Výsledky vyhledávání - "SHRINIVAS D. JOSHI"

Akademický článek

Ionic liquid Mediated Pd-catalyzed sonochemistry for facile synthesis of carbazoles: Molecular Modelling and antimicrobial studies

Autor: Imamhusen Jamadar, Athmanand Anchi, Shruti S. Malunavar, Rajesh G. Kalkhambkar, Suraj M. Sutar, Shrinivas D. Joshi

Publikováno v: Tetrahedron Green Chem, Vol 3, Iss , Pp 100038- (2024)

Herein we have described the Pd-catalyzed sonochemistry driven by [BMIM]-IL as re-useable solvent to synthesize various carbazole scaffolds from 2,2′-dibromodiphenyl. Diverse primary amines were utilised as coupling partners in the presence of [PAI

Externí odkaz: https://doaj.org/article/bd73e6a25bc34fd4990f9204a383acc6

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Akademický článek

Synthesis, molecular docking study and biological evaluation of new pyrrole scaffolds as potential antitubercular agents for dual targeting of enoyl ACP reductase and dihydrofolate reductase

Autor: Mater H. Mahnashi, Sravanthi Avunoori, Sanjay Gopi, Ibrahim Ahmed Shaikh, Ahmed Saif, Farkad Bantun, Hani Saleh Faidah, Abdulrahman Ali Alhadi, Jaber Hassan Alshehri, Abdullah Ali Alharbi, Prem Kumar S. R., Shrinivas D. Joshi

Publikováno v: PLoS ONE, Vol 19, Iss 5 (2024)

Externí odkaz: https://doaj.org/article/05d6beda2b284e288f690485448d86c4

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Akademický článek

In vitro antimicrobial combat, molecular modelling and structure activity relationship studies of novel class of aryl-ethyne tethered coumarin analogues and some 3-aryl coumarin derivatives

Autor: Pavankumar Prabhala, Suraj M. Sutar, Hemantkumar M. Savanur, Shrinivas D. Joshi, Rajesh G. Kalkhambkar

Publikováno v: European Journal of Medicinal Chemistry Reports, Vol 5, Iss , Pp 100048- (2022)

A series of novel class of aryl ethyne-tethered coumarin analogues (series 1) and some 3-aryl coumarin cognates (series 2) were synthesized, and their in vitro antimicrobial activities aided by molecular modelling and the structure activity relations

Externí odkaz: https://doaj.org/article/c6412ae62302463394ecebd8f7208748

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Akademický článek

Synthesis, Molecular Docking Study, and Biological Evaluation of New 4-(2,5-Dimethyl-1H-pyrrol-1-yl)-N’-(2-(substituted)acetyl)benzohydrazides as Dual Enoyl ACP Reductase and DHFR Enzyme Inhibitors

Autor: Mater H. Mahnashi, Pooja Koganole, Prem Kumar S. R., Sami S. Ashgar, Ibrahim Ahmed Shaikh, Shrinivas D. Joshi, Ali S. Alqahtani

Publikováno v: Antibiotics, Vol 12, Iss 4, p 763 (2023)

In this study, a new series of 4-(2,5-dimethyl-1H-pyrrol-1-yl)-N’-(2-(substituted)acetyl) benzohydrazides (5a–n) were prepared and new heterocycles underwent thorough characterization and evaluation for antibacterial activity; some of them underw

Externí odkaz: https://doaj.org/article/74418f7c57cb43bd80ab163b1730443c

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Akademický článek

In silico binding affinity studies of N-9 substituted 6-(4-(4-propoxyphenyl)piperazin-1-yl)-9H-purine derivatives-Target for P70-S6K1 & PI3K-δ kinases

Autor: Manjunath G. Sunagar, P. Aravind, Supreet Gaonkar, K.S. Devaraju, Shrinivas D. Joshi, Sheshagiri R. Dixit, B.M. Harish, Imtiyaz Ahmed M. Khazi

Publikováno v: Beni-Suef University Journal of Basic and Applied Sciences, Vol 7, Iss 1, Pp 84-91 (2018)

P70-S6K1 & PI3K-δ kinases are identified to be involved in many physiological processes associated with cancer, therefore many of the inhibitors being designed to target these kinases are in clinical trials. In the current study we have exploited th

Externí odkaz: https://doaj.org/article/007ebcee080b42878ea1f26b09aa4902

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Akademický článek

Functionalization of 3-chloroformylcoumarin to coumarin Schiff bases using reusable catalyst: an approach to molecular docking and biological studies

Autor: Suresh S. Kumbar, Kallappa M. Hosamani, Gangadhar C. Gouripur, Shrinivas D. Joshi

Publikováno v: Royal Society Open Science, Vol 5, Iss 5 (2018)

Recently, heterogeneous catalysts have been explored eximiously in the synthesis of heterocyclic compounds. Therefore, here we used solid-supported heterogeneous silica sulfuric acid as a catalyst for the synthesis of Schiff's base of 3-chloroformylc

Externí odkaz: https://doaj.org/article/7dbac89b06fa4080b03e0d0460ecef71

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Akademický článek

Multi-spectroscopic investigation of the binding interaction of fosfomycin with bovine serum albumin

Autor: Manjunath D. Meti, Sharanappa T. Nandibewoor, Shrinivas D. Joshi, Uttam A. More, Shivamurti A. Chimatadar

Publikováno v: Journal of Pharmaceutical Analysis, Vol 5, Iss 4, Pp 249-255 (2015)

The interaction between fosfomycin (FOS) and bovine serum albumin (BSA) has been investigated effectively by multi-spectroscopic techniques under physiological pH 7.4. FOS quenched the intrinsic fluorescence of BSA via static quenching. The number of

Externí odkaz: https://doaj.org/article/ed95592838434bd09f6b60e905370d66

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Akademický článek

New Urea Derivatives as Potential Antimicrobial Agents: Synthesis, Biological Evaluation, and Molecular Docking Studies

Autor: Mahadev Patil, Anurag Noonikara-Poyil, Shrinivas D. Joshi, Shivaputra A. Patil, Siddappa A. Patil, Alejandro Bugarin

Publikováno v: Antibiotics, Vol 8, Iss 4, p 178 (2019)

A series of new urea derivatives, containing aryl moieties as potential antimicrobial agents, were designed, synthesized, and characterized by 1H NMR, 13C NMR, FT-IR, and LCMS spectral techniques. All newly synthesized compounds were screened in vitr

Externí odkaz: https://doaj.org/article/25429dd1980e492d83a9bbf220377b36

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