Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Sharad H. Bhosale"'
Autor:
Kakasaheb R. Mahadik, Radha Charan Dash, Mugdha R. Suryawanshi, Sharad H. Bhosale, Suhas M. Shelke
Publikováno v:
Medicinal Chemistry. 8:1069-1075
A series of novel N,N-diphenyl-2-[4-(substituted phenyl)piperazin-1-yl]acetamides was designed, synthesized and evaluated for anti-dopaminergic activity, anti-serotonergic activity and catalepsy induction studies in mice as an approach to novel poten
Autor:
Suhas M. Shelke, Mugdha R. Suryawanshi, Ashish M. Kanhed, Kakasaheb R. Mahadik, Radha Charan Dash, Sharad H. Bhosale
Publikováno v:
Molecular Diversity. 16:367-375
The dopamine D(2) receptor is involved in the etiology of a number of disorders, such as Parkinson's disease, Huntington's Chorea, tardive dyskinesia and schizophrenia. Antagonism of D(2) receptors is implicated in the treatment of various psychiatri
Autor:
Suhas M. Shelke, Mugdha R. Suryawanshi, Kakasaheb R. Mahadik, Radha Charan Dash, Sharad H. Bhosale
Publikováno v:
Medicinal Chemistry Research. 20:29-35
The present research paper reports the synthesis and biological evaluation of 6-(3-substitutedpropoxyl)benzo[d][1,3]oxathiol-2-ones as potential atypical antipsychotic agents. Accordingly, 10 derivatives with either amino or aryloxy substituents were
Publikováno v:
European journal of medicinal chemistry. 74
This article describes the design of biphenyl moiety linked with aryl piperazine and syntheses of fourteen 1-(biphenyl-4-yl)-2-[4-(substituted phenyl)-piperazin-1-yl]ethanone derivatives along with their pharmacological evaluation for antipsychotic a
To study the derivatives of 1,2,4-triazino[5,6-b]indole-3-thione for antidepressant activity in olfactory bulbectomized (OBX) rats. Out of various derivatives tested for acute tail suspension test, the two derivatives showing prominent action were se
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::368f67dd8a01f907112d9ed4c96d79fb
https://europepmc.org/articles/PMC3621477/
https://europepmc.org/articles/PMC3621477/
Autor:
Mugdha R. Suryawanshi, Kakasaheb R. Mahadik, Radha Charan Dash, Sharad H. Bhosale, Suhas M. Shelke
Publikováno v:
Bioorganicmedicinal chemistry letters. 21(8)
Monoamine oxidase-A (MAO-A) inhibitors are of particular importance in the treatment of depressive disorders. Herein described is pharmacophore generation and atom-based 3D-QSAR analysis of previously reported pyrrole based MAO-A inhibitors in order
Autor:
Sushilkumar Sushilkumar, K. R. Mahadik, Suhas M. Shelke, V. S. Veer, Sharad H. Bhosale, Shivajirao S. Kadam, Nitin Sati, Subhash L. Bodhankar
Publikováno v:
ChemInform. 37