Výsledky vyhledávání - "Shailee V. Tiwari"

Akademický článek

Appraisal and synthesis of novel indole-thiazole derivatives as epidermal growth factor receptor tyrosine kinase (EGFR-TK) inhibitors against resistance mutation for lung cancer treatment

Autor: Shailee V. Tiwari, Dattatraya N. Pansare, Deepak K. Lokwani, Shashikant V. Bhandari, Vijay V. Kanode, Omkar V. Tandale, Akshay R. Kadam

Publikováno v: Results in Chemistry, Vol 11, Iss , Pp 101760- (2024)

For the treatment of NSCLC one of the promising strategies is targeted inhibition of EGFR and its mutants. In this research work, we tend to epitomize design, synthesis, in-vitro anticancer evaluation of novel indole-thiazole derivatives as novel rev

Externí odkaz: https://doaj.org/article/39474eb0cf224a37bc25e6fe10c53228

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Akademický článek

A facile synthesis and characterization of some novel benzimidazole derivatives

Autor: Rahul B. Shinde, Dattatraya N. Pansare, Rohini N. Shelke, Aniket P. Sarkate, Shailee V. Tiwari, Mukund N. Bangal, Devidas S. Bhagat, Ashok M. Zine

Publikováno v: Results in Chemistry, Vol 6, Iss , Pp 101134- (2023)

We successfully synthesized a series of novel benzimidazole derivatives with high yields in our current research study. The synthesis procedure involved condensing Ethyl 3-[[3-amino-4-(treiethylamino) benzoyl] (pyridine-5-yl) amino]-propanoate with v

Externí odkaz: https://doaj.org/article/dccc19cabab74209a6305c34fd97572b

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Akademický článek

New 2-Oxoindolin Phosphonates as Novel Agents to Treat Cancer: A Green Synthesis and Molecular Modeling

Autor: Shailee V. Tiwari, Nawaz S. Sharif, Rekha I. Gajare, Julio A. Seijas Vazquez, Jaiprakash N. Sangshetti, Manoj D. Damale, Anna Pratima G. Nikalje

Publikováno v: Molecules, Vol 23, Iss 8, p 1981 (2018)

The work reports the facile synthesis of novel α-aminophosphonate derivatives coupled with indole-2,3-dione moieties, namely the diethyl(substituted phenyl/heteroaryl)(2-(2-oxoindolin-3-ylidene)hydrazinyl)methylphosphonates derivatives 4(a–n). One

Externí odkaz: https://doaj.org/article/af4e8a2e4ab64588a7235dc391d1f86e

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Akademický článek

Ionic Liquid-Promoted Synthesis of Novel Chromone-Pyrimidine Coupled Derivatives, Antimicrobial Analysis, Enzyme Assay, Docking Study and Toxicity Study

Autor: Shailee V. Tiwari, Julio A. Seijas, Maria Pilar Vazquez-Tato, Aniket P. Sarkate, Kshipra S. Karnik, Anna Pratima G. Nikalje

Publikováno v: Molecules, Vol 23, Iss 2, p 440 (2018)

Herein, we report an environmentally friendly, rapid, and convenient ionic liquid ([Et3NH][HSO4])-promoted facile synthesis of ethyl 4-(6-substituted-4-oxo-4H-chromen-3-yl)-6-methyl-2-thioxo/oxo-1,2,3,4-tetrahydropyrimidine-5-carboxylate derivatives

Externí odkaz: https://doaj.org/article/69cbc475ae444a56a471a6ccebf06ca1

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Akademický článek

Facile Synthesis of Novel Coumarin Derivatives, Antimicrobial Analysis, Enzyme Assay, Docking Study, ADMET Prediction and Toxicity Study

Autor: Shailee V. Tiwari, Julio A. Seijas, Maria Pilar Vazquez-Tato, Aniket P. Sarkate, Kshipra S. Karnik, Anna Pratima G. Nikalje

Publikováno v: Molecules, Vol 22, Iss 7, p 1172 (2017)

The work reports the synthesis under solvent-free condition using the ionic liquid [Et3NH][HSO4] as a catalyst of fifteen novel 3-((dicyclohexylamino)(substituted phenyl/heteryl)-methyl)-4-hydroxy-2H-chromen-2-onederivatives 4a–o as potential antim

Externí odkaz: https://doaj.org/article/cb2d96bef405491a865871b2fb926e32

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Akademický článek

Microwave-Assisted Facile Synthesis, Anticancer Evaluation and Docking Study of N-((5-(Substituted methylene amino)-1,3,4-thiadiazol-2-yl)methyl) Benzamide Derivatives

Autor: Shailee V. Tiwari, Sumaiya Siddiqui, Julio A. Seijas, M. Pilar Vazquez-Tato, Aniket P. Sarkate, Deepak K. Lokwani, Anna Pratima G. Nikalje

Publikováno v: Molecules, Vol 22, Iss 6, p 995 (2017)

In the present work, 12 novel Schiff’s bases containing a thiadiazole scaffold and benzamide groups coupled through appropriate pharmacophore were synthesized. These moieties are associated with important biological properties. A facile, solvent-fr

Externí odkaz: https://doaj.org/article/2d4c82c99a5441a3af01c8dd473669e0

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