-triazole derivatives as potential glucosidase inhibitors
Autor: Ramesh S Gani, Karabasanagouda Timanagouda, S. Madhushree, Shrinivas D Joshi, Murigendra B. Hiremath, Salma Begum Hussain Mujawar, Avinash Kundadka Kudva
Publikováno v: Journal of King Saud University: Science, Vol 32, Iss 8, Pp 3388-3399 (2020)
Objective: In the present study a series of eleven bis-heterocyclic compounds with indole derivative carrying 1,2,4-triazole moiety were synthesized and assessed for their in vitro α-amylase and α-glucosidase inhibition activity. Method: The synthe
Externí odkaz: https://doaj.org/article/d15d00bee57248bc97908211872c79e9
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3
Akademický článek
Synthesis and in vitro anticancer activity of 6-chloro-7-methyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one derivatives: molecular docking and interaction with bovine serum albumin
Autor: Supreet Gaonkar, Manjunath G. Sunagar, Narahari Deshapande, Ningaraddi S. Belavagi, Shrinivas D Joshi, Sheshagiri R Dixit, Imtiyaz Ahmed M. Khazi
Publikováno v: Journal of Taibah University for Science, Vol 12, Iss 4, Pp 382-392 (2018)
A novel series of 6-chloro-7-methyl-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one derivatives were synthesized. Structure of the newly synthesized compounds was established by their analytical and spectroscopic data. The title compounds were evaluated
Externí odkaz: https://doaj.org/article/bd03bd99d00e4e59b653c8e46abaf65a
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4
Akademický článek
In vitro antimicrobial combat, molecular modelling and structure activity relationship studies of novel class of aryl-ethyne tethered coumarin analogues and some 3-aryl coumarin derivatives
Autor: Pavankumar Prabhala, Suraj M. Sutar, Hemantkumar M. Savanur, Shrinivas D. Joshi, Rajesh G. Kalkhambkar
Publikováno v: European Journal of Medicinal Chemistry Reports, Vol 5, Iss , Pp 100048- (2022)
A series of novel class of aryl ethyne-tethered coumarin analogues (series 1) and some 3-aryl coumarin cognates (series 2) were synthesized, and their in vitro antimicrobial activities aided by molecular modelling and the structure activity relations
Externí odkaz: https://doaj.org/article/c6412ae62302463394ecebd8f7208748
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5
Akademický článek
Synthesis, Molecular Docking Study, and Biological Evaluation of New 4-(2,5-Dimethyl-1H-pyrrol-1-yl)-N’-(2-(substituted)acetyl)benzohydrazides as Dual Enoyl ACP Reductase and DHFR Enzyme Inhibitors
Autor: Mater H. Mahnashi, Pooja Koganole, Prem Kumar S. R., Sami S. Ashgar, Ibrahim Ahmed Shaikh, Shrinivas D. Joshi, Ali S. Alqahtani
Publikováno v: Antibiotics, Vol 12, Iss 4, p 763 (2023)
In this study, a new series of 4-(2,5-dimethyl-1H-pyrrol-1-yl)-N’-(2-(substituted)acetyl) benzohydrazides (5a–n) were prepared and new heterocycles underwent thorough characterization and evaluation for antibacterial activity; some of them underw
Externí odkaz: https://doaj.org/article/74418f7c57cb43bd80ab163b1730443c
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6
Microwave-assisted copper(i) catalyzed A3 cascade coupling of imidazo[1,2-a]pyridines via C–H bond functionalization as selective COX-2 inhibitors and antioxidants, and in silico studies
Autor: Aravind R. Nesaragi, Ravindra R. Kamble, Swati R. Hoolageri, Shruti Dixit, Shrinivas D. Joshi, Shyamkumar Vootla, Vijay M. Kumbar
Publikováno v: New Journal of Chemistry. 47:9401-9413
A proficient copper(i) catalyzed one pot synthetic protocol has been established to synthesize medicinally essential substituted imidazo[1,2-a]pyridines via C–H bond amination followed by acetylene incorporation under microwave irradiation.
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::06d33e630ee76ffafc0c2cd0317ece1a
https://doi.org/10.1039/d3nj00524k
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10
SYNTHESIS AND ANTITUBERCULAR EVALUATION OF CERTAIN PYRROLE DERIVATIVES
Autor: Sandhya Chinnamulagund, Ashwini S. Joshi, Chetana, Sravanthi Avunoori, V. H. Kulkarni, Shrinivas D. Joshi
A series of 2-aryl-5-[4-(1H-pyrrol-1-yl)phenyl]-1,3,4-oxadiazole derivatives (VIa-g) have been synthesized in good yields. These compounds were synthesized with an approach to reduce the growing anti-tubercular resistance and to develop more potent a
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::302a29d51620edac2012887938147f07
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