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pro vyhledávání: '"S. Skala"'
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Publikováno v:
Journal of Minimally Invasive Gynecology. 28:S131
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::212fd542b1d9b6efc0d8b4a4e1b409fe
https://doi.org/10.1016/j.jmig.2021.09.231
https://doi.org/10.1016/j.jmig.2021.09.231
Autor:
L. L. Ong, J. D. Vasta, L. Monereau, G. Locke, H. Ribeiro, M. A. Pattoli, S. Skala, J. R. Burke, S. H. Watterson, J. A. Tino, P. L. Meisenheimer, B. Arey, J. Lippy, L. Zhang, M. B. Robers, A. Tebben, C. Chaudhry
Supplemental material, Supplementary_Material for A High-Throughput BRET Cellular Target Engagement Assay Links Biochemical to Cellular Activity for Bruton’s Tyrosine Kinase by L. L. Ong, J. D. Vasta, L. Monereau, G. Locke, H. Ribeiro, M. A. Pattol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::341fb039f56e93d190c5a5ea56022e64
Autor:
Loran M. Killar, S. Skala, James M. Chen, X. Du, G. Jin, Roy A. Black, A. Zask, Michele A. Sharr, Gu Yansong, R. Cowling, C.J March, J.S. Skotnicki, J. D. Albright, Amy Sung, Dauphine Barone, John F. DiJoseph, C. E. Roth, Kendall M. Mohler, Jeremy I. Levin, M. Hogan
Publikováno v:
Bioorganicmedicinal chemistry letters. 13(8)
Potent and selective bicyclic heteroaryl hydroxamic acid MMP and TACE inhibitors were synthesized by a novel convergent route. Selectivity and efficacy versus MMPs and TACE could be controlled by appropriate substitution on the scaffolds and by varia
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4826251a694d81522423585eb9f7e98
https://pubmed.ncbi.nlm.nih.gov/12668018
https://pubmed.ncbi.nlm.nih.gov/12668018
Autor:
Terri Cummons, X. Du, James M. Chen, Dauphine Barone, E. Delos Santos, Amy Sung, G. Jin, Jun Xu, R. Cowling, Jay D. Albright, Mila T. Du, R. Mulvey, Frances C. Nelson, S. Skala, Roy A. Black, J.S. Skotnicki, Jeremy I. Levin
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::359c750cebb10f7dfdca1ec34e96a6db
https://doi.org/10.1016/b978-0-08-044304-1.50138-6
https://doi.org/10.1016/b978-0-08-044304-1.50138-6
Publikováno v:
9th International Vacuum Microelectronics Conference.
Volcano emitters with gate dimensions of 6, 9, 15, 25, and 50 /spl mu/m have been processed using chemical mechanical polishing (CMP) for the removal of the emitter material and the gate-to-emitter dielectric on top of the gate plateau. Devices were
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ddcfbc9602e95e67255efab378503958
https://doi.org/10.1109/ivmc.1996.601848
https://doi.org/10.1109/ivmc.1996.601848
Autor:
R. Rao, J. Hubacek, R. Nowicki, W. Urbanek, G. Gammie, S. Skala, H. Busta, J.E. Pogemiller, D. Devine
Publikováno v:
Proceedings of International Electron Devices Meeting.
Individual and groups of 3/spl times/3 and 10/spl times/10 gated volcano-shaped field emitters have been processed with gate dimensions of 4, 8, 14, 25 and 50 /spl mu/m and gate-to-emitter rim distances of 1.0 and 0.25 /spl mu/m. The 0.25 /spl mu/m d
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ab913d88d0ee3cb685b3661e09be40c0
https://doi.org/10.1109/iedm.1995.499225
https://doi.org/10.1109/iedm.1995.499225
Autor:
R. Cowling, Amy Sung, C.J March, Jeremy I. Levin, Roy A. Black, G. Jin, Frances C. Nelson, S. Skala, Dauphine Barone, James M. Chen, Kendall M. Mohler, Loran M. Killar, Mila T. Du, J.S. Skotnicki
Publikováno v:
Bioorganicmedicinal chemistry letters. 12(8)
The SAR of a series of potent sulfonamide hydroxamate TACE inhibitors bearing novel acetylenic P1′ groups was explored. In particular, compound 4t bearing a butynyloxy P1′ moiety has excellent in vitro potency against isolated TACE enzyme and in
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1b841da89ea8fcc430f56a96972ec73c
https://pubmed.ncbi.nlm.nih.gov/11934588
https://pubmed.ncbi.nlm.nih.gov/11934588
Autor:
J.S. Skotnicki, Zhang-Bao Xu, T. Wehr, Mila T. Du, Roy A. Black, C. E. Roth, Li Di, James M. Chen, Jeremy I. Levin, Michele A. Sharr, C.J March, R. Cowling, John F. DiJoseph, S. Skala, Kendall M. Mohler, Amy Sung, Mary M. Sherman, Frances C. Nelson, Loran M. Killar, G. Jin
Publikováno v:
Bioorganicmedicinal chemistry letters. 11(22)
Anthranilic acid derivatives bearing basic amines were prepared and evaluated in vitro and in vivo as inhibitors of MMP-1, MMP-9, MMP-13, and TACE. Piperazine 4u has been identified as a potent, selective, orally active inhibitor of MMP-9 and MMP-13.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6d5e19bf3f666ee2e11c3aa0f30e660c
https://pubmed.ncbi.nlm.nih.gov/11677139
https://pubmed.ncbi.nlm.nih.gov/11677139
Autor:
A. Zask, John F. DiJoseph, S. Kincaid, Michele A. Sharr, R. Cowling, James K. Chen, Roy A. Black, T. Wehr, Frances C. Nelson, M. Hogan, A.M. Venkatesan, G. Jin, C. E. Roth, Mila T. Du, Jeremy I. Levin, J.S. Skotnicki, C.J March, Loran M. Killar, Amy Sung, Kendall M. Mohler, S. Skala
Publikováno v:
Bioorganicmedicinal chemistry letters. 11(16)
A novel series of anthranilic acid-based inhibitors of MMP-1, MMP-9, MMP-13, and TACE was prepared and evaluated. Selective inhibitors of MMP-9, MMP-13, and TACE were identified, including the potent, orally active MMP-13 inhibitor 4p.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::75b619b5fce7adf9d5f18c317a84810d
https://pubmed.ncbi.nlm.nih.gov/11514167
https://pubmed.ncbi.nlm.nih.gov/11514167