Zobrazeno 1 - 10
of 68
pro vyhledávání: '"Serge R. Piettre"'
Publikováno v:
European Journal of Organic Chemistry. 2022
Autor:
Baptiste Picard, Serge R. Piettre, Sonia Diab, Maxime Beuvin, Julien Legros, Maxime Manneveau, Isabelle Chataigner, Morgane Sanselme
Publikováno v:
Tetrahedron Letters
Tetrahedron Letters, Elsevier, 2018, 59 (51), pp.4487-4491. ⟨10.1016/j.tetlet.2018.11.020⟩
Tetrahedron Letters, Elsevier, 2018, 59 (51), pp.4487-4491. ⟨10.1016/j.tetlet.2018.11.020⟩
International audience; An efficient access to 4-aryl imidazole scaffolds is described in two steps and one operation. Cyanoaryl-imidazolines are easily obtained by a (3 + 2) heterocyloaddition involving cyanobenzenes as dipolarophiles and a non-stab
Publikováno v:
Journal of Organic Chemistry
Journal of Organic Chemistry, American Chemical Society, 2019, 84 (9), pp.5245-5260. ⟨10.1021/acs.joc.9b00232⟩
Journal of Organic Chemistry, American Chemical Society, 2019, 84 (9), pp.5245-5260. ⟨10.1021/acs.joc.9b00232⟩
International audience; A simple, two-step procedure to convert α,α-difluorinated H-phosphinic acids into the corresponding H-phosphinothioates is described. The usefulness of these species is demonstrated by their transformation into difluorinated
Autor:
Serge R. Piettre, Karine Pasturaud, Fabien Chapellas, Sonia Diab, Manuel Andreini, Julien Legros, Isabelle Chataigner
Publikováno v:
Organic and Biomolecular Chemistry
Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2016, 14 (10), pp.2833-2839. ⟨10.1039/c5ob02595h⟩
Organic and Biomolecular Chemistry, Royal Society of Chemistry, 2016, 14 (10), pp.2833-2839. ⟨10.1039/c5ob02595h⟩
International audience; Nucleophilic enamines add spontaneously on heteroarenes 3-nitroindole and benzofuran to form a new C–C bond. With nitroindole (1) and enamine (2a), an unprecedented dearomatizing formal ene reaction occurs in a totally regio
Publikováno v:
The Journal of Organic Chemistry. 74:1237-1246
Dearomatization of electron-poor benzofurans is possible through involvement of the aromatic 2,3-carbon-carbon double bond as dienophile in normal electron demand [4 + 2] cycloadditions. The tricyclic heterocycles thereby produced bear a quaternary c
Autor:
Serge R. Piettre, Isabelle Chataigner
Publikováno v:
Organic Letters. 9:4159-4162
Activation by high pressure allows 3-nitroindole and 3-nitropyrrole derivatives to behave as electron-poor heterodienes in multicomponent domino [4+2]/[3+2] cycloaddition processes. The primary [4+2] inverse demand cycloaddition appears to be complet
Publikováno v:
The Journal of Organic Chemistry. 71:31-37
[reaction: see text] Selanylated difluoromethylphosphonates and difluoromethylphosphonothioates are good precursors to phosphonodifluoromethyl and phosphonothiodifluoromethyl radicals, respectively. When generated in the presence of alkenes and a hyd
Publikováno v:
Tetrahedron Letters. 46:8027-8031
Alcohols are solvents of choice to react boronates, aldehydes and either primary or secondary amines. Thus, while the reaction proceeds sluggishly, or not at all, in aprotic solvents, the desired aminoacids are in most cases obtained in high yields w
Publikováno v:
Tetrahedron. 61:4755-4759
An improved, convergent synthesis of CB92834 is relying on a Suzuki cross-coupling reaction and easily allows multigram-scale preparation of the compound. The approach features three highly stereoselective steps.
Publikováno v:
Tetrahedron. 60:4895-4900
A practical, eight-step synthesis of the key intermediate 14 in 19% overall yield from α- d -xylose is described. The preparation can be carried out on multi-gram scale and involves the use of the organomagnesium reagent 2d . The capability of deriv