Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Rosamaria Micheletti"'
Autor:
Rosamaria Micheletti, Myrna Gil Quintero, Luciano Maiocchi, Ettore Giraldo, Marco Turconi, Massimo Nicola, Arturo Donetti
Publikováno v:
ChemInform. 22
A series of 2,3-dihydro-2-oxo-1H-benzimidazole-1-carboxylic acid esters and amides containing a basic azacyclo- or azabicycloalkyl moiety has been synthesized and evaluated for 5-HT3 antagonistic activity in a radioligand binding assay ([3H]ICS 20593
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::15131cae1d7d1dbb7344df4c681a5fd0
https://doi.org/10.1002/chin.199104210
https://doi.org/10.1002/chin.199104210
Autor:
Rosamaria Micheletti, Massimo Nicola, Marco Turconi, Ettore Giraldo, Myrna Gil Quintero, Arturo Donetti, Luciano Maiocchi
Publikováno v:
Journal of Medicinal Chemistry. 33:2101-2108
A series of 2,3-dihydro-2-oxo-1H-benzimidazole-1-carboxylic acid esters and amides containing a basic azacyclo- or azabicycloalkyl moiety has been synthesized and evaluated for 5-HT3 antagonistic activity in a radioligand binding assay ([3H]ICS 20593
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::17ba3e9201f711ee5396c6fed5aeea60
https://doi.org/10.1021/jm00170a009
https://doi.org/10.1021/jm00170a009
Autor:
Aalt Bast, Giuseppe Bietti, Hendrik Timmerman, Arturo Donetti, E. Cereda, Antonio Giachetti, Rosamaria Micheletti
Publikováno v:
European Journal of Medicinal Chemistry. 23:267-273
Studies on protonation of the amidino group present in mifentidine have shown that this H2-receptor antagonist exists predominantly as a formamidinium monocation (95.3%) at physiological pH. Further studies on the preferred conformation by quantum me
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::274ed1c35c75364d5bce7280b8981bca
https://doi.org/10.1016/0223-5234(88)90009-8
https://doi.org/10.1016/0223-5234(88)90009-8
Autor:
E. Cereda, P. Vanoni, C. Bazzano, Arturo Donetti, Antonio Giachetti, A. Gallazzi, Rosamaria Micheletti, E. Bellora, P. Del Soldato, Ferdinando Pagani
Publikováno v:
Chemischer Informationsdienst. 15
Structure-activity considerations of N alpha-guanylhistamine, the first compound found with detectable H2-antagonist activity, led to the synthesis of a series of conformationally rigid guanylhistamine analogues, namely, (imidazolylphenyl)guanidines,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::76000529c6a13a1d507b2747adcf8dba
https://doi.org/10.1002/chin.198432198
https://doi.org/10.1002/chin.198432198
Autor:
C. Bazzano, Arturo Donetti, Ferdinando Pagani, A. Gallazzi, E. Cereda, Antonio Giachetti, Rosamaria Micheletti, P. Vanoni, P. Del Soldato, E. Bellora
Publikováno v:
Journal of medicinal chemistry. 27(3)
Structure-activity considerations of N alpha-guanylhistamine, the first compound found with detectable H2-antagonist activity, led to the synthesis of a series of conformationally rigid guanylhistamine analogues, namely, (imidazolylphenyl)guanidines,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b40497d52ef0ad6cf19d457c4a295703
https://pubmed.ncbi.nlm.nih.gov/6142117
https://pubmed.ncbi.nlm.nih.gov/6142117