Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Sandeep Kumar Marvadi"'
Autor:
R. Gajendra Reddy, Goverdhan Surineni, Dwaipayan Bhattacharya, Sandeep Kumar Marvadi, Arpita Sagar, Arunasree M. Kalle, Arvind Kumar, Srinivas Kantevari, Sumana Chakravarty
Publikováno v:
ACS Omega, Vol 4, Iss 17, Pp 17279-17294 (2019)
Externí odkaz:
https://doaj.org/article/8776df72d7eb4de494462e78fc2e8c9f
Autor:
Dharmarajan Sriram, Srinivas Kantevari, Syeda Safoora, Devendra Nagineni, Vagolu Siva Krishna, Sandeep Kumar Marvadi
Publikováno v:
Monatshefte für Chemie - Chemical Monthly. 151:405-415
A series of novel 5-chloro-2-(thiophen-2-yl)-7,8-dihydroquinoline-6-carboxamides was designed, synthesized, and evaluated for antitubercular activity. The required 5-chloro-2-(thiophen-2-yl)-7,8-dihydroquinoline-6-carboxylic acid intermediate was pre
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7295c7a87f66dc7b6a363b4926ebe0fc
https://doi.org/10.1007/s00706-020-02560-2
https://doi.org/10.1007/s00706-020-02560-2
Autor:
Sumana Chakravarty, R. Gajendra Reddy, Arvind Kumar, Arunasree M. Kalle, Goverdhan Surineni, Arpita Sagar, Dwaipayan Bhattacharya, Sandeep Kumar Marvadi, Srinivas Kantevari
Publikováno v:
ACS Omega, Vol 4, Iss 17, Pp 17279-17294 (2019)
ACS Omega
ACS Omega
Small-molecule inhibitors of HDACs (HDACi) induce hyperacetylation of histone and nonhistone proteins and have emerged as potential therapeutic agents in most animal models tested. The established HDACi vorinostat and tubastatin-A alleviate neurodege
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aa5c8626266a7416d57bb481de5f80e6
https://doaj.org/article/8776df72d7eb4de494462e78fc2e8c9f
https://doaj.org/article/8776df72d7eb4de494462e78fc2e8c9f
Autor:
Vagolu Siva Krishna, Alexandrina S. Volobueva, Dharmarajan Sriram, Sandeep Kumar Marvadi, Vladimir V. Zarubaev, Ekaterina O. Sinegubova, Dmitry G. Tentler, Yana L Esaulkova, Srinivas Kantevari, Anna A. Muryleva
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 29:2664-2669
This study describes synthesis and evaluation of novel 5-Chloro-2-thiophenyl-1,2,3-triazolylmethyldihydroquinolines 7a-o as dual inhibitors of Mycobacterium tuberculosis and influenza virus. Huisgen’s [3+2] dipolar cycloaddition of 6-(azidomethyl)-
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::00be46294ecdfeb39d5b61aa7861a2f9
https://doi.org/10.1016/j.bmcl.2019.07.040
https://doi.org/10.1016/j.bmcl.2019.07.040
Autor:
B. Sridhar, Sandeep Kumar Marvadi, Dharmarajan Sriram, Goverdhan Surineni, Srinivas Kantevari, Rudraraju Srilakshmi Reshma, Vagolu Siva Krishna
Publikováno v:
Bioorganic chemistry. 96
We, herein, describe the synthesis of a series of novel aryl tethered 7,8-dihydroquinolin-5(6H)-ylidenehydrazinecarbothioamides 4a–v, which showed in vitro and in vivo antimycobacterial activity against Mycobacterium tuberculosis (Mtb) H37Rv. The i
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::23a48e0a4265a67b37e97085531387ea
https://pubmed.ncbi.nlm.nih.gov/32007719
https://pubmed.ncbi.nlm.nih.gov/32007719
Publikováno v:
Bioorganicmedicinal chemistry letters. 29(4)
A series of novel substituted 1,2,3-triazolyldihydroquinolines 6a–o was designed and synthesized from 2-acetylthiophene in five-step reaction sequence involving modified Boltzmann-Rahtz reaction of β-Enaminone; Vilsmeier-Haack chloroformylation us
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9435ecf11e459c31b54456fde2b02d7d
https://pubmed.ncbi.nlm.nih.gov/30638877
https://pubmed.ncbi.nlm.nih.gov/30638877
Publikováno v:
European journal of medicinal chemistry. 164
A series of novel morpholine, thiomorpholine and N-substituted piperazine coupled 2-(thiophen-2-yl)dihydroquinolines 7a–p was designed and synthesized from 2-acetyl thiophene in six step reaction sequence involving modified Bohlmann-Rahtz and Vilsm
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3553d06af700edbfdb78d75f2e16d994
https://pubmed.ncbi.nlm.nih.gov/30594675
https://pubmed.ncbi.nlm.nih.gov/30594675
Autor:
Sandeep Kumar Marvadi, Srinivas Kantevari, Goverdhan Surineni, Perumal Yogeeswari, Dharmarajan Sriram
Publikováno v:
Bioorganicmedicinal chemistry letters. 28(9)
Herein described the design, synthesis and antitubercular evaluation of novel series of dibenzofuran, dibenzothiophene and N-methyl carbazole tethered 2-aminothiazoles and their cinnamamide analogs. One pot condensation of N-methyl carbazole, dibenzo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5c68bf5a697b3409a592c27bfaae26ad
https://pubmed.ncbi.nlm.nih.gov/29598909
https://pubmed.ncbi.nlm.nih.gov/29598909