Zobrazeno 1 - 10
of 34
pro vyhledávání: '"Setsuo Funasaka"'
Autor:
Akihiko Tsuruoka, Toshimitsu Uenaka, Masao Iwata, Junji Matsui, Tomohiro Matsushima, Toshimi Okada, Yoshinobu Yamane, Isao Ohashi, Yuki Karoji, Yusuke Nakatani, Yukinori Minoshima, Kiyoshi Okamoto, Naoko Hata Sugi, Satoshi Nagao, Setsuo Funasaka, Hiroko Kuramochi, Takayuki Nakagawa, Masaki Mikamoto, Yukiko Miyajima, Kotaro Kodama, Yuji Yamamoto, Saori Watanabe Miyano
IC50 values for the inhibition of 93 human kinases by E7090.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::727d71c17112f88bd1dc928969d95751
https://doi.org/10.1158/1535-7163.22506370
https://doi.org/10.1158/1535-7163.22506370
Autor:
Akihiko Tsuruoka, Toshimitsu Uenaka, Masao Iwata, Junji Matsui, Tomohiro Matsushima, Toshimi Okada, Yoshinobu Yamane, Isao Ohashi, Yuki Karoji, Yusuke Nakatani, Yukinori Minoshima, Kiyoshi Okamoto, Naoko Hata Sugi, Satoshi Nagao, Setsuo Funasaka, Hiroko Kuramochi, Takayuki Nakagawa, Masaki Mikamoto, Yukiko Miyajima, Kotaro Kodama, Yuji Yamamoto, Saori Watanabe Miyano
Western blot analysis of FGFR1 in human lung cancer cell lines harboring FGFR1 amplifications.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3f0cbd7b4c4157ac6029645427248557
https://doi.org/10.1158/1535-7163.22506373
https://doi.org/10.1158/1535-7163.22506373
Autor:
Akihiko Tsuruoka, Toshimitsu Uenaka, Masao Iwata, Junji Matsui, Tomohiro Matsushima, Toshimi Okada, Yoshinobu Yamane, Isao Ohashi, Yuki Karoji, Yusuke Nakatani, Yukinori Minoshima, Kiyoshi Okamoto, Naoko Hata Sugi, Satoshi Nagao, Setsuo Funasaka, Hiroko Kuramochi, Takayuki Nakagawa, Masaki Mikamoto, Yukiko Miyajima, Kotaro Kodama, Yuji Yamamoto, Saori Watanabe Miyano
The FGFR signaling pathway has a crucial role in proliferation, survival, and migration of cancer cells, tumor angiogenesis, and drug resistance. FGFR genetic abnormalities, such as gene fusion, mutation, and amplification, have been implicated in se
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::99edbb82e8632667d9aa9e5d5b108ead
https://doi.org/10.1158/1535-7163.c.6538381.v1
https://doi.org/10.1158/1535-7163.c.6538381.v1
Autor:
Akihiko Tsuruoka, Toshimitsu Uenaka, Masao Iwata, Junji Matsui, Tomohiro Matsushima, Toshimi Okada, Yoshinobu Yamane, Isao Ohashi, Yuki Karoji, Yusuke Nakatani, Yukinori Minoshima, Kiyoshi Okamoto, Naoko Hata Sugi, Satoshi Nagao, Setsuo Funasaka, Hiroko Kuramochi, Takayuki Nakagawa, Masaki Mikamoto, Yukiko Miyajima, Kotaro Kodama, Yuji Yamamoto, Saori Watanabe Miyano
Supplementary Table legends and Supplementary Figure legends.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::32c2fb8189ca1bb305f817e3eb3cfb0e
https://doi.org/10.1158/1535-7163.22506364.v1
https://doi.org/10.1158/1535-7163.22506364.v1
Autor:
Wei Li, Ying Cheng, Shude Cui, Tao Sun, Masahide Hiraiwa, Peng Yuan, Setsuo Funasaka, Kenichi Saito, Xichun Hu, Xiaojia Wang, Qingyuan Zhang, Binghe Xu, Zhendong Chen, Quchang Ouyang
Publikováno v:
European Journal of Cancer. 112:57-65
Introduction The objective of this study was to evaluate the efficacy and safety of eribulin monotherapy, relative to vinorelbine, in Chinese women with locally recurrent/metastatic breast cancer (MBC). Methods This phase III open-label, randomised,
Autor:
Tsutomu Takashima, Hiroki Hara, Masashi Ueno, J. Furuse, Takako Eguchi Nakajima, Yasuo Komatsu, Kensei Yamaguchi, Masakazu Yashiro, Hiroshi Yabusaki, Manabu Muto, Takatoshi Sahara, Tomohiro Nishina, Tatsuya Ioka, Chigusa Morizane, Satoru Iwasa, Atsushi Miyamoto, Masataka Ikeda, Keiko Minashi, Setsuo Funasaka, Masahiro Tajika
Publikováno v:
Annals of Oncology. 31:S1292-S1293
Autor:
Masakazu Yashiro, Chigusa Morizane, Takatoshi Sahara, Masafumi Ikeda, Tatsuya Ioka, Kensei Yamaguchi, Manabu Muto, Hiroki Hara, Junji Furuse, Yoshito Komatsu, Atsushi Miyamoto, Hiroshi Yabusaki, Makoto Ueno, Taisuke Uehara, Tsutomu Takashima, Masahiro Tajika, Keiko Minashi, Satoru Iwasa, Setsuo Funasaka, Takako Nakajima, Tomohiro Nishina
Publikováno v:
Annals of Oncology. 32:S324
Autor:
Yoshito Komatsu, Takako Eguchi Nakajima, Takatoshi Sahara, Tatsuya Ioka, Kensei Yamaguchi, Tsutomu Takashima, Junji Furuse, Manabu Muto, Chigusa Morizane, Masafumi Ikeda, Tomohiro Nishina, Masakazu Yashiro, Makoto Ueno, Hiroshi Yabusaki, Atsushi Miyamoto, Satoru Iwasa, Hiroki Hara, Keiko Minashi, Setsuo Funasaka, Masahiro Tajika
Publikováno v:
Journal of Clinical Oncology. 38:538-538
538 Background: E7090 is a selective tyrosine kinase inhibitor against FGFR1-3. This first-in-human phase I study has been conducted in Japan and consists of 2 parts. Based on the toxic, pharmacokinetic, and pharmacodynamic profiles in Part 1, dose e
Autor:
Saori Watanabe-Miyano, Kiyoshi Okamoto, Kazuki Miyazaki, Setsuo Funasaka, Yoshinobu Yamane, Yoshiharu Mizui, Yoichi Ozawa, Junichi Kamata, Keigo Tanaka, Daisuke Ito, Yoshihiko Kotake, Nagao Satoshi, Osamu Toyama
Publikováno v:
Bioorganic & Medicinal Chemistry. 22:5513-5529
Hypoxia-inducible factor-1 (HIF-1) is the chief transcription factor regulating hypoxia-driven gene expression. HIF-1 overexpression is associated with poor prognosis in several cancers and therefore represents an attractive target for novel antitumo
Autor:
Masaki Mikamoto, Yusuke Nakatani, Kotaro Kodama, Hiroko Kuramochi, Akihiko Tsuruoka, Yoshinobu Yamane, Nagao Satoshi, Kiyoshi Okamoto, Saori Watanabe Miyano, Tomohiro Matsushima, Junji Matsui, Toshimitsu Uenaka, Yuji Yamamoto, Masao Iwata, Naoko Hata Sugi, Yukinori Minoshima, Yuki Karoji, Isao Ohashi, Setsuo Funasaka, Yukiko Miyajima, Toshimi Okada, Takayuki Nakagawa
Publikováno v:
Molecular cancer therapeutics. 15(11)
The FGFR signaling pathway has a crucial role in proliferation, survival, and migration of cancer cells, tumor angiogenesis, and drug resistance. FGFR genetic abnormalities, such as gene fusion, mutation, and amplification, have been implicated in se