Zobrazeno 1 - 4
of 4
pro vyhledávání: '"S V, Schuster"'
Autor:
H. N. Bramson, Kenneth Batchelor, J. E. Long, Roger N. Hiner, Frank Lee, Marcia L. Moss, R. A. Jun. Mook, J. D. Stuart, J. Van Arnold, Stephen V. Frye, Stephanie L. Schweiker, Mary K. Grizzle, Curt D. Haffner, Michael K. James, Timothy K. Tippin, G. Tian, Patrick R. Maloney, S V Schuster, D. M. Bickett, Rayomand J. Unwalla, G. F. Jun. Dorsey
Publikováno v:
ChemInform. 25
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::c365d9b240d68257c530bd93326438d1
https://doi.org/10.1002/chin.199426234
https://doi.org/10.1002/chin.199426234
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 263(1)
Hemodynamic effects of GI 87084B, a novel ultra-short acting mu-opioid agonist, were studied in anesthetized dogs. In these studies, GI 87084B (0.3-20 nmol/kg/min i.v.) produced dose-dependent decreases in heart rate, arterial blood pressure, +dP/dt
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::050fd1f06d49f5e6f5e908fd5ee41e02
https://pubmed.ncbi.nlm.nih.gov/1403806
https://pubmed.ncbi.nlm.nih.gov/1403806
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 259(2)
GI 87084B (3-[4-methoxycarbonyl-4-[(1-oxopropyl) phenylamino]1-piperidine]propanoic acid, methyl ester, hydrochloride) was found to be a potent opioid agonist in the guinea pig ileum (EC50 = 2.4 +/- 0.6 nM), the rat vas deferens (EC50 = 387 +/- 44 nM
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::8db42cd1602391c459d79742fdf4290a
https://pubmed.ncbi.nlm.nih.gov/1658308
https://pubmed.ncbi.nlm.nih.gov/1658308
Autor:
A P Lahey, S V Schuster, Paul L. Feldman, Marcus F. Brackeen, H J Leighton, Michael K. James, Michael W. Lutz, M R Johnson, J M Bilotta
Publikováno v:
Journal of medicinal chemistry. 34(7)
In an effort to discover a potent ultrashort-acting mu opioid analgetic that is capable of metabolizing to an inactive species independent of hepatic function, several classes of 4-anilidopiperidine analgetics were synthesized and evaluated. One seri
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4485ede6c6c1b14551348d53eb1a5c48
https://pubmed.ncbi.nlm.nih.gov/2066993
https://pubmed.ncbi.nlm.nih.gov/2066993