Zobrazeno 1 - 10
of 26
pro vyhledávání: '"Rupesh L. Gawade"'
Autor:
Amol S. Kotmale, Rajesh G. Gonnade, Samir R. Shaikh, Tobias Stürzer, Rupesh L. Gawade, Deepak Kumar
Publikováno v:
Crystal Growth & Design. 19:5665-5678
A small library of ten sulfonamide derivatives comprising two aromatic rings was synthesized to investigate the effect of chronological positioning of the F-atom on the intramolecular π-stacking as...
Autor:
Kumar Vanka, Pranaya V. Joshi, Vedavati G. Puranik, Susanta Das, Pattuparambil R. Rajamohanan, Rupesh L. Gawade, Awais Ahmed, Rajesh G. Gonnade, Debamitra Chakravarty, Manoj V. Mane, Ekta Sangtani, Amol S. Kotmale
Publikováno v:
Crystal Growth & Design. 16:2416-2428
Understanding the process of prenucleation clustering at supersaturating stage is of significant importance to envisage the polymorphism in crystalline materials. Preferential formation of a thermodynamically stable crystal form suggests energeticall
Autor:
Kuruppanthara N. Vijayadas, K. N. Chaitanya, Rajesh G. Gonnade, Tukaram S. Ingole, Amol S. Kotmale, Gangadhar J. Sanjayan, P. R. Rajamohanan, Rupesh L. Gawade
Publikováno v:
European Journal of Organic Chemistry. 2016:1380-1388
Autor:
Gangadhar J. Sanjayan, Rajesh G. Gonnade, Pattuparambil R. Rajamohanan, Rupesh L. Gawade, Tukaram S. Ingole, Amol S. Kotmale
Publikováno v:
New Journal of Chemistry. 40:9205-9210
This paper describes the consequences of incorporating a constrained heterocyclic aromatic β-amino acid 3-aminothiophenecarboxylic acid (3-Atc) into peptides containing β-turn forming elements such as Pro-Gly motif and the effect on the secondary s
Autor:
Rupesh L. Gawade, Ekta Sangtani, Santosh C. Narwade, Rajesh G. Gonnade, Deepti D. Deobagkar, Vedavati G. Puranik, Debamitra Chakravarty, Joyashish Debgupta
Publikováno v:
RSC Advances. 6:5350-5358
Procainamide derivatives have been synthesized to investigate the role of side chains in modulating the DNA methylation level in cancer cells and gain insight into its mechanism of action. The synthesized derivatives comprised of flexible (dimethyl),
Autor:
Rajesh G. Gonnade, Ekta Sangtani, Parthapratim Munshi, Kunal Kumar Jha, Rupesh L. Gawade, Shridhar H. Thorat, Sanjay Kumar Sahu
Publikováno v:
Crystal Growth & Design. 15:5858-5872
Furosemide (FS), a loop diuretic drug commonly used for the treatment of hypertension and edema, exhibited color cocrystal polymorphism with coformer 4,4′-bipyridine (4BPY) in the stoichiometry 2:1, albeit both the API and the cocrystal former are
Autor:
Vedavati G. Puranik, Paramasivam Parthiban, Se-Kwon Kim, Someshwar D. Dindulkar, Dong Hyun Anh, Rupesh L. Gawade, Yeon Tae Jeong, Ira Bhatnagar
Publikováno v:
Journal of Chemical Sciences. 126:861-873
A series of fifteen diversified N-benzylpiperidin-4-one oximes were synthesized and characterized by their NMR spectral data. Additionally, single-crystal XRD analysis was performed for the representative symmetrically and unsymmetrically substituted
Autor:
Rajesh G. Gonnade, Veera V. E. Ramesh, Vijaykumar H. Thorat, Pattuparambil R. Rajamohanan, Roshna V. Nair, Tukaram S. Ingole, Kuruppanthara N. Vijayadas, Hilda C. Davis, Gangadhar J. Sanjayan, Panchami Prabhakaran, Rupesh L. Gawade, Sangram S. Kale, Vedavati G. Puranik
Publikováno v:
European Journal of Organic Chemistry. 2013:3529-3542
This article details the characteristic conformational features of the Ant-Pro reverse turn ― a folded pseudo β-turn motif that displays a closed nine-membered-ring hydrogen-bonded network involving just two amino acid residues, namely anthranilic
Autor:
Aadil A. Momin, Radhika S. Kusurkar, Vedavati G. Puranik, Rupesh L. Gawade, Shrikar M. Bhosale
Publikováno v:
Tetrahedron Letters. 53:5327-5330
An efficient method has been established for the preparation of 1,2-diketones by unexpected C–C bond cleavage in 4-keto-2-hydroxy esters using pyridiniumchlorochromate (PCC).
Publikováno v:
Tetrahedron Letters. 53:2647-2650
The formal synthesis of (−)-stemoamide was achieved starting from l -pyroglutamic acid. The key steps used are the allylation using BF3·OEt2, ring closing metathesis, allylic oxidation and a novel epimerization at C8.