Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Ronald Suayan"'
Autor:
Richard Hernandez, Girija Krishnamurthy, Frank Loganzo, Arie Zask, Ayako Yamashita, Gary Harold Birnberg, Lee M. Greenberger, Zhilian Tang, Sylvia Musto, Tami Annable, Derek C. Cole, Xiaoran Yang, Robert Williamson, Semiramis Ayral-Kaloustian, Gulnaz Khafizova, Carolyn Discafani, Emily B. Norton, Katherine Cheung, Chuan Niu, Ronald Suayan, Joshua Kaplan, Carl Beyer
Publikováno v:
Journal of Medicinal Chemistry. 47:4774-4786
Hemiasterlin (1), a tripeptide isolated from marine sponges, induces microtubule depolymerization and mitotic arrest in cells. HTI-286 (2), an analogue from an initial study of the hemiasterlins, is presently in clinical trials. In addition to its po
Autor:
Arie, Zask, Gary, Birnberg, Katherine, Cheung, Joshua, Kaplan, Chuan, Niu, Emily, Norton, Ronald, Suayan, Ayako, Yamashita, Derek, Cole, Zhilian, Tang, Girija, Krishnamurthy, Robert, Williamson, Gulnaz, Khafizova, Sylvia, Musto, Richard, Hernandez, Tami, Annable, Xiaoran, Yang, Carolyn, Discafani, Carl, Beyer, Lee M, Greenberger, Frank, Loganzo, Semiramis, Ayral-Kaloustian
Publikováno v:
Journal of medicinal chemistry. 47(19)
Hemiasterlin, a tripeptide isolated from marine sponges, induces microtubule depolymerization and mitotic arrest in cells. HTI-286, an analogue from an initial study of the hemiasterlins, is presently in clinical trials. In addition to its potent ant