Zobrazeno 1 - 10
of 13
pro vyhledávání: '"Sergei A Evteev"'
Publikováno v:
Journal of Chemical Information and Modeling. 63:1124-1132
Autor:
Anastasiia A. Uspenskaya, Ekaterina A. Nimenko, Radik R. Shafikov, Nikolay Y. Zyk, Sergei A. Evteev, Natalia S. Dashkova, Yan A. Ivanenkov, Alexander G. Majouga, Dmitry A. Skvortsov, Anastasiia S. Garanina, Elena K. Beloglazkina, Aleksei E. Machulkin
Publikováno v:
Medicinal Chemistry Research. 32:32-37
Autor:
Sergei V. Evteev
Publikováno v:
Vestnik MGIMO-Universiteta, Vol 38, Iss 5, Pp 237-241 (2014)
Department of German is one of the oldest language departments at MGIMO. Since its foundation in 1944 the military experienced teachers of the department, most of whom were native speakers, have begun to develop a unique method of teaching the German
Externí odkaz:
https://doaj.org/article/5ec42d9bcb994701a55253695cc52cb7
Autor:
Nikolai Y. Zyk, Anton P. Ber, Ekaterina A. Nimenko, Radik R. Shafikov, Sergei A. Evteev, Stanislav A. Petrov, Anastasia A. Uspenskaya, Natalia S. Dashkova, Yan A. Ivanenkov, Dmitry A. Skvortsov, Elena K. Beloglazkina, Alexander G. Majouga, Aleksei E. Machulkin
Publikováno v:
Bioorganicmedicinal chemistry letters. 71
We report an improved series of ligands targeting prostate specific membrane antigen (PSMA). The new compounds were designed by the introduction of changes in the structure of the aromatic fragment at ε-nitrogen atom of lysine that resulted in impro
Autor:
Anton V. Lopuhov, E. Yu. Yamansarov, Elena K. Beloglazkina, Sergei A Evteev, A. S. Olshanova, E. I. Seleznev, Alexander G. Majouga, Ya. A. Ivanenkov, Dmitry A. Skvortsov, Natalia L. Klyachko, Sergey V. Kovalev
Publikováno v:
Russian Chemical Bulletin. 69:158-163
A new promising conjugate of betulinic acid with N-acetyl-d-galactosamine was synthesized by the simple reaction sequence: esterification and copper-catalyzed azide-alkyne cycloaddition. The obtained glycoderivative exhibited high activity against he
Autor:
Ya. A. Ivanenkov, Sergey V. Kovalev, Elena K. Beloglazkina, E. Yu. Yamansarov, Natalia L. Klyachko, Nikolai V. Zyk, Rostislav A Petrov, Dmitry A. Skvortsov, Sergei A Evteev, Anton V Lopukhov, Alexander G. Majouga
Publikováno v:
Russian Chemical Bulletin. 68:2331-2338
New ligands for targeted delivery to the liver based on glycoconjugated natural triterpenoids are proposed. Simple chemical transformations of starting lupane triterpenes led to betulin or betulinic acid conjugates with N-acetyl-d-galactosamine linke
Autor:
Dmitry O Shkil, Petr V. Gorelkin, Alexander N. Lobov, V.A. Naumenko, Alexander Erofeev, Olga Y. Burenina, Yan A. Ivanenkov, Emil Yu. Yamansarov, Roman Akasov, Dmitry A. Skvortsov, Natalia L. Klyachko, Elena K. Beloglazkina, Sergey V. Kovalev, Alexander G. Majouga, Oxana Ryabaya, Elena V Lopatukhina, Ekaterina N Pavlova, Alexander Vaneev, Sergei A Evteev, Anton V Lopukhov
Publikováno v:
Bioconjugate chemistry. 32(4)
Herein, we describe the design, synthesis, and biological evaluation of novel betulin and N-acetyl-d-galactosamine (GalNAc) glycoconjugates and suggest them as targeted agents against hepatocellular carcinoma. We prepared six conjugates derived via t
Autor:
Olga Y. Burenina, Dmitrii A Grishin, Yan A. Ivanenkov, Sergey V. Kovalev, Yury V. Timchenko, Alexander Vaneev, Svetlana Yu. Maklakova, Alexander G. Majouga, Natalia L. Klyachko, Rostislav A Petrov, Alexander Erofeev, Elena K. Beloglazkina, Emil Yu. Yamansarov, Roman Timoshenko, Petr V. Gorelkin, Elena V Lopatukhina, Evgenia E Ondar, Sergei A Evteev, Anton V Lopukhov, Sofiia R Mefedova
Publikováno v:
Molecular pharmaceutics. 18(1)
In this work, we have developed covalent and low molecular weight docetaxel delivery systems based on conjugation with N-acetyl-d-galactosamine and studied their properties related to hepatocellular carcinoma cells. The resulting glycoconjugates have
Autor:
Alexander N. Lobov, Natalia L. Klyachko, Olga Y. Burenina, Ivan V Kislyakov, Yan A. Ivanenkov, Galina S Reshitko, Sergey V. Kovalev, Elena K. Beloglazkina, Irina V. Saltykova, Alexander Erofeev, Dmitry O Shkil, Emil Yu. Yamansarov, Elena V Lopatukhina, Peter Gorelkin, Anastasiia S Garanina, Olga A. Dontsova, Alexander G. Majouga, Sergei A Evteev, Anton V Lopukhov
Publikováno v:
Bioconjugate chemistry. 31(5)
Since the asialoglycoprotein receptor (also known as the "Ashwell-Morell receptor" or ASGPR) was discovered as the first cellular mammalian lectin, numerous drug delivery systems have been developed and several gene delivery systems associated with m
Autor:
Yan A. Ivanenkov, Elvira T. Yamansarova, Dmitry A. Skvortsov, Sergei A Evteev, Amina Yu. Adelgareeva, Egor I. Seleznev, Alexander G. Majouga, Emil Yu. Yamansarov, Anton V. Lopuhov, Elena K. Beloglazkina, Natalia L. Klyachko, Elena V Lopatukhina
Publikováno v:
Mendeleev Communications. 29:526-528
New allobetulin conjugates were obtained through its O-esterification with hex-5-ynoic acid followed by [3+2]-cycloaddition with three azido derivatives of N-acetyl- d -galactosamine. The conjugates are non-toxic in micromolar range against hepatocel