Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Sanjay Gite"'
Autor:
Jigar N. Desai, Bhaumin Patel, Archana Gite, Nandini Panchal, Sanjay Gite, Anil Argade, Jeevan Kumar, Sachchidanand s, Debdutta Bandyopadhyay, KRISHNARUP DASTIDAR, Hoshang Patel, Abhijit Chatterjee, Jogeshwar Mahapatra, Manoranjan Sharma, Poonam Giri, Sanjay Kumar, Mukul Jain, Rajiv Sharma, Ranjit Desai
Publikováno v:
Bioorganicmedicinal chemistry letters. 66
Dysregulated JAK-STAT signaling has been proven to be involved in several immune-mediated diseases. Several janus kinase (JAK) inhibitors have been approved for the treatment of various inflammatory and autoimmune diseases such as rheumatoid arthriti
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::562f5c0d97c9943bcf89352c107b020c
https://pubmed.ncbi.nlm.nih.gov/35413417
https://pubmed.ncbi.nlm.nih.gov/35413417
Autor:
Debdutta Bandyopadhyay, Jigar Desai, Abhijit Chatterjee, Hoshang Patel, S. Sachchidanand, Rajesh Bahekar, Jeevan Kumar, Dipam Patel, Krishnarup Ghoshdastidar, Anil Argade, Harilal Patel, Archana Gite, Bhaumin Patel, Sanjay Gite, Jogeswar Mahapatra, Nandini Panchal, Rajesh Sundar, Ranjit C. Desai, Shubhangi S. Soman
Publikováno v:
Bioorganic Chemistry. 99:103851
Selective inhibition of janus kinase (JAK) has been identified as an important strategy for the treatment of autoimmune disorders. Optimization at the C2 and C4-positions of pyrimidine ring of Cerdulatinib led to the discovery of a potent and orally
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1f57c25ee9d80ecff1fec355cd350348
https://doi.org/10.1016/j.bioorg.2020.103851
https://doi.org/10.1016/j.bioorg.2020.103851
Autor:
Anil Argade, Pravin Thombare, Mukul R. Jain, Sanjay Gite, Vijay M. Prajapati, Jigar Desai, Kiran Shah, Pankaj R. Patel, Bipin Pandey, Rajesh Bahekar
Publikováno v:
Synthetic Communications. 42:3140-3149
One-pot synthesis of 3,4-diaryl substituted 2(5H)-furanones was established and its commercial application has been demonstrated by accomplishing total synthesis of rofecoxib, under mild reaction conditions, with good yields and purity.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e1c8e11aa3d9d51d929cf9953cd9d66b
https://doi.org/10.1080/00397911.2011.577923
https://doi.org/10.1080/00397911.2011.577923
Autor:
Pankaj R. Patel, Kiran Shah, Jigar Desai, Pravin Thombare, Sanjay Gite, Laxmikant S. Pavase, Anil Argade
Publikováno v:
Synthetic Communications. 41:748-753
A convenient and cost-effective synthesis of pharmacologically important tert-butyl-2-(4-2-aminoethyl)phenylthio)-2-methylpropanoate from commercially available 2-2-phenyl-1-ethanol is described.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::fb8bae8b146417a9d99f83d7b8627f7f
https://doi.org/10.1080/00397911003644399
https://doi.org/10.1080/00397911003644399
Autor:
Anil Argade, Pravin Thombare, Jigar Desai, Laxmikant Pavase, Kiran Shah, Sanjay Gite, Pankaj R. Patel
Publikováno v:
Synthetic Communications. 39:2423-2429
4-Aryl-substituted 2(5H)-furanones were prepared by reaction of diethylphosphono acetic acid and phenacyl bromides, followed by an intramolecular Horner–Emmons-type cyclization. Both the reactions were carried out in situ to give the desired 4-aryl
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3969e9834c0bf260cf897a740d080ace
https://doi.org/10.1080/00397910802656026
https://doi.org/10.1080/00397910802656026
Autor:
Pravin Thombare, Pankaj R. Patel, Laxmikant S. Pavase, Sanjay Gite, Anil Argade, Kiran Shah, Jigar Desai
Publikováno v:
ChemInform. 42
A convenient and cost-effective synthesis of pharmacologically important tert-butyl-2-(4-2-aminoethyl)phenylthio)-2-methylpropanoate from commercially available 2-2-phenyl-1-ethanol is described.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8ad8004aa2331f20b4c5e1d33b15ad6e
https://doi.org/10.1002/chin.201132073
https://doi.org/10.1002/chin.201132073
Autor:
Pankaj R. Patel, Abhijit Chatterjee, Amit Joharapurkar, Debdutta Bandyopadhyay, Anil Argade, Ganes Chakrabarti, Rajesh Sunder, Sanjay Gite, Mubeen Shaikh, Jigar Desai, Kalapatapu V.V.M. Sairam, Ramchandra Ranvir, Harilal Patel, Jogeswar Mahapatra, Rajesh Bahekar, Kiran Shah, Mukul R. Jain, Pravin Thombare
Publikováno v:
MedChemComm. 2:966
A new series of γ-lactam hydroxamate based TACE inhibitors was designed mainly by introducing various substitutions at the 2nd position of the quinoline nucleus to achieve high potency and good selectivity towards TACE over matrix metalloproteases (
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::faa0ff83f0fc635d35972a8e3536648a
https://doi.org/10.1039/c0md00261e
https://doi.org/10.1039/c0md00261e