Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Sandesh, Jatheendranath"'
Autor:
Venkatraman, Janani *, Bhat, Jyothi, Solapure, Suresh M., Sandesh, Jatheendranath, Sarkar, Debasmita, Aishwarya, Sundaram, Mukherjee, Kakoli, Datta, Santanu, Malolanarasimhan, Krishnan, Bandodkar, Balachandra, Das, Kaveri S.
Publikováno v:
In SLAS Discovery March 2012 17(3):293-302
Autor:
Sandesh Jatheendranath, Gayathri Balakrishnan, Sreenivasaiah Menasinakai, Sudha Ravishankar, Vasanthi Ramachandran, Sreevalli Sharma, Charles J. Eyermann, Anisha Ambady, Suresh Rudrapatna, Naina Vinay Mudugal, Disha Awasthy, Umender Sharma, Supreeth Guptha, Vasan K. Sambandamurthy, Radha Nandishaiah, Folkert Reck
Publikováno v:
Tuberculosis. 95:589-598
DNA topoisomerases perform the essential function of maintaining DNA topology in prokaryotes. DNA gyrase, an essential enzyme that introduces negative supercoils, is a clinically validated target. However, topoisomerase I (Topo I), an enzyme responsi
Autor:
David Waterson, Stefan Kavanagh, V. Balasubramanian, Vijender Panduga, Francisco-Javier Gamo, María Santos Martínez, Shahul Hameed P, Vinayak Hosagrahara, María Belén Jiménez-Díaz, Shubhada Barde, Kakoli Mukherjee, Sandra Duffy, Santiago Ferrer, Vikas Patil, Balachandra Bandodkar, Ramachandran Sreekanth A, K.R. Prabhakar, Suresh Rudrapatna, Praveena Manjrekar, Iñigo Angulo-Barturen, Pravin Iyer, Vasan K. Sambandamurthy, Nikhil Rautela, Pamela Magistrado, Dyann F. Wirth, Sowmya Bharath, Chandan Narayan, Sapna Morayya, Murugan Chinnapattu, Pavithra Viswanath, Anandkumar Raichurkar, Krishna Koushik, Jitender Reddy, Vicky M. Avery, Achyut Sinha, Amanda K. Lukens, Disha Awasthy, Shridhar Narayanan, Laura M. Sanz, Gajanan Shanbag, Sandesh Jatheendranath, Abhishek Srivastava, Ramanatha Saralaya
Publikováno v:
Journal of medicinal chemistry. 57(13)
Whole-cell high-throughput screening of the AstraZeneca compound library against the asexual blood stage of Plasmodium falciparum (Pf) led to the identification of amino imidazoles, a robust starting point for initiating a hit-to-lead medicinal chemi
Autor:
Monalisa Chatterji, João Neres, Sreevalli Sharma, Prashanti Madhavapeddi, Vijender Panduga, James D. Whiteaker, Suresh Rudrapatna, Chandan Narayan, Krishna Koushik, Laurent R. Chiarelli, Gajanan Shanbhag, Vaishali Humnabadkar, Gopinath Gorai, Claudia Binda, Sandeep R. Ghorpade, Radha Shandil, Neeraj Dhar, Maria Rosalia Pasca, Stefan Kavanagh, Vasan K. Sambandamurthy, M. R. Manjunatha, K.R. Prabhakar, Vijayashree Achar, John D. McKinney, Neela Dinesh, Naina Hegde, Praveena Manjrekar, François Signorino-Gelo, Parvinder Kaur, Shridhar Narayanan, Jitendar Reddy, Subramanyam J. Tantry, Ashwini Narayan, Sandesh Jatheendranath, Lalit kumar Jena, Tommasi Ruben A, Jyothi Mahadevaswamy, Disha Awasthy, Ramanatha Saralaya, Manoranjan Panda, Bob McLaughlin, Anisha Ambady, Vinayak Hosagrahara, Pravin Iyer, Chandramohan Bathula, Maruti Naik, Giovanna Riccardi, Supreeth Guptha, Sudha Ravishankar, Vasanthi Ramachandran
Publikováno v:
Journal of medicinal chemistry. 57(12)
4-Aminoquinolone piperidine amides (AQs) were identified as a novel scaffold starting from a whole cell screen, with potent cidality on Mycobacterium tuberculosis (Mtb). Evaluation of the minimum inhibitory concentrations, followed by whole genome se
Autor:
Venkatraman, Janani, Bhat, Jyothi, Solapure, Suresh M., Sandesh, Jatheendranath, Sarkar, Debasmita, Aishwarya, Sundaram, Mukherjee, Kakoli, Datta, Santanu, Malolanarasimhan, Krishnan, Bandodkar, Balachandra, Das, Kaveri S.
Publikováno v:
SLAS Discovery: Advancing Life Sciences R&D; March 2012, Vol. 17 Issue: 3 p293-302, 10p