Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Shafiya Yaseen"'
Autor:
Syed Ovais, Kalim Javed, H. Pushpalatha, Mymoona Akthar, Rafia Bashir, Pooja Rathore, Omprakash Tanwar, G. Bhanuprakash Reddy, Alhamza Dheyaa, Shafiya Yaseen, Mohammed Samim, Raed Yaseen
Publikováno v:
European Journal of Medicinal Chemistry. 80:209-217
Seventeen new pyrazoline substituted benzenesulfonylurea/thiourea derivatives (2a–q) were synthesized and characterized by elemental analysis and various spectroscopic techniques viz; IR, 1H NMR, 13C NMR, and MS data. Thirteen compounds showed mode
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry. 29:362-366
Some new benzenesulfonylthiourea derivatives substituted with phthalazones (2a–q) were synthesized by refluxing the appropriate 4-aryl-1-oxophthalazin-2(1H)yl benzenesulfonamides with isothiocyanate in dry acetone over anhydrous K2CO3. All the synt
Autor:
Syed Ovais, Vinod Nair, Rafia Bashir, Mohammed Samim, Surender Singh, Kalim Javed, Pooja Rathore, Shafiya Yaseen
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry. 28:1105-1112
Nine novel 4-[3-(4-Dimethylamino-phenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]-benzenesulfonamides (2a-i) were synthesized and evaluated for their anti-inflammatory and antiproliferative activities. These compounds (2a-i) showed moderate to strong anti-in
Publikováno v:
Medicinal Chemistry Research. 22:1378-1385
A series of novel pyrazolines (2a–l) bearing benzenesulfonamide moiety were synthesized by condensing appropriate chalcone (1a–l) with 4-hydrazinobenzenesulfonamide hydrochloride. Structure of all novel synthesized compounds was characterized on
Autor:
Syed Ovais, Hinna Hamid, Kalim Javed, Mohammad Sarwar Alam, Rafia Bashir, Shafiya Yaseen, Mohammed Samim
Publikováno v:
Medicinal Chemistry Research. 21:4352-4356
Five (2a–e) benzenesulfonylurea derivatives bearing pyridazinone were synthesized by refluxing the appropriate 6-aryl-2-(p-sulfamylphenyl)-4,5-dihydropyridazine-3(2H)-one with benzylisocyanate in dry acetone over anhydrous K2CO3. These compounds we
Autor:
Hinna Hamid, Rafia Bashir, Shafiya Yaseen, Mohammad Sarwar Alam, Syed Ovais, Kalim Javed, Mohammad Samim
Publikováno v:
Medicinal Chemistry Research. 21:428-436
Some new benzenesulfonylthiourea derivatives substituted with pyridazinone (2a–o) were synthesized by refluxing the appropriate 6-aryl-2-(p-sulfamylphenyl)-4,5-dihydropyridazine-3(2H)-ones with isothiocyanate in dry acetone over anhydrous K2CO3. Al
Autor:
Kalim Javed, Alhamzah Dh. Hameed, Mohammed Samim, Pooja Rathore, Rakesh Gupta, Shafiya Yaseen, Syed Ovais, Rafia Bashir, Raed Yaseen, Firasat Hussain
Publikováno v:
Bioorganicmedicinal chemistry letters. 24(7)
Twenty six new pyrazoline substituted benzenesulfonylureas (2a–z) were synthesized and tested for in vitro anticancer activity. Fourteen derivatives (2i, 2k–2p, 2r, 2s–2x) were screened for their antiproliferative activity towards 60 human canc
Autor:
Surender Singh, Syed Ovais, Vinod Nair, Shafiya Yaseen, Pooja Rathore, Mohammed Samim, Kalim Javed, Rafia Bashir
Publikováno v:
ChemInform. 44
The synthesized compounds are tested for their anti-inflammatory and anticancer activities.
Autor:
Mohammed Samim, Surender Singh, Rafia Bashir, Pooja Rathore, Syed Ovais, Shafiya Yaseen, Vinod Nair, Kalim Javed
Publikováno v:
Archiv der Pharmazie. 346(6)
Nine 4-arylphthalazones bearing benzenesulfonamide (2a–i) were synthesized by the condensation of the appropriate 2-aroylbenzoic acid (1a–i) and 4-hydrazinobenzenesulfonamide in ethanol. The structures of these compounds were elucidated by elemen
Autor:
Rafia Bashir, Raed Yaseen, Alhamzah Dh. Hameed, Kalim Javed, Syed Ovais, Pooja Rathore, Shafiya Yaseen, Mohammad Samim
Publikováno v:
European journal of medicinal chemistry. 67
Sixteen new 6-aryl-2-( p -(methanesulfonyl)phenyl)-4,5-dihydropyridazi-3(2 H )-ones ( 2a – p ) were synthesized and tested for in vitro anticancer and in vivo anti-inflammatory activities. Eleven ( 2b , 2d , 2e – j and 2m – p ) of the obtained