Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Santosh Jangir"'
Autor:
Sanjay Krishna, Sonal Gupta, Mala Singh, Jagdamba P. Maikhuri, Satya Narayan Sankhwar, Santosh Jangir, Veenu Bala, Gopal Gupta, Dhanaraju Mandalapu, Kavita Rawat, Hardik Chandasana, Bhavana Kushwaha, R.P. Tripathi, Atul Krishna, Praveen K. Shukla, Yashpal S. Chhonker, Vishnu L. Sharma, Mohammad Imran Siddiqi, Rabi Sankar Bhatta
Publikováno v:
European Journal of Medicinal Chemistry. 101:640-650
The growing population and health-care burden (due to STIs and HIV) imposes a particular economic crisis over resource-poor countries. Thus a novel approach as vaginal microbicides emerges as integrated tool to control both population and anti-STIs/H
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ea890e44e76df6386b91a171c2a30237
https://doi.org/10.1016/j.ejmech.2015.07.021
https://doi.org/10.1016/j.ejmech.2015.07.021
Autor:
Mohammad Imran Siddiqi, Hardik Chandasana, Gopal Gupta, Dhanaraju Mandalapu, Vishnu L. Sharma, Veenu Bala, Rabi Sankar Bhatta, Yashpal S. Chhonker, Jagdamba P. Maikhuri, Sanjay Krishna, Santosh Jangir, Sonal Gupta, Bhavana Kushwaha, Kavita Rawat, Nand Lal, R.P. Tripathi
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 25:881-886
Prophylactic prevention is considered as the most promising strategy to tackle STI/HIV. Twenty-five dithiocarbamate-thiourea hybrids (14-38) were synthesized as woman controlled topical vaginal microbicides to counter Trichomonas vaginalis and sperm
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2a23492f2fc3bbd7b8ff4f7f530763e4
https://doi.org/10.1016/j.bmcl.2014.12.062
https://doi.org/10.1016/j.bmcl.2014.12.062
Autor:
Praveen K. Shukla, Vikas Kumar, Veenu Bala, Gopal Gupta, Dhanaraju Mandalapu, Sonal Gupta, Rabi Sankar Bhatta, Santosh Jangir, Yashpal S. Chhonker, Lalit Kumar, Vishnu L. Sharma, Jagdamba P. Maikhuri, Bhavana Kushwaha, Atul Krishna
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 24:5782-5786
A series of seventeen morpholin/piperidin-1-yl-carbamodithioate (3-19) were synthesized as topical vaginal microbicidal spermicides. The synthesized compounds were evaluated for their anti-Trichomonas activity against MTZ susceptible and resistant st
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4a405e827459e1209fb5466963ed99d0
https://doi.org/10.1016/j.bmcl.2014.10.040
https://doi.org/10.1016/j.bmcl.2014.10.040
Autor:
Lalit Kumar, Veenu Bala, Amit Sarswat, Karthik Nandikonda, Santosh Jangir, Nand Lal, Vishnu L. Sharma
Publikováno v:
Journal of Heterocyclic Chemistry. 52:156-162
A green and facile synthesis of dithiocarbamate derivatives containing disulfide linkage by the ring opening reaction of trithiocarbonate with amines under solvent and catalyst-free condition with excellent yields is being reported. Environmental ben
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7e8e0d22567f1e7a7ff093d2121c4067
https://doi.org/10.1002/jhet.1995
https://doi.org/10.1002/jhet.1995
Autor:
Pratiksha Singh, Gopal Gupta, Veenu Bala, Vishnu L. Sharma, Nand Lal, Amit Sarswat, Santosh Jangir, Praveen K. Shukla, Bhavana Kushwaha, Lokesh Kumar, Jagdamba P. Maikhuri, Lalit Kumar
Publikováno v:
Org. Biomol. Chem.. 12:3090-3099
1-Substituted piperazinecarbodithioates were obtained by an unusual removal of CS2 in benzyl substituted dithiocarbamate derivatives under acid and basic conditions during design and synthesis of 1,4-(disubstituted)piperazinedicarbodithioates as doub
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::36cc27fc6b53e0bd62d16a41e6f276fd
https://doi.org/10.1039/c4ob00005f
https://doi.org/10.1039/c4ob00005f
Autor:
Vishnu L. Sharma, Mohammad Imran Siddiqi, Praveen K. Shukla, Sanjay Krishna, Amit Sarswat, Tara Rawat, Gopal Gupta, Dhanaraju Mandalapu, Atindra K. Pandey, Veenu Bala, Jagdamba P. Maikhuri, Santosh Jangir, Lokesh Kumar, Ashish Jain, Bhavana Kushwaha, Nand Lal, Lalit Kumar
Publikováno v:
European journal of medicinal chemistry. 115
Trichomoniasis and candidiasis are amongst the most common morbidity-causing reproductive tract infections, generally treated by Metronidazole and Fluconazole respectively. Poor vaginal efficacy, drug-resistance and non-spermicidal nature limit their
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5ec6075838eed043e1f06efd5cbe7e76
https://pubmed.ncbi.nlm.nih.gov/27084496
https://pubmed.ncbi.nlm.nih.gov/27084496
Publikováno v:
Organic Letters. 13:2330-2333
A facile synthesis of S-(2-thioxo-1,3-dithiolan-4-yl)methyl dialkylcarbamothioates (3) and S-thiiran-2-ylmethyl dialkylcarbamothioate (5) has been reported by the reaction of 5-(chloromethyl)-1,3-oxathiolane-2-thione (1) with sodium dialkylcarbamodit
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::eec1eab63c5cdbdc90572753a64a78eb
https://doi.org/10.1021/ol2005825
https://doi.org/10.1021/ol2005825
Autor:
Karthik Nandikonda, Veenu Bala, Vishnu L. Sharma, Santosh Jangir, Nand Lal, Lalit Kumar, Amit Sarswat
Publikováno v:
ChemInform. 46
A green and facile synthesis of dithiocarbamate derivatives containing disulfide linkage by the ring opening reaction of trithiocarbonate with amines under solvent and catalyst-free condition with excellent yields is being reported. Environmental ben
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3900ae48f516b57de051454a504d4655
https://doi.org/10.1002/chin.201524074
https://doi.org/10.1002/chin.201524074
Publikováno v:
Current molecular pharmacology. 7(2)
The spermatogenesis is a precisely-timed cellular proliferation that takes place in the seminiferous tubules of testes and is meticulously regulated by gonadotrophins, androgens and temperature. Hormonal, nonhormonal and thermal methods of male contr
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8a543287c88ef9211dc2e393c6b6f0bf
https://pubmed.ncbi.nlm.nih.gov/25620226
https://pubmed.ncbi.nlm.nih.gov/25620226
Autor:
Amit Kumar, Vishnu L. Sharma, Vikas Verma, Veenu Bala, Vikas Sharma, Jagdamba P. Maikhuri, Amit Sarswat, Gopal Gupta, Nand Lal, Lalit Kumar, Karan Singh Saini, Hamidullah, Santosh Jangir, Rituraj Konwar
Publikováno v:
European journal of medicinal chemistry. 85
A new series of 2-(alkoxy(hydroxy)phosphoryloxy)ethyl dialkylcarbodithioate derivatives was synthesized and evaluated against endocrine related cancers, acting via modulation of Akt-pathway. Eighteen compounds were active at 7.24–100 μM against MD
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d0f8693e4c4cef967ae2d83f430f577c
https://pubmed.ncbi.nlm.nih.gov/25128666
https://pubmed.ncbi.nlm.nih.gov/25128666