Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Sangram Keshari, Saraf"'
Autor:
Kiran Kumar Kandukuri, Anil Shinde, Santoshkumar Pandey, Thrinath Reddy Bandyala, Abdul Rasheed Mohammed, Raghava Choudary Palacharla, Ramkumar Subramanian, Kumar Bojja, Sravanthi Manchineella, Pramod Kumar Achanta, Sangram Keshari Saraf, Venkat Jasti, Ramakrishna Nirogi, Rajesh Kumar Badange, Pradeep Jayarajan, Vijay Benade, Veena Reballi
Publikováno v:
Journal of Medicinal Chemistry. 62:1203-1217
A series of chemical optimizations guided by in vitro affinity at a histamine H3 receptor (H3R), physicochemical properties, and pharmacokinetics in rats resulted in identification of N-[4-(1-cyclobutyl-piperidin-4-yloxy)phenyl]-2-(morpholin-4-yl)ace
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3a6a6e9590419cd78629224ee0312c10
https://doi.org/10.1021/acs.jmedchem.8b01280
https://doi.org/10.1021/acs.jmedchem.8b01280
Autor:
Sangram Keshari Saraf, Vinod Kumar Goyal, Ramkumar Subramanian, Rama Sastry Kambhampati, Venugopalarao Bhatta, Abdul Rasheed Mohammed, Ramakrishna Nirogi, Thrinath Reddy Bandyala, Gopinadh Bhyrapuneni, Rajesh Kumar Badange, Raghava Choudary Palacharla, Kumar Bojja, Venkat Jasti, Veena Reballi, Vijay Benade, Pradeep Jayarajan, Anil Shinde
Publikováno v:
Journal of Medicinal Chemistry. 60:1843-1859
Optimization of a novel series of 3-(piperazinylmethyl) indole derivatives as 5-hydroxytryptamine-6 receptor (5-HT6R) antagonists resulted in identification of 1-[(2-bromophenyl)sulfonyl]-5-methoxy-3-[(4-methyl-1-piperazinyl)methyl]-1H-indole dimesyl
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::bd524b552dd775bcb94861bf46741193
https://doi.org/10.1021/acs.jmedchem.6b01662
https://doi.org/10.1021/acs.jmedchem.6b01662
Autor:
Ramakrishna, Nirogi, Anil, Shinde, Abdul Rasheed, Mohammed, Rajesh Kumar, Badange, Veena, Reballi, Thrinath Reddy, Bandyala, Sangram Keshari, Saraf, Kumar, Bojja, Sravanthi, Manchineella, Pramod Kumar, Achanta, Kiran Kumar, Kandukuri, Ramkumar, Subramanian, Vijay, Benade, Raghava Choudary, Palacharla, Pradeep, Jayarajan, Santoshkumar, Pandey, Venkat, Jasti
Publikováno v:
Journal of medicinal chemistry. 62(3)
A series of chemical optimizations guided by in vitro affinity at a histamine H
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::d3bc504790aa828f322e741792955470
https://pubmed.ncbi.nlm.nih.gov/30629436
https://pubmed.ncbi.nlm.nih.gov/30629436
Autor:
Ramakrishna, Nirogi, Anil, Shinde, Rama Sastry, Kambhampati, Abdul Rasheed, Mohammed, Sangram Keshari, Saraf, Rajesh Kumar, Badange, Thrinath Reddy, Bandyala, Venugopalarao, Bhatta, Kumar, Bojja, Veena, Reballi, Ramkumar, Subramanian, Vijay, Benade, Raghava Choudary, Palacharla, Gopinadh, Bhyrapuneni, Pradeep, Jayarajan, Vinod, Goyal, Venkat, Jasti
Publikováno v:
Journal of medicinal chemistry. 60(5)
Optimization of a novel series of 3-(piperazinylmethyl) indole derivatives as 5-hydroxytryptamine-6 receptor (5-HT
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::d0e4e406b5e20ebd25f2983a863c4079
https://pubmed.ncbi.nlm.nih.gov/28212021
https://pubmed.ncbi.nlm.nih.gov/28212021
Autor:
Rajesh Babu Medapati, Sangram Keshari Saraf, Narender Ganuga, Renny Abraham, Hemasundar Reddy Talakanti, Jayaprakash Tadiparthi, Ramakrishna Nirogi, Venkat Jasti, Venkata Ramalingayya Grandhi, Pradeep Jayarajan
Publikováno v:
Alzheimer's & Dementia. 15:P604-P604
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::dde0eefcd22b77fd9a3a3111bfde513d
https://doi.org/10.1016/j.jalz.2019.06.2490
https://doi.org/10.1016/j.jalz.2019.06.2490
Autor:
Sangram Keshari Saraf, Renny Abraham, Venkatesh Kamuju, Ramakrishna Nirogi, Shantaveer Irappanavar, Laxman Kota, Ranjith Kumar Ponnamaneni, Gopinadh Bhyrapuneni, Vijay Benade, Pradeep Jayarajan
Publikováno v:
Alzheimer's & Dementia. 11
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::33f978a5d147c71481efb10a6ca3640a
https://doi.org/10.1016/j.jalz.2015.06.526
https://doi.org/10.1016/j.jalz.2015.06.526