Hybridization of cluster-based LDA and ANN for student performance prediction and comments evaluation

Autor: Munish Saini, Sakshi Sood

Publikováno v: Education and Information Technologies. 26:2863-2878

For a productive life, education plays a critical role to fill individual life with value and excellence. Education is compulsory to provide things that individuals partake in to compete in the modern world. Predicting the academic performance of the

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::ee73fb6c10200ef07aee3dd51eb07bbe
https://doi.org/10.1007/s10639-020-10381-3

Design and Synthesis of Imidazole and Triazole Pyrazoles as

Autor: Safaa M, Kishk, Kirsty J, McLean, Sakshi, Sood, Darren, Smith, Jack W D, Evans, Mohamed A, Helal, Mohamed S, Gomaa, Ismail, Salama, Samia M, Mostafa, Luiz Pedro S, de Carvalho, Colin W, Levy, Andrew W, Munro, Claire, Simons

Publikováno v: ChemistryOpen

The emergence of untreatable drug‐resistant strains of Mycobacterium tuberculosis is a major public health problem worldwide, and the identification of new efficient treatments is urgently needed. Mycobacterium tuberculosis cytochrome P450 CYP121A1

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::1d298e8d5dc90c56f271092380f9a770
https://pubmed.ncbi.nlm.nih.gov/31367508

Synthesis and biological evaluation of novel cYY analogues targeting Mycobacterium tuberculosis CYP121A1

Autor: Safaa M Kishk, McLean, Kirsty J, Sakshi Sood, Helal, Mohamed A, Gomaa, Mohamed S, Salama, Ismail, Mostafa, Samia M, Luiz Pedro S De Carvalho, Munro, Andrew W, Simons, Claire

The rise in multidrug resistant (MDR) cases of tuberculosis (TB) has led to the need for the development of TB drugs with different mechanisms of action. The genome sequence of Mycobacterium tuberculosis (Mtb) revealed twenty different genes coding f

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::2a53f983322c567c2ecead8c5434cd51

Novel aryl substituted pyrazoles as small molecule inhibitors of cytochrome P450 CYP121A1: Synthesis and antimycobacterial evaluation

Autor: Sakshi Sood, Hosam A. Elshihawy, Colin Levy, Beyza Torun, Leonardo B. Marino, Dania Altuwairigi, Kirsty J. McLean, Ismail M. Taban, Adeline S. T. Ngu, Clare J. Williamson, Luiz Pedro S. de Carvalho, Benedetta Zucchini, Andrew W. Munro, Claire Simons

Publikováno v: Taban, I M, Elshihawy, H E A E, Torun, B, Zucchini, B, Williamson, C J, Altuwairigi, D, Ngu, A S T, Mclean, K, Levy, C, Sood, S, Marino, L B, Munro, A, De Carvalho, L P S & Simons, C 2017, ' Novel Aryl Substituted Pyrazoles as Small Molecule Inhibitors of Cytochrome P450 CYP121A1: Synthesis and Antimycobacterial Evaluation ', Journal of Medicinal Chemistry . https://doi.org/10.1021/acs.jmedchem.7b01562
Journal of Medicinal Chemistry

Three series of biarylpyrazole imidazole and triazoles are described, which vary in the linker between the biaryl pyrazole and imidazole/triazole group. The imidazole and triazole series with the short −CH2– linker displayed promising antimycobac

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6f3ced2aae350e0c2cb8935d17611657

Edonamides, the first secondary metabolites from the recently described myxobacterium Aggregicoccus edonensis

Autor: Marc Stadler, Steffen Bernecker, Kathrin I. Mohr, Rolf Jansen, Sakshi Sood, Sabrina Karwehl

Publikováno v: Tetrahedron Letters. 56:6402-6404

Two fatty acid styryl amides, edonamides A ( 1 ) and B ( 2 ), were isolated as the first secondary metabolites from the recently described myxobacterial genus and family Aggregicoccus edonensis . Their molecular structures were elucidated using exten

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3aea071465ed4ef4d172578742bf1fb8
https://doi.org/10.1016/j.tetlet.2015.09.139